| Dataset | CMAP Signatures of Differentially Expressed Genes for Small Molecules |
| Category | transcriptomics |
| Type | small molecule perturbation |
| Description | small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis) |
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195 genes differentially expressed following the karakoline-4297 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.
| Symbol | Name |
|---|---|
| ABCG1 | ATP-binding cassette, sub-family G (WHITE), member 1 |
| ACE2 | angiotensin I converting enzyme 2 |
| ACRV1 | acrosomal vesicle protein 1 |
| ADAMDEC1 | ADAM-like, decysin 1 |
| ADAMTS7 | ADAM metallopeptidase with thrombospondin type 1 motif, 7 |
| AHI1 | Abelson helper integration site 1 |
| AIM2 | absent in melanoma 2 |
| ALDOB | aldolase B, fructose-bisphosphate |
| ANK3 | ankyrin 3, node of Ranvier (ankyrin G) |
| AQP4 | aquaporin 4 |
| C10ORF10 | chromosome 10 open reading frame 10 |
| C9ORF156 | chromosome 9 open reading frame 156 |
| CACNA2D1 | calcium channel, voltage-dependent, alpha 2/delta subunit 1 |
| CAMK4 | calcium/calmodulin-dependent protein kinase IV |
| CASP2 | caspase 2, apoptosis-related cysteine peptidase |
| CD40 | CD40 molecule, TNF receptor superfamily member 5 |
| CD58 | CD58 molecule |
| CDKAL1 | CDK5 regulatory subunit associated protein 1-like 1 |
| CEACAM1 | carcinoembryonic antigen-related cell adhesion molecule 1 (biliary glycoprotein) |
| CLCA1 | chloride channel accessory 1 |
| CR1 | complement component (3b/4b) receptor 1 (Knops blood group) |
| DGCR14 | DiGeorge syndrome critical region gene 14 |
| DMRT1 | doublesex and mab-3 related transcription factor 1 |
| DSTYK | dual serine/threonine and tyrosine protein kinase |
| EDN1 | endothelin 1 |
| EGR1 | early growth response 1 |
| EIF5A | eukaryotic translation initiation factor 5A |
| EPM2A | epilepsy, progressive myoclonus type 2A, Lafora disease (laforin) |
| EPS8L3 | EPS8-like 3 |
| ESR1 | estrogen receptor 1 |
| ESRRG | estrogen-related receptor gamma |
| FAM46C | family with sequence similarity 46, member C |
| FHL3 | four and a half LIM domains 3 |
| FLI1 | Fli-1 proto-oncogene, ETS transcription factor |
| FOLH1 | folate hydrolase (prostate-specific membrane antigen) 1 |
| GPM6B | glycoprotein M6B |
| HHAT | hedgehog acyltransferase |
| HIST1H1D | histone cluster 1, H1d |
| HIST1H1E | histone cluster 1, H1e |
| HMGB3P1 | high mobility group box 3 pseudogene 1 |
| HTR2A | 5-hydroxytryptamine (serotonin) receptor 2A, G protein-coupled |
| IGSF6 | immunoglobulin superfamily, member 6 |
| IRF4 | interferon regulatory factor 4 |
| ITPR3 | inositol 1,4,5-trisphosphate receptor, type 3 |
| KCNAB2 | potassium channel, voltage gated subfamily A regulatory beta subunit 2 |
| KCNG1 | potassium channel, voltage gated modifier subfamily G, member 1 |
| KCTD14 | potassium channel tetramerization domain containing 14 |
| KIR2DL5A | killer cell immunoglobulin-like receptor, two domains, long cytoplasmic tail, 5A |
| LAT2 | linker for activation of T cells family, member 2 |
| LCMT2 | leucine carboxyl methyltransferase 2 |
| LLGL1 | lethal giant larvae homolog 1 (Drosophila) |
| MCF2L | MCF.2 cell line derived transforming sequence-like |
| MINK1 | misshapen-like kinase 1 |
| MTNR1A | melatonin receptor 1A |
| MUC3A | mucin 3A, cell surface associated |
| MYO15B | myosin XVB |
| NDUFA2 | NADH dehydrogenase (ubiquinone) 1 alpha subcomplex, 2, 8kDa |
| NDUFAF5 | NADH dehydrogenase (ubiquinone) complex I, assembly factor 5 |
| NR4A1 | nuclear receptor subfamily 4, group A, member 1 |
| OR7E19P | olfactory receptor, family 7, subfamily E, member 19 pseudogene |
| OSR2 | odd-skipped related transciption factor 2 |
| PCDHB3 | protocadherin beta 3 |
| PKP4 | plakophilin 4 |
| PLXNA2 | plexin A2 |
| PRDX2 | peroxiredoxin 2 |
| PRKAR1B | protein kinase, cAMP-dependent, regulatory, type I, beta |
| PVRL1 | poliovirus receptor-related 1 (herpesvirus entry mediator C) |
| PVT1 | Pvt1 oncogene (non-protein coding) |
| QPCTL | glutaminyl-peptide cyclotransferase-like |
| RAB40B | RAB40B, member RAS oncogene family |
| RAB6B | RAB6B, member RAS oncogene family |
| RASSF4 | Ras association (RalGDS/AF-6) domain family member 4 |
| RBFOX1 | RNA binding protein, fox-1 homolog (C. elegans) 1 |
| REM1 | RAS (RAD and GEM)-like GTP-binding 1 |
| RET | ret proto-oncogene |