gabapentin-3472 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

195 genes differentially expressed following the gabapentin-3472 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
A4GALT alpha 1,4-galactosyltransferase
ABCB9 ATP-binding cassette, sub-family B (MDR/TAP), member 9
ADAP2 ArfGAP with dual PH domains 2
AHCYL1 adenosylhomocysteinase-like 1
ANXA2P3 annexin A2 pseudogene 3
APAF1 apoptotic peptidase activating factor 1
APPBP2 amyloid beta precursor protein (cytoplasmic tail) binding protein 2
ARAP1 ArfGAP with RhoGAP domain, ankyrin repeat and PH domain 1
ARHGEF4 Rho guanine nucleotide exchange factor (GEF) 4
ARPIN actin-related protein 2/3 complex inhibitor
ATM ATM serine/threonine kinase
ATXN7L3B ataxin 7-like 3B
AUTS2 autism susceptibility candidate 2
C1QTNF3 C1q and tumor necrosis factor related protein 3
CALCOCO1 calcium binding and coiled-coil domain 1
CALM1 calmodulin 1 (phosphorylase kinase, delta)
CAMK2G calcium/calmodulin-dependent protein kinase II gamma
CASP2 caspase 2, apoptosis-related cysteine peptidase
CCDC186 coiled-coil domain containing 186
CFLAR CASP8 and FADD-like apoptosis regulator
CKMT2 creatine kinase, mitochondrial 2 (sarcomeric)
CLN8 ceroid-lipofuscinosis, neuronal 8 (epilepsy, progressive with mental retardation)
COL1A1 collagen, type I, alpha 1
DAPP1 dual adaptor of phosphotyrosine and 3-phosphoinositides
DDR1-AS1 DDR1 antisense RNA 1 (head to head)
DFFB DNA fragmentation factor, 40kDa, beta polypeptide (caspase-activated DNase)
DPYS dihydropyrimidinase
DSC3 desmocollin 3
EGFR epidermal growth factor receptor
ELP6 elongator acetyltransferase complex subunit 6
ENTPD4 ectonucleoside triphosphate diphosphohydrolase 4
EPOR erythropoietin receptor
ETAA1 Ewing tumor-associated antigen 1
FOXG1 forkhead box G1
FSCN1 fascin actin-bundling protein 1
FUT4 fucosyltransferase 4 (alpha (1,3) fucosyltransferase, myeloid-specific)
GINS4 GINS complex subunit 4 (Sld5 homolog)
GNL3L guanine nucleotide binding protein-like 3 (nucleolar)-like
GPR153 G protein-coupled receptor 153
GUSBP3 glucuronidase, beta pseudogene 3
HERC3 HECT and RLD domain containing E3 ubiquitin protein ligase 3
HFE hemochromatosis
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
IGFBP5 insulin-like growth factor binding protein 5
IL6ST interleukin 6 signal transducer
IQCC IQ motif containing C
KAZN kazrin, periplakin interacting protein
KLHL25 kelch-like family member 25
LMO4 LIM domain only 4
LRCH1 leucine-rich repeats and calponin homology (CH) domain containing 1
LRRC37A3 leucine rich repeat containing 37, member A3
MED18 mediator complex subunit 18
METTL7A methyltransferase like 7A
MLLT10 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 10
MYCL v-myc avian myelocytomatosis viral oncogene lung carcinoma derived homolog
MZT2B mitotic spindle organizing protein 2B
NCOA2 nuclear receptor coactivator 2
NEDD9 neural precursor cell expressed, developmentally down-regulated 9
NFIB nuclear factor I/B
NGLY1 N-glycanase 1
NOL12 nucleolar protein 12
PAX5 paired box 5
PCDHGB5 protocadherin gamma subfamily B, 5
PGF placental growth factor
PPIA peptidylprolyl isomerase A (cyclophilin A)
PSMB2 proteasome (prosome, macropain) subunit, beta type, 2
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RABGAP1 RAB GTPase activating protein 1
REEP1 receptor accessory protein 1
RETN resistin
RNF31 ring finger protein 31
SMARCD3 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 3
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SNAPC3 small nuclear RNA activating complex, polypeptide 3, 50kDa
SPATA2L spermatogenesis associated 2-like
SPINK5 serine peptidase inhibitor, Kazal type 5
SPTAN1 spectrin, alpha, non-erythrocytic 1
SRCAP Snf2-related CREBBP activator protein
ST3GAL2 ST3 beta-galactoside alpha-2,3-sialyltransferase 2
STARD3 StAR-related lipid transfer (START) domain containing 3
TNFRSF11B tumor necrosis factor receptor superfamily, member 11b
TREX1 three prime repair exonuclease 1
TTLL5 tubulin tyrosine ligase-like family member 5
UBE3A ubiquitin protein ligase E3A
UPP1 uridine phosphorylase 1
USP36 ubiquitin specific peptidase 36
VPS13B vacuolar protein sorting 13 homolog B (yeast)
WDR76 WD repeat domain 76
WFDC2 WAP four-disulfide core domain 2
WIPF1 WAS/WASL interacting protein family, member 1
XRCC2 X-ray repair complementing defective repair in Chinese hamster cells 2
ZBTB43 zinc finger and BTB domain containing 43
ZBTB7A zinc finger and BTB domain containing 7A
ZFP36L2 ZFP36 ring finger protein-like 2
ZMYND8 zinc finger, MYND-type containing 8
ZNF117 zinc finger protein 117
ZNF451 zinc finger protein 451
ZNF652 zinc finger protein 652

