glimepiride-2809 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the glimepiride-2809 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABI2 abl-interactor 2
APOE apolipoprotein E
ARHGEF4 Rho guanine nucleotide exchange factor (GEF) 4
ARL4D ADP-ribosylation factor-like 4D
ATP2A3 ATPase, Ca++ transporting, ubiquitous
ATP6AP2 ATPase, H+ transporting, lysosomal accessory protein 2
BPIFA1 BPI fold containing family A, member 1
CA9 carbonic anhydrase IX
CABIN1 calcineurin binding protein 1
CAMK4 calcium/calmodulin-dependent protein kinase IV
CAMSAP1 calmodulin regulated spectrin-associated protein 1
CC2D1A coiled-coil and C2 domain containing 1A
CD82 CD82 molecule
CDH15 cadherin 15, type 1, M-cadherin (myotubule)
CDH8 cadherin 8, type 2
CDRT1 CMT1A duplicated region transcript 1
CNPY4 canopy FGF signaling regulator 4
COL16A1 collagen, type XVI, alpha 1
CSNK1E casein kinase 1, epsilon
CTSZ cathepsin Z
DAAM2 dishevelled associated activator of morphogenesis 2
DIO2 deiodinase, iodothyronine, type II
DLK2 delta-like 2 homolog (Drosophila)
DSTYK dual serine/threonine and tyrosine protein kinase
DUSP1 dual specificity phosphatase 1
DVL2 dishevelled segment polarity protein 2
DYRK1A dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A
EDA ectodysplasin A
ELL2 elongation factor, RNA polymerase II, 2
EPHB2 EPH receptor B2
EVPL envoplakin
FCGRT Fc fragment of IgG, receptor, transporter, alpha
FFAR2 free fatty acid receptor 2
FN1 fibronectin 1
FOS FBJ murine osteosarcoma viral oncogene homolog
GMPR guanosine monophosphate reductase
GNA14 guanine nucleotide binding protein (G protein), alpha 14
GSK3A glycogen synthase kinase 3 alpha
GZMK granzyme K (granzyme 3; tryptase II)
HGF hepatocyte growth factor (hepapoietin A; scatter factor)
HLA-DRA major histocompatibility complex, class II, DR alpha
HSF2BP heat shock transcription factor 2 binding protein
IL27RA interleukin 27 receptor, alpha
ITGA10 integrin, alpha 10
ITGA3 integrin, alpha 3 (antigen CD49C, alpha 3 subunit of VLA-3 receptor)
KCNN1 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 1
KDM5C lysine (K)-specific demethylase 5C
KLHL22 kelch-like family member 22
LIME1 Lck interacting transmembrane adaptor 1
LOXL3 lysyl oxidase-like 3
LPPR2 lipid phosphate phosphatase-related protein type 2
MAP2K7 mitogen-activated protein kinase kinase 7
MAPK8IP1 mitogen-activated protein kinase 8 interacting protein 1
MBNL2 muscleblind-like splicing regulator 2
MCM3AP minichromosome maintenance complex component 3 associated protein
MTA2 metastasis associated 1 family, member 2
MYL10 myosin, light chain 10, regulatory
MYOF myoferlin
NCR3 natural cytotoxicity triggering receptor 3
NDST1 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 1
ONECUT2 one cut homeobox 2
PDZD2 PDZ domain containing 2
PGLYRP4 peptidoglycan recognition protein 4
PLCD1 phospholipase C, delta 1
PLTP phospholipid transfer protein
PPP2R5B protein phosphatase 2, regulatory subunit B', beta
PPP5C protein phosphatase 5, catalytic subunit
PTCH2 patched 2
PTGIS prostaglandin I2 (prostacyclin) synthase
PVRL1 poliovirus receptor-related 1 (herpesvirus entry mediator C)
RPH3A rabphilin 3A
RPS6KA6 ribosomal protein S6 kinase, 90kDa, polypeptide 6
SAG S-antigen; retina and pineal gland (arrestin)
SECTM1 secreted and transmembrane 1
SEMA3B sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3B
SFTPB surfactant protein B
SGCD sarcoglycan, delta (35kDa dystrophin-associated glycoprotein)
SLC16A5 solute carrier family 16 (monocarboxylate transporter), member 5
SLC30A3 solute carrier family 30 (zinc transporter), member 3
SLC48A1 solute carrier family 48 (heme transporter), member 1
SLC52A1 solute carrier family 52 (riboflavin transporter), member 1
SMARCA1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 1
ST5 suppression of tumorigenicity 5
STX2 syntaxin 2
SULT4A1 sulfotransferase family 4A, member 1
SYNDIG1 synapse differentiation inducing 1
TG thyroglobulin
TLN2 talin 2
TNKS tankyrase, TRF1-interacting ankyrin-related ADP-ribose polymerase
TRBC1 T cell receptor beta constant 1
TTC38 tetratricopeptide repeat domain 38
UBE3A ubiquitin protein ligase E3A
UBXN6 UBX domain protein 6
VWA5A von Willebrand factor A domain containing 5A
