gramine-2143 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

194 genes differentially expressed following the gramine-2143 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
APP amyloid beta (A4) precursor protein
ATP9B ATPase, class II, type 9B
B9D2 B9 protein domain 2
CAMSAP1 calmodulin regulated spectrin-associated protein 1
CCDC57 coiled-coil domain containing 57
CCNK cyclin K
CD200 CD200 molecule
CD47 CD47 molecule
CDC42BPA CDC42 binding protein kinase alpha (DMPK-like)
CFLAR CASP8 and FADD-like apoptosis regulator
CHST7 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 7
COL10A1 collagen, type X, alpha 1
COL9A3 collagen, type IX, alpha 3
CPTP ceramide-1-phosphate transfer protein
CREM cAMP responsive element modulator
CSF2RA colony stimulating factor 2 receptor, alpha, low-affinity (granulocyte-macrophage)
CXCR3 chemokine (C-X-C motif) receptor 3
CYHR1 cysteine/histidine-rich 1
CYP1B1 cytochrome P450, family 1, subfamily B, polypeptide 1
DCAF17 DDB1 and CUL4 associated factor 17
EDRF1 erythroid differentiation regulatory factor 1
EEF1A2 eukaryotic translation elongation factor 1 alpha 2
EFR3B EFR3 homolog B (S. cerevisiae)
ELP6 elongator acetyltransferase complex subunit 6
FAM105A family with sequence similarity 105, member A
FAM65B family with sequence similarity 65, member B
FBXW4P1 F-box and WD repeat domain containing 4 pseudogene 1
FLOT1 flotillin 1
FN1 fibronectin 1
FUBP1 far upstream element (FUSE) binding protein 1
GK3P glycerol kinase 3 pseudogene
GPR135 G protein-coupled receptor 135
GRWD1 glutamate-rich WD repeat containing 1
H2AFX H2A histone family, member X
HCFC1R1 host cell factor C1 regulator 1 (XPO1 dependent)
HDGFRP3 hepatoma-derived growth factor, related protein 3
HIC2 hypermethylated in cancer 2
HIF1AN hypoxia inducible factor 1, alpha subunit inhibitor
HIST1H2AK histone cluster 1, H2ak
HOXA10 homeobox A10
HRH2 histamine receptor H2
INPP4A inositol polyphosphate-4-phosphatase, type I, 107kDa
ISG20 interferon stimulated exonuclease gene 20kDa
KIAA1109 KIAA1109
KLF12 Kruppel-like factor 12
KMT2A lysine (K)-specific methyltransferase 2A
LENEP lens epithelial protein
LIN7B lin-7 homolog B (C. elegans)
LINC00652 long intergenic non-protein coding RNA 652
LPAR6 lysophosphatidic acid receptor 6
LSM14B LSM14B, SCD6 homolog B (S. cerevisiae)
MERTK MER proto-oncogene, tyrosine kinase
MLLT3 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 3
MMP14 matrix metallopeptidase 14 (membrane-inserted)
MMP24 matrix metallopeptidase 24 (membrane-inserted)
MRPS12 mitochondrial ribosomal protein S12
MTUS1 microtubule associated tumor suppressor 1
N4BP2L2-IT2 N4BPL2 intronic transcript 2
NFKBIB nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, beta
NMT2 N-myristoyltransferase 2
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18
NUMA1 nuclear mitotic apparatus protein 1
OR10J1 olfactory receptor, family 10, subfamily J, member 1
OR2H2 olfactory receptor, family 2, subfamily H, member 2
P2RY1 purinergic receptor P2Y, G-protein coupled, 1
PDE6H phosphodiesterase 6H, cGMP-specific, cone, gamma
PKNOX1 PBX/knotted 1 homeobox 1
PMS2P3 postmeiotic segregation increased 2 pseudogene 3
PPARD peroxisome proliferator-activated receptor delta
PPFIBP2 PTPRF interacting protein, binding protein 2 (liprin beta 2)
PRKAR2A protein kinase, cAMP-dependent, regulatory, type II, alpha
PTGDS prostaglandin D2 synthase 21kDa (brain)
RAB3D RAB3D, member RAS oncogene family
RANBP3 RAN binding protein 3
RDX radixin
RPS28 ribosomal protein S28
RRN3P1 RNA polymerase I transcription factor homolog (S. cerevisiae) pseudogene 1
SEC24A SEC24 family member A
SLC17A7 solute carrier family 17 (vesicular glutamate transporter), member 7
SLC29A3 solute carrier family 29 (equilibrative nucleoside transporter), member 3
SLC48A1 solute carrier family 48 (heme transporter), member 1
SLC7A9 solute carrier family 7 (amino acid transporter light chain, bo,+ system), member 9
SLMO1 slowmo homolog 1 (Drosophila)
SPHK2 sphingosine kinase 2
TBC1D1 TBC1 (tre-2/USP6, BUB2, cdc16) domain family, member 1
THAP10 THAP domain containing 10
THY1 Thy-1 cell surface antigen
TMCC2 transmembrane and coiled-coil domain family 2
TRIM25 tripartite motif containing 25
TRIM3 tripartite motif containing 3
UBR2 ubiquitin protein ligase E3 component n-recognin 2
VAMP2 vesicle-associated membrane protein 2 (synaptobrevin 2)
WNT16 wingless-type MMTV integration site family, member 16
XIST X inactive specific transcript (non-protein coding)
ZER1 zyg-11 related, cell cycle regulator
ZMAT5 zinc finger, matrin-type 5
ZNF778 zinc finger protein 778

