geldanamycin-1066 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

200 genes differentially expressed following the geldanamycin-1066 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABHD4 abhydrolase domain containing 4
AKAP17A A kinase (PRKA) anchor protein 17A
ALOX12P2 arachidonate 12-lipoxygenase pseudogene 2
ARFGAP3 ADP-ribosylation factor GTPase activating protein 3
ARG2 arginase 2
ARMCX1 armadillo repeat containing, X-linked 1
ARMCX3 armadillo repeat containing, X-linked 3
ASNS asparagine synthetase (glutamine-hydrolyzing)
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
BAG2 BCL2-associated athanogene 2
BAG3 BCL2-associated athanogene 3
BET1 Bet1 golgi vesicular membrane trafficking protein
BTN2A2 butyrophilin, subfamily 2, member A2
CALR calreticulin
CAP2 CAP, adenylate cyclase-associated protein, 2 (yeast)
CCNG2 cyclin G2
CDC6 cell division cycle 6
CDK2AP2 cyclin-dependent kinase 2 associated protein 2
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
CLK4 CDC-like kinase 4
CREB3L2 cAMP responsive element binding protein 3-like 2
CRELD2 cysteine-rich with EGF-like domains 2
CSRP2 cysteine and glycine-rich protein 2
CTH cystathionine gamma-lyase
DDIT3 DNA-damage-inducible transcript 3
DDIT4 DNA-damage-inducible transcript 4
DHRS2 dehydrogenase/reductase (SDR family) member 2
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJB9 DnaJ (Hsp40) homolog, subfamily B, member 9
DNAJC12 DnaJ (Hsp40) homolog, subfamily C, member 12
DNAJC3 DnaJ (Hsp40) homolog, subfamily C, member 3
EAF2 ELL associated factor 2
FGFR2 fibroblast growth factor receptor 2
FKBP11 FK506 binding protein 11, 19 kDa
FKBP14 FK506 binding protein 14, 22 kDa
FNDC3A fibronectin type III domain containing 3A
FNDC3B fibronectin type III domain containing 3B
GFPT1 glutamine--fructose-6-phosphate transaminase 1
GLRX glutaredoxin (thioltransferase)
GTF3C3 general transcription factor IIIC, polypeptide 3, 102kDa
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HMGCR 3-hydroxy-3-methylglutaryl-CoA reductase
HMOX1 heme oxygenase 1
HNRNPD heterogeneous nuclear ribonucleoprotein D (AU-rich element RNA binding protein 1, 37kDa)
HSD17B7 hydroxysteroid (17-beta) dehydrogenase 7
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1
HSPA13 heat shock protein 70kDa family, member 13
HSPA1A heat shock 70kDa protein 1A
HSPA4L heat shock 70kDa protein 4-like
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPH1 heat shock 105kDa/110kDa protein 1
HTATIP2 HIV-1 Tat interactive protein 2, 30kDa
HYOU1 hypoxia up-regulated 1
LDLR low density lipoprotein receptor
LPIN1 lipin 1
LZTFL1 leucine zipper transcription factor-like 1
MANF mesencephalic astrocyte-derived neurotrophic factor
MBNL2 muscleblind-like splicing regulator 2
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11
MT1F metallothionein 1F
MYDGF myeloid-derived growth factor
NUCB2 nucleobindin 2
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PDIA4 protein disulfide isomerase family A, member 4
PEX26 peroxisomal biogenesis factor 26
PPID peptidylprolyl isomerase D
PRRC1 proline-rich coiled-coil 1
PRSS16 protease, serine, 16 (thymus)
RHOQ ras homolog family member Q
RNASE4 ribonuclease, RNase A family, 4
RRBP1 ribosome binding protein 1
RSRC2 arginine/serine-rich coiled-coil 2
SDF2L1 stromal cell-derived factor 2-like 1
SEC24D SEC24 family member D
SEL1L sel-1 suppressor of lin-12-like (C. elegans)
SERP1 stress-associated endoplasmic reticulum protein 1
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SETX senataxin
SH3BGR SH3 domain binding glutamate-rich protein
SLC1A4 solute carrier family 1 (glutamate/neutral amino acid transporter), member 4
SLC7A1 solute carrier family 7 (cationic amino acid transporter, y+ system), member 1
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMCO4 single-pass membrane protein with coiled-coil domains 4
SMEK2 SMEK homolog 2, suppressor of mek1 (Dictyostelium)
SNAP23 synaptosomal-associated protein, 23kDa
TES testin LIM domain protein
TMEM41B transmembrane protein 41B
TMEM50B transmembrane protein 50B
TRIM2 tripartite motif containing 2
TSPYL2 TSPY-like 2
TUBA4A tubulin, alpha 4a
ULBP2 UL16 binding protein 2
WFS1 Wolfram syndrome 1 (wolframin)
WIPI1 WD repeat domain, phosphoinositide interacting 1
ZMYND8 zinc finger, MYND-type containing 8
ZNF165 zinc finger protein 165
ZNF227 zinc finger protein 227