decreased expression

Symbol Name
ACTL8 actin-like 8
AGPAT3 1-acylglycerol-3-phosphate O-acyltransferase 3
ARSB arylsulfatase B
ASAP1-IT1 ASAP1 intronic transcript 1
ASTE1 asteroid homolog 1 (Drosophila)
BEX4 brain expressed, X-linked 4
BGLAP bone gamma-carboxyglutamate (gla) protein
BRAF B-Raf proto-oncogene, serine/threonine kinase
C11ORF80 chromosome 11 open reading frame 80
C1ORF216 chromosome 1 open reading frame 216
C1ORF35 chromosome 1 open reading frame 35
C2ORF54 chromosome 2 open reading frame 54
CABYR calcium binding tyrosine-(Y)-phosphorylation regulated
CAPG capping protein (actin filament), gelsolin-like
CCP110 centriolar coiled coil protein 110kDa
CDK3 cyclin-dependent kinase 3
CEMIP cell migration inducing protein, hyaluronan binding
CERK ceramide kinase
CHST7 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 7
CLN6 ceroid-lipofuscinosis, neuronal 6, late infantile, variant
CNGB3 cyclic nucleotide gated channel beta 3
CST6 cystatin E/M
DCP1A decapping mRNA 1A
DHX35 DEAH (Asp-Glu-Ala-His) box polypeptide 35
DUSP5 dual specificity phosphatase 5
DZANK1 double zinc ribbon and ankyrin repeat domains 1
EDAR ectodysplasin A receptor
ENTPD7 ectonucleoside triphosphate diphosphohydrolase 7
EYA2 EYA transcriptional coactivator and phosphatase 2
FAM198B family with sequence similarity 198, member B
FBXL15 F-box and leucine-rich repeat protein 15
GBP2 guanylate binding protein 2, interferon-inducible
GDAP2 ganglioside induced differentiation associated protein 2
GLTSCR1 glioma tumor suppressor candidate region gene 1
GTF3C5 general transcription factor IIIC, polypeptide 5, 63kDa
HIST1H2AJ histone cluster 1, H2aj
HIST1H3B histone cluster 1, H3b
IGBP1 immunoglobulin (CD79A) binding protein 1
IL15RA interleukin 15 receptor, alpha
IQCE IQ motif containing E
ISG20 interferon stimulated exonuclease gene 20kDa
KCNK12 potassium channel, two pore domain subfamily K, member 12
KLK5 kallikrein-related peptidase 5
LYPLA2P1 lysophospholipase II pseudogene 1
LZTS3 leucine zipper, putative tumor suppressor family member 3
MCM3 minichromosome maintenance complex component 3
METTL16 methyltransferase like 16
MFAP2 microfibrillar-associated protein 2
MMACHC methylmalonic aciduria (cobalamin deficiency) cblC type, with homocystinuria
MMP9 matrix metallopeptidase 9
MRPL52 mitochondrial ribosomal protein L52
MTG1 mitochondrial ribosome-associated GTPase 1
NDEL1 nudE neurodevelopment protein 1-like 1
NEK11 NIMA-related kinase 11
NOL6 nucleolar protein 6 (RNA-associated)
NPFFR1 neuropeptide FF receptor 1
NPM3 nucleophosmin/nucleoplasmin 3
NR1H3 nuclear receptor subfamily 1, group H, member 3
PIGL phosphatidylinositol glycan anchor biosynthesis, class L
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
PMCH pro-melanin-concentrating hormone
PPT2 palmitoyl-protein thioesterase 2
PRRG2 proline rich Gla (G-carboxyglutamic acid) 2
RAD51AP1 RAD51 associated protein 1
RBM23 RNA binding motif protein 23
RHPN1-AS1 RHPN1 antisense RNA 1 (head to head)
RNH1 ribonuclease/angiogenin inhibitor 1
ROM1 retinal outer segment membrane protein 1
RPGR retinitis pigmentosa GTPase regulator
SCPEP1 serine carboxypeptidase 1
SEMA4A sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4A
SERPINF1 serpin peptidase inhibitor, clade F (alpha-2 antiplasmin, pigment epithelium derived factor), member 1
SKA1 spindle and kinetochore associated complex subunit 1
SLC12A5 solute carrier family 12 (potassium/chloride transporter), member 5
SLC12A8 solute carrier family 12, member 8
SLC22A5 solute carrier family 22 (organic cation/carnitine transporter), member 5
SLC25A15 solute carrier family 25 (mitochondrial carrier; ornithine transporter) member 15
SLC46A3 solute carrier family 46, member 3
SLC9A1 solute carrier family 9, subfamily A (NHE1, cation proton antiporter 1), member 1
SPINK4 serine peptidase inhibitor, Kazal type 4
ST6GALNAC2 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 2
STAG3L4 stromal antigen 3-like 4 (pseudogene)
SYT17 synaptotagmin XVII
TBC1D17 TBC1 domain family, member 17
TINF2 TERF1 (TRF1)-interacting nuclear factor 2
TNS2 tensin 2
TRABD TraB domain containing
TRPV1 transient receptor potential cation channel, subfamily V, member 1
TSPYL2 TSPY-like 2
TUBA3C tubulin, alpha 3c
TUBA3D tubulin, alpha 3d
XAB2 XPA binding protein 2
ZC3H3 zinc finger CCCH-type containing 3
ZNF586 zinc finger protein 586
ZNF74 zinc finger protein 74
ZNF747 zinc finger protein 747
ZNF770 zinc finger protein 770