glipizide-1508 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the glipizide-1508 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACBD4 acyl-CoA binding domain containing 4
ACYP1 acylphosphatase 1, erythrocyte (common) type
ADAM17 ADAM metallopeptidase domain 17
AKR1C1 aldo-keto reductase family 1, member C1
ANKRD12 ankyrin repeat domain 12
APBA2 amyloid beta (A4) precursor protein-binding, family A, member 2
ATAD5 ATPase family, AAA domain containing 5
ATAT1 alpha tubulin acetyltransferase 1
ATF6B activating transcription factor 6 beta
BAHCC1 BAH domain and coiled-coil containing 1
BTN2A2 butyrophilin, subfamily 2, member A2
CALCR calcitonin receptor
CD34 CD34 molecule
CDC25C cell division cycle 25C
CDK20 cyclin-dependent kinase 20
CEP97 centrosomal protein 97kDa
CNTFR ciliary neurotrophic factor receptor
CRHR2 corticotropin releasing hormone receptor 2
CTNND2 catenin (cadherin-associated protein), delta 2
DHRS2 dehydrogenase/reductase (SDR family) member 2
DMXL2 Dmx-like 2
DNAJB12 DnaJ (Hsp40) homolog, subfamily B, member 12
DNPEP aspartyl aminopeptidase
DYRK3 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 3
EGR1 early growth response 1
EHMT1 euchromatic histone-lysine N-methyltransferase 1
EPOR erythropoietin receptor
FAM110B family with sequence similarity 110, member B
FHL1 four and a half LIM domains 1
FLOT1 flotillin 1
FLRT2 fibronectin leucine rich transmembrane protein 2
FSCN1 fascin actin-bundling protein 1
FSCN3 fascin actin-bundling protein 3, testicular
GPR137 G protein-coupled receptor 137
GPRC5D G protein-coupled receptor, class C, group 5, member D
GRK6 G protein-coupled receptor kinase 6
HEMK1 HemK methyltransferase family member 1
HFE hemochromatosis
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
HOXC4 homeobox C4
IDI2-AS1 IDI2 antisense RNA 1
IGHA1 immunoglobulin heavy constant alpha 1
IL6ST interleukin 6 signal transducer
IMPG2 interphotoreceptor matrix proteoglycan 2
JAK2 Janus kinase 2
JUN jun proto-oncogene
KAT6B K(lysine) acetyltransferase 6B
KIAA0319L KIAA0319-like
KIAA1107 KIAA1107
KRIT1 KRIT1, ankyrin repeat containing
LPXN leupaxin
MARK4 MAP/microtubule affinity-regulating kinase 4
MLXIP MLX interacting protein
MMP15 matrix metallopeptidase 15 (membrane-inserted)
MSR1 macrophage scavenger receptor 1
MXD4 MAX dimerization protein 4
NFIB nuclear factor I/B
NMT2 N-myristoyltransferase 2
NR2C1 nuclear receptor subfamily 2, group C, member 1
NRSN2 neurensin 2
NTF3 neurotrophin 3
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18
OGFOD2 2-oxoglutarate and iron-dependent oxygenase domain containing 2
PARVA parvin, alpha
PDK1 pyruvate dehydrogenase kinase, isozyme 1
PGAP1 post-GPI attachment to proteins 1
PGBD5 piggyBac transposable element derived 5
POFUT1 protein O-fucosyltransferase 1
POMT2 protein-O-mannosyltransferase 2
PPP2R5B protein phosphatase 2, regulatory subunit B', beta
PRKACA protein kinase, cAMP-dependent, catalytic, alpha
PRPH peripherin
PRRC2A proline-rich coiled-coil 2A
PTK6 protein tyrosine kinase 6
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RASA3 RAS p21 protein activator 3
RBM19 RNA binding motif protein 19
RUNDC3B RUN domain containing 3B
SCAF4 SR-related CTD-associated factor 4
SCAPER S-phase cyclin A-associated protein in the ER
SH2D2A SH2 domain containing 2A
SIRT6 sirtuin 6
SLC22A4 solute carrier family 22 (organic cation/zwitterion transporter), member 4
SLC45A2 solute carrier family 45, member 2
SLC52A1 solute carrier family 52 (riboflavin transporter), member 1
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SLCO3A1 solute carrier organic anion transporter family, member 3A1
SMIM14 small integral membrane protein 14
SPG20 spastic paraplegia 20 (Troyer syndrome)
SRD5A3 steroid 5 alpha-reductase 3
SYNJ1 synaptojanin 1
TAF6L TAF6-like RNA polymerase II, p300/CBP-associated factor (PCAF)-associated factor, 65kDa
TJAP1 tight junction associated protein 1 (peripheral)
TNFAIP3 tumor necrosis factor, alpha-induced protein 3
TNFRSF25 tumor necrosis factor receptor superfamily, member 25
XDH xanthine dehydrogenase
ZC3H3 zinc finger CCCH-type containing 3
ZNF204P zinc finger protein 204, pseudogene
ZNF573 zinc finger protein 573
ZNF862 zinc finger protein 862

decreased expression

Symbol Name
AHDC1 AT hook, DNA binding motif, containing 1