WIZ widely interspaced zinc finger motifs
ZC3H7B zinc finger CCCH-type containing 7B
ZFP64 ZFP64 zinc finger protein
ZNF76 zinc finger protein 76

decreased expression

Symbol Name
ADCK3 aarF domain containing kinase 3
ADCY7 adenylate cyclase 7
ANXA1 annexin A1
BCL11B B-cell CLL/lymphoma 11B (zinc finger protein)
BCORL1 BCL6 corepressor-like 1
C1ORF106 chromosome 1 open reading frame 106
C1ORF159 chromosome 1 open reading frame 159
C7ORF43 chromosome 7 open reading frame 43
CCBL1 cysteine conjugate-beta lyase, cytoplasmic
CCDC85C coiled-coil domain containing 85C
CDK20 cyclin-dependent kinase 20
CDK3 cyclin-dependent kinase 3
CEMIP cell migration inducing protein, hyaluronan binding
CEP170B centrosomal protein 170B
COPZ2 coatomer protein complex, subunit zeta 2
CUEDC1 CUE domain containing 1
CYP20A1 cytochrome P450, family 20, subfamily A, polypeptide 1
DBF4B DBF4 zinc finger B
DGAT1 diacylglycerol O-acyltransferase 1
EGR3 early growth response 3
FAM53B family with sequence similarity 53, member B
FOXC1 forkhead box C1
GPR87 G protein-coupled receptor 87
H2AFY2 H2A histone family, member Y2
HIRA histone cell cycle regulator
HIST1H3E histone cluster 1, H3e
HIST1H4F histone cluster 1, H4f
IL15RA interleukin 15 receptor, alpha
IQCG IQ motif containing G
KCNK12 potassium channel, two pore domain subfamily K, member 12
LY6D lymphocyte antigen 6 complex, locus D
LYPD1 LY6/PLAUR domain containing 1
LYPD3 LY6/PLAUR domain containing 3
LYPLA2P1 lysophospholipase II pseudogene 1
LZTR1 leucine-zipper-like transcription regulator 1
MAST3 microtubule associated serine/threonine kinase 3
MMP15 matrix metallopeptidase 15 (membrane-inserted)
MOSPD3 motile sperm domain containing 3
MTCL1 microtubule crosslinking factor 1
MUL1 mitochondrial E3 ubiquitin protein ligase 1
MYH9 myosin, heavy chain 9, non-muscle
NAV2 neuron navigator 2
NEAT1 nuclear paraspeckle assembly transcript 1 (non-protein coding)
NHLRC2 NHL repeat containing 2
NPY1R neuropeptide Y receptor Y1
NPY5R neuropeptide Y receptor Y5
NSMF NMDA receptor synaptonuclear signaling and neuronal migration factor
NT5E 5'-nucleotidase, ecto (CD73)
NXPE3 neurexophilin and PC-esterase domain family, member 3
OLFML3 olfactomedin-like 3
P3H4 prolyl 3-hydroxylase family member 4 (non-enzymatic)
PARP12 poly (ADP-ribose) polymerase family, member 12
PARP16 poly (ADP-ribose) polymerase family, member 16
PCBP4 poly(rC) binding protein 4
PCSK7 proprotein convertase subtilisin/kexin type 7
PDZRN3 PDZ domain containing ring finger 3
PEX26 peroxisomal biogenesis factor 26
PIM1 Pim-1 proto-oncogene, serine/threonine kinase
PLD2 phospholipase D2
PLEC plectin
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
PLXNA3 plexin A3
PODXL podocalyxin-like
PPIP5K1 diphosphoinositol pentakisphosphate kinase 1
QDPR quinoid dihydropteridine reductase
RBM42 RNA binding motif protein 42
RGS19 regulator of G-protein signaling 19
RHOBTB2 Rho-related BTB domain containing 2
RNF126P1 ring finger protein 126 pseudogene 1
SETD1A SET domain containing 1A
SLC12A8 solute carrier family 12, member 8
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SMPD2 sphingomyelin phosphodiesterase 2, neutral membrane (neutral sphingomyelinase)
SOWAHC sosondowah ankyrin repeat domain family member C
STARD5 StAR-related lipid transfer (START) domain containing 5
STON1 stonin 1
SYNGR3 synaptogyrin 3
TAP1 transporter 1, ATP-binding cassette, sub-family B (MDR/TAP)
TCIRG1 T-cell, immune regulator 1, ATPase, H+ transporting, lysosomal V0 subunit A3
TESC tescalcin
THBS3 thrombospondin 3
TIMM50 translocase of inner mitochondrial membrane 50 homolog (S. cerevisiae)
TMEM209 transmembrane protein 209
TMEM62 transmembrane protein 62
TNKS2 tankyrase, TRF1-interacting ankyrin-related ADP-ribose polymerase 2
TPST2 tyrosylprotein sulfotransferase 2
TRABD TraB domain containing
TTF2 transcription termination factor, RNA polymerase II
TUBA3C tubulin, alpha 3c
UNC119 unc-119 homolog (C. elegans)
USP19 ubiquitin specific peptidase 19
VPS54 vacuolar protein sorting 54 homolog (S. cerevisiae)
YY2 YY2 transcription factor
ZNF165 zinc finger protein 165
ZNF286A zinc finger protein 286A
ZNF394 zinc finger protein 394
ZNF428 zinc finger protein 428
ZSCAN26 zinc finger and SCAN domain containing 26