decreased expression

Symbol Name
A2M alpha-2-macroglobulin
ACPP acid phosphatase, prostate
ADTRP androgen-dependent TFPI-regulating protein
ALDH2 aldehyde dehydrogenase 2 family (mitochondrial)
ANKZF1 ankyrin repeat and zinc finger domain containing 1
ARAF A-Raf proto-oncogene, serine/threonine kinase
BAHCC1 BAH domain and coiled-coil containing 1
C17ORF53 chromosome 17 open reading frame 53
C17ORF70 chromosome 17 open reading frame 70
C22ORF29 chromosome 22 open reading frame 29
C7ORF43 chromosome 7 open reading frame 43
CDH10 cadherin 10, type 2 (T2-cadherin)
CEP97 centrosomal protein 97kDa
CHST2 carbohydrate (N-acetylglucosamine-6-O) sulfotransferase 2
CIDEB cell death-inducing DFFA-like effector b
CILP cartilage intermediate layer protein, nucleotide pyrophosphohydrolase
COPS7B COP9 signalosome subunit 7B
CORT cortistatin
DAP death-associated protein
DGKG diacylglycerol kinase, gamma 90kDa
DOK5 docking protein 5
DPF2 D4, zinc and double PHD fingers family 2
DUSP8 dual specificity phosphatase 8
DYNC2H1 dynein, cytoplasmic 2, heavy chain 1
EFNA3 ephrin-A3
ERCC2 excision repair cross-complementation group 2
FAM57A family with sequence similarity 57, member A
FBXO46 F-box protein 46
FOSB FBJ murine osteosarcoma viral oncogene homolog B
FOXC1 forkhead box C1
FRAT1 frequently rearranged in advanced T-cell lymphomas 1
GALE UDP-galactose-4-epimerase
GJA1 gap junction protein, alpha 1, 43kDa
GNL3LP1 guanine nucleotide binding protein-like 3 (nucleolar)-like pseudogene 1
GSTT1 glutathione S-transferase theta 1
HIRA histone cell cycle regulator
HIST1H2AM histone cluster 1, H2am
HIST1H4D histone cluster 1, H4d
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
HPS6 Hermansky-Pudlak syndrome 6
HPSE heparanase
IFIT3 interferon-induced protein with tetratricopeptide repeats 3
IGLL3P immunoglobulin lambda-like polypeptide 3, pseudogene
ITGA2 integrin, alpha 2 (CD49B, alpha 2 subunit of VLA-2 receptor)
ITPKC inositol-trisphosphate 3-kinase C
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNMB4 potassium channel subfamily M regulatory beta subunit 4
KIF24 kinesin family member 24
KIFC1 kinesin family member C1
KLK5 kallikrein-related peptidase 5
LIMD2 LIM domain containing 2
LOC157562 uncharacterized LOC157562
LY6G6C lymphocyte antigen 6 complex, locus G6C
MAP1S microtubule-associated protein 1S
MCTP2 multiple C2 domains, transmembrane 2
MRM1 mitochondrial rRNA methyltransferase 1 homolog (S. cerevisiae)
NTSR1 neurotensin receptor 1 (high affinity)
OR12D2 olfactory receptor, family 12, subfamily D, member 2 (gene/pseudogene)
OXCT2 3-oxoacid CoA transferase 2
PADI1 peptidyl arginine deiminase, type I
PAPD7 PAP associated domain containing 7
PECR peroxisomal trans-2-enoyl-CoA reductase
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PKIG protein kinase (cAMP-dependent, catalytic) inhibitor gamma
POLL polymerase (DNA directed), lambda
PRAMEF11 PRAME family member 11
RAB33A RAB33A, member RAS oncogene family
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RASAL1 RAS protein activator like 1 (GAP1 like)
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
RPAP1 RNA polymerase II associated protein 1
RRAS related RAS viral (r-ras) oncogene homolog
SEMA4D sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4D
SHARPIN SHANK-associated RH domain interactor
SLC2A9 solute carrier family 2 (facilitated glucose transporter), member 9
SLC4A2 solute carrier family 4 (anion exchanger), member 2
SULT1B1 sulfotransferase family, cytosolic, 1B, member 1
TAGLN transgelin
TCTN2 tectonic family member 2
TICAM1 toll-like receptor adaptor molecule 1
TM7SF2 transmembrane 7 superfamily member 2
TMEM127 transmembrane protein 127
TMEM180 transmembrane protein 180
TMEM212 transmembrane protein 212
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TRAF2 TNF receptor-associated factor 2
TRNAU1AP tRNA selenocysteine 1 associated protein 1
UBE2NL ubiquitin-conjugating enzyme E2N-like (gene/pseudogene)
UCN urocortin
USP19 ubiquitin specific peptidase 19
WNT10B wingless-type MMTV integration site family, member 10B
ZBTB38 zinc finger and BTB domain containing 38
ZNF185 zinc finger protein 185 (LIM domain)
ZNF215 zinc finger protein 215
ZNF665 zinc finger protein 665
ZNF747 zinc finger protein 747
ZNF749 zinc finger protein 749