heliotrine-6035 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the heliotrine-6035 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
A4GNT alpha-1,4-N-acetylglucosaminyltransferase
AADAC arylacetamide deacetylase
ACRV1 acrosomal vesicle protein 1
ALDOAP2 aldolase A, fructose-bisphosphate pseudogene 2
AMPH amphiphysin
ANGPTL2 angiopoietin-like 2
ARFGEF2 ADP-ribosylation factor guanine nucleotide-exchange factor 2 (brefeldin A-inhibited)
ARHGEF38 Rho guanine nucleotide exchange factor (GEF) 38
BMP1 bone morphogenetic protein 1
BMP8B bone morphogenetic protein 8b
C11ORF21 chromosome 11 open reading frame 21
C19ORF66 chromosome 19 open reading frame 66
CACNB2 calcium channel, voltage-dependent, beta 2 subunit
CALD1 caldesmon 1
CAMK4 calcium/calmodulin-dependent protein kinase IV
CCL19 chemokine (C-C motif) ligand 19
CCL23 chemokine (C-C motif) ligand 23
CD58 CD58 molecule
CD84 CD84 molecule
CIITA class II, major histocompatibility complex, transactivator
CNPY4 canopy FGF signaling regulator 4
CPED1 cadherin-like and PC-esterase domain containing 1
CR1 complement component (3b/4b) receptor 1 (Knops blood group)
CROCC ciliary rootlet coiled-coil, rootletin
CYP3A5 cytochrome P450, family 3, subfamily A, polypeptide 5
DAB2 Dab, mitogen-responsive phosphoprotein, homolog 2 (Drosophila)
DGCR8 DGCR8 microprocessor complex subunit
DLK1 delta-like 1 homolog (Drosophila)
DMP1 dentin matrix acidic phosphoprotein 1
DNAJB5 DnaJ (Hsp40) homolog, subfamily B, member 5
DOK4 docking protein 4
ECE1 endothelin converting enzyme 1
EDA ectodysplasin A
ERC2-IT1 ERC2 intronic transcript 1
ERO1LB ERO1-like beta (S. cerevisiae)
FABP3 fatty acid binding protein 3, muscle and heart
FAM66D family with sequence similarity 66, member D
FCMR Fc fragment of IgM receptor
FUT6 fucosyltransferase 6 (alpha (1,3) fucosyltransferase)
GPR137 G protein-coupled receptor 137
GRIP2 glutamate receptor interacting protein 2
HGF hepatocyte growth factor (hepapoietin A; scatter factor)
IFI6 interferon, alpha-inducible protein 6
IL18 interleukin 18
IL1RN interleukin 1 receptor antagonist
JMJD6 jumonji domain containing 6
KIT v-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog
KRT83 keratin 83, type II
LIPE lipase, hormone-sensitive
LRRC15 leucine rich repeat containing 15
LYVE1 lymphatic vessel endothelial hyaluronan receptor 1
MAOA monoamine oxidase A
MAPK7 mitogen-activated protein kinase 7
MIR622 microRNA 622
MLN motilin
MLXIPL MLX interacting protein-like
MRPS12 mitochondrial ribosomal protein S12
MUC5AC mucin 5AC, oligomeric mucus/gel-forming
MYO7B myosin VIIB
NDUFA2 NADH dehydrogenase (ubiquinone) 1 alpha subcomplex, 2, 8kDa
NLRP3 NLR family, pyrin domain containing 3
NMBR neuromedin B receptor
NR2F1 nuclear receptor subfamily 2, group F, member 1
OPCML opioid binding protein/cell adhesion molecule-like
PBXIP1 pre-B-cell leukemia homeobox interacting protein 1
PCDH7 protocadherin 7
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
PKNOX2 PBX/knotted 1 homeobox 2
POLM polymerase (DNA directed), mu
PRTN3 proteinase 3
PSG6 pregnancy specific beta-1-glycoprotein 6
PTPN12 protein tyrosine phosphatase, non-receptor type 12
PVR poliovirus receptor
RAB6B RAB6B, member RAS oncogene family
RAP1GAP RAP1 GTPase activating protein
RARRES2 retinoic acid receptor responder (tazarotene induced) 2
RASGRF1 Ras protein-specific guanine nucleotide-releasing factor 1
RXRB retinoid X receptor, beta
SATB2 SATB homeobox 2
SIPA1L3 signal-induced proliferation-associated 1 like 3
SLC2A1 solute carrier family 2 (facilitated glucose transporter), member 1
SLC52A1 solute carrier family 52 (riboflavin transporter), member 1
SLCO2A1 solute carrier organic anion transporter family, member 2A1
SLURP1 secreted LY6/PLAUR domain containing 1
SOGA1 suppressor of glucose, autophagy associated 1
SP140 SP140 nuclear body protein
SSX1 synovial sarcoma, X breakpoint 1
STAB1 stabilin 1
SYN3 synapsin III
THY1 Thy-1 cell surface antigen
TIMM8A translocase of inner mitochondrial membrane 8 homolog A (yeast)
TIMP4 TIMP metallopeptidase inhibitor 4
TJAP1 tight junction associated protein 1 (peripheral)
TRAPPC9 trafficking protein particle complex 9
URB1 URB1 ribosome biogenesis 1 homolog (S. cerevisiae)
ZBTB22 zinc finger and BTB domain containing 22
ZNF280A zinc finger protein 280A
ZNF639 zinc finger protein 639

decreased expression

Symbol Name
ACAD10 acyl-CoA dehydrogenase family, member 10
ADM adrenomedullin
AHNAK2 AHNAK nucleoprotein 2
AOC2 amine oxidase, copper containing 2 (retina-specific)
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
BAHD1 bromo adjacent homology domain containing 1
BCL11B B-cell CLL/lymphoma 11B (zinc finger protein)
C7ORF43 chromosome 7 open reading frame 43
CACNA1H calcium channel, voltage-dependent, T type, alpha 1H subunit
CD83 CD83 molecule
CDK3 cyclin-dependent kinase 3
CDON cell adhesion associated, oncogene regulated
CEACAM4 carcinoembryonic antigen-related cell adhesion molecule 4
CEP97 centrosomal protein 97kDa
CLDN17 claudin 17
CNNM1 cyclin and CBS domain divalent metal cation transport mediator 1
CNR2 cannabinoid receptor 2 (macrophage)
COPZ2 coatomer protein complex, subunit zeta 2
CTSF cathepsin F
DMTN dematin actin binding protein
DNMT3A DNA (cytosine-5-)-methyltransferase 3 alpha
EN2 engrailed homeobox 2
ENTPD5 ectonucleoside triphosphate diphosphohydrolase 5
ERCC6 excision repair cross-complementation group 6
ERN2 endoplasmic reticulum to nucleus signaling 2
FAM76A family with sequence similarity 76, member A
FBXL2 F-box and leucine-rich repeat protein 2
FGF23 fibroblast growth factor 23
FGL1 fibrinogen-like 1
FKBP8 FK506 binding protein 8, 38kDa
GBP2 guanylate binding protein 2, interferon-inducible
GIT1 G protein-coupled receptor kinase interacting ArfGAP 1
GPC3 glypican 3
GPR21 G protein-coupled receptor 21
GRPR gastrin-releasing peptide receptor
GUCY1B2 guanylate cyclase 1, soluble, beta 2 (pseudogene)
HDAC11 histone deacetylase 11
HIST1H2AJ histone cluster 1, H2aj
HOXA4 homeobox A4
HOXC8 homeobox C8
HS3ST3A1 heparan sulfate (glucosamine) 3-O-sulfotransferase 3A1
IDI2-AS1 IDI2 antisense RNA 1
IFT22 intraflagellar transport 22
ISG20 interferon stimulated exonuclease gene 20kDa
KIAA0754 KIAA0754
KREMEN2 kringle containing transmembrane protein 2
LINC00597 long intergenic non-protein coding RNA 597
LMX1B LIM homeobox transcription factor 1, beta
LZTFL1 leucine zipper transcription factor-like 1
MED9 mediator complex subunit 9
MPP3 membrane protein, palmitoylated 3 (MAGUK p55 subfamily member 3)
NIPAL2 NIPA-like domain containing 2
NKX3-2 NK3 homeobox 2
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18
OLFML2A olfactomedin-like 2A
PC pyruvate carboxylase
PCDHA5 protocadherin alpha 5
PCYT2 phosphate cytidylyltransferase 2, ethanolamine
POLL polymerase (DNA directed), lambda
PORCN porcupine homolog (Drosophila)
PRF1 perforin 1 (pore forming protein)
PRODH proline dehydrogenase (oxidase) 1
PRPH peripherin
PTDSS2 phosphatidylserine synthase 2
RAB30 RAB30, member RAS oncogene family
SALL2 spalt-like transcription factor 2
SCGB2A2 secretoglobin, family 2A, member 2
SERPINE2 serpin peptidase inhibitor, clade E (nexin, plasminogen activator inhibitor type 1), member 2
SIGLEC15 sialic acid binding Ig-like lectin 15
SIPA1 signal-induced proliferation-associated 1
SLC17A2 solute carrier family 17, member 2
SLC3A1 solute carrier family 3 (amino acid transporter heavy chain), member 1
SLC8B1 solute carrier family 8 (sodium/lithium/calcium exchanger), member B1
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SPAG7 sperm associated antigen 7
SPTBN2 spectrin, beta, non-erythrocytic 2
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5
TBC1D19 TBC1 domain family, member 19
TESC tescalcin
TGFB1I1 transforming growth factor beta 1 induced transcript 1
TMCC2 transmembrane and coiled-coil domain family 2
TMEM104 transmembrane protein 104
TMEM180 transmembrane protein 180
TMEM242 transmembrane protein 242
TOP3B topoisomerase (DNA) III beta
TOR4A torsin family 4, member A
TRAPPC11 trafficking protein particle complex 11
TRDMT1 tRNA aspartic acid methyltransferase 1
TRPM4 transient receptor potential cation channel, subfamily M, member 4
VWA1 von Willebrand factor A domain containing 1
WDR62 WD repeat domain 62
WLS wntless Wnt ligand secretion mediator
YY2 YY2 transcription factor
ZC3H3 zinc finger CCCH-type containing 3
ZFHX4 zinc finger homeobox 4
ZNF136 zinc finger protein 136
ZNF205 zinc finger protein 205
ZNF532 zinc finger protein 532
ZNF551 zinc finger protein 551