ANKEF1 ankyrin repeat and EF-hand domain containing 1
ANKRD2 ankyrin repeat domain 2 (stretch responsive muscle)
ARID3A AT rich interactive domain 3A (BRIGHT-like)
ART1 ADP-ribosyltransferase 1
ASPSCR1 alveolar soft part sarcoma chromosome region, candidate 1
BCL2L2 BCL2-like 2
BMP4 bone morphogenetic protein 4
C11ORF30 chromosome 11 open reading frame 30
C11ORF63 chromosome 11 open reading frame 63
C22ORF29 chromosome 22 open reading frame 29
CCDC85C coiled-coil domain containing 85C
CCP110 centriolar coiled coil protein 110kDa
CD83 CD83 molecule
CDK3 cyclin-dependent kinase 3
CDKN2D cyclin-dependent kinase inhibitor 2D (p19, inhibits CDK4)
CGA glycoprotein hormones, alpha polypeptide
CIR1 corepressor interacting with RBPJ, 1
CNGB3 cyclic nucleotide gated channel beta 3
CNN2 calponin 2
CTDP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1
CTSV cathepsin V
CUL9 cullin 9
EPHA2 EPH receptor A2
ERN2 endoplasmic reticulum to nucleus signaling 2
FAM53B family with sequence similarity 53, member B
FBXO4 F-box protein 4
FER fer (fps/fes related) tyrosine kinase
GCNT1 glucosaminyl (N-acetyl) transferase 1, core 2
GCNT2 glucosaminyl (N-acetyl) transferase 2, I-branching enzyme (I blood group)
GLB1L galactosidase, beta 1-like
GLI3 GLI family zinc finger 3
GNG7 guanine nucleotide binding protein (G protein), gamma 7
GPR27 G protein-coupled receptor 27
GRTP1 growth hormone regulated TBC protein 1
HEY2 hes-related family bHLH transcription factor with YRPW motif 2
HIRA histone cell cycle regulator
HIST1H2AE histone cluster 1, H2ae
IFT54 intraflagellar transport 54
IL17RA interleukin 17 receptor A
IQSEC2 IQ motif and Sec7 domain 2
IRF1 interferon regulatory factor 1
KCNMB4 potassium channel subfamily M regulatory beta subunit 4
KLK5 kallikrein-related peptidase 5
LHX1 LIM homeobox 1
LIME1 Lck interacting transmembrane adaptor 1
LRP2 low density lipoprotein receptor-related protein 2
LRRC37A2 leucine rich repeat containing 37, member A2
LTBP2 latent transforming growth factor beta binding protein 2
LY6D lymphocyte antigen 6 complex, locus D
LYL1 lymphoblastic leukemia associated hematopoiesis regulator 1
MANBA mannosidase, beta A, lysosomal
MCOLN3 mucolipin 3
MSI1 musashi RNA-binding protein 1
NACA2 nascent polypeptide-associated complex alpha subunit 2
NAT6 N-acetyltransferase 6 (GCN5-related)
NPFFR1 neuropeptide FF receptor 1
NR1H3 nuclear receptor subfamily 1, group H, member 3
OR1D2 olfactory receptor, family 1, subfamily D, member 2
OR2F1 olfactory receptor, family 2, subfamily F, member 1 (gene/pseudogene)
ORAI3 ORAI calcium release-activated calcium modulator 3
P3H1 prolyl 3-hydroxylase 1
PEX26 peroxisomal biogenesis factor 26
PICK1 protein interacting with PRKCA 1
PLCXD1 phosphatidylinositol-specific phospholipase C, X domain containing 1
PLEKHG6 pleckstrin homology domain containing, family G (with RhoGef domain) member 6
PPP1R14D protein phosphatase 1, regulatory (inhibitor) subunit 14D
PROCR protein C receptor, endothelial
PTPN9 protein tyrosine phosphatase, non-receptor type 9
RALGPS2 Ral GEF with PH domain and SH3 binding motif 2
RANBP17 RAN binding protein 17
RHBDD3 rhomboid domain containing 3
ROM1 retinal outer segment membrane protein 1
RUSC2 RUN and SH3 domain containing 2
SAA4 serum amyloid A4, constitutive
SAYSD1 SAYSVFN motif domain containing 1
SCN1B sodium channel, voltage gated, type I beta subunit
SLC12A6 solute carrier family 12 (potassium/chloride transporter), member 6
SLC17A2 solute carrier family 17, member 2
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SLC3A1 solute carrier family 3 (amino acid transporter heavy chain), member 1
SMARCD3 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 3
SNAPC2 small nuclear RNA activating complex, polypeptide 2, 45kDa
SP1 Sp1 transcription factor
TAF13 TAF13 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 18kDa
TFF2 trefoil factor 2
TMC5 transmembrane channel-like 5
TNFRSF11A tumor necrosis factor receptor superfamily, member 11a, NFKB activator
TPCN1 two pore segment channel 1
TSPAN5 tetraspanin 5
UBQLN4 ubiquilin 4
UPP1 uridine phosphorylase 1
VIM vimentin
VPS33A vacuolar protein sorting 33 homolog A (S. cerevisiae)
XYLT2 xylosyltransferase II
ZNF134 zinc finger protein 134
ZNF350 zinc finger protein 350
ZNF669 zinc finger protein 669