decreased expression

Symbol Name
ACKR3 atypical chemokine receptor 3
ALG6 ALG6, alpha-1,3-glucosyltransferase
ANKEF1 ankyrin repeat and EF-hand domain containing 1
ANKRD36B ankyrin repeat domain 36B
APPL1 adaptor protein, phosphotyrosine interaction, PH domain and leucine zipper containing 1
BAMBI BMP and activin membrane-bound inhibitor
BAZ1A bromodomain adjacent to zinc finger domain, 1A
BTBD3 BTB (POZ) domain containing 3
C9ORF3 chromosome 9 open reading frame 3
CCNE1 cyclin E1
CD3EAP CD3e molecule, epsilon associated protein
CDIPT CDP-diacylglycerol--inositol 3-phosphatidyltransferase
CNNM3 cyclin and CBS domain divalent metal cation transport mediator 3
CPTP ceramide-1-phosphate transfer protein
CSTF3 cleavage stimulation factor, 3' pre-RNA, subunit 3, 77kDa
DBR1 debranching RNA lariats 1
DIP2A DIP2 disco-interacting protein 2 homolog A (Drosophila)
DNA2 DNA replication helicase/nuclease 2
DNAJC22 DnaJ (Hsp40) homolog, subfamily C, member 22
E2F8 E2F transcription factor 8
EGR3 early growth response 3
ERF Ets2 repressor factor
ESRP2 epithelial splicing regulatory protein 2
FAM188A family with sequence similarity 188, member A
FAM86B1 family with sequence similarity 86, member B1
FANCL Fanconi anemia, complementation group L
FASTKD1 FAST kinase domains 1
FCHSD2 FCH and double SH3 domains 2
GPRC5C G protein-coupled receptor, class C, group 5, member C
HYAL2 hyaluronoglucosaminidase 2
ID1 inhibitor of DNA binding 1, dominant negative helix-loop-helix protein
IER2 immediate early response 2
IRX5 iroquois homeobox 5
KATNBL1 katanin p80 subunit B-like 1
KIAA0922 KIAA0922
KLF10 Kruppel-like factor 10
KRCC1 lysine-rich coiled-coil 1
LAMA5 laminin, alpha 5
LIAS lipoic acid synthetase
LRFN4 leucine rich repeat and fibronectin type III domain containing 4
MANSC1 MANSC domain containing 1
MAP3K11 mitogen-activated protein kinase kinase kinase 11
MAP3K3 mitogen-activated protein kinase kinase kinase 3
MEX3C mex-3 RNA binding family member C
MKNK1 MAP kinase interacting serine/threonine kinase 1
MTERF3 mitochondrial transcription termination factor 3
MYC v-myc avian myelocytomatosis viral oncogene homolog
NACC2 NACC family member 2, BEN and BTB (POZ) domain containing
NEIL3 nei endonuclease VIII-like 3 (E. coli)
NEO1 neogenin 1
NFKBIA nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, alpha
NR1H3 nuclear receptor subfamily 1, group H, member 3
NRIP1 nuclear receptor interacting protein 1
PCF11 PCF11 cleavage and polyadenylation factor subunit
PLK2 polo-like kinase 2
PMS1 PMS1 postmeiotic segregation increased 1 (S. cerevisiae)
POLE2 polymerase (DNA directed), epsilon 2, accessory subunit
PRKCD protein kinase C, delta
RBM14 RNA binding motif protein 14
RBM4B RNA binding motif protein 4B
RDH14 retinol dehydrogenase 14 (all-trans/9-cis/11-cis)
RGL2 ral guanine nucleotide dissociation stimulator-like 2
RGS16 regulator of G-protein signaling 16
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RIPK4 receptor-interacting serine-threonine kinase 4
RPP25 ribonuclease P/MRP 25kDa subunit
RRS1 RRS1 ribosome biogenesis regulator homolog (S. cerevisiae)
SACS sacsin molecular chaperone
SALL2 spalt-like transcription factor 2
SCO2 SCO2 cytochrome c oxidase assembly protein
SEMA4C sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4C
SETD6 SET domain containing 6
SETMAR SET domain and mariner transposase fusion gene
SH2B2 SH2B adaptor protein 2
SHPK sedoheptulokinase
SIGIRR single immunoglobulin and toll-interleukin 1 receptor (TIR) domain
SLC16A6 solute carrier family 16, member 6
SLC25A20 solute carrier family 25 (carnitine/acylcarnitine translocase), member 20
SLC25A28 solute carrier family 25 (mitochondrial iron transporter), member 28
SLC37A1 solute carrier family 37 (glucose-6-phosphate transporter), member 1
SMAD7 SMAD family member 7
SMAGP small cell adhesion glycoprotein
SMARCAL1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a-like 1
SP140L SP140 nuclear body protein-like
SPAG1 sperm associated antigen 1
SPATA2L spermatogenesis associated 2-like
ST3GAL1 ST3 beta-galactoside alpha-2,3-sialyltransferase 1
TBC1D31 TBC1 domain family, member 31
TDRD7 tudor domain containing 7
TERF2 telomeric repeat binding factor 2
TFRC transferrin receptor
TOE1 target of EGR1, member 1 (nuclear)
TRAPPC12 trafficking protein particle complex 12
URM1 ubiquitin related modifier 1
VPS54 vacuolar protein sorting 54 homolog (S. cerevisiae)
ZCCHC6 zinc finger, CCHC domain containing 6
ZFP36 ZFP36 ring finger protein
ZNF672 zinc finger protein 672
ZNF787 zinc finger protein 787
ZXDC ZXD family zinc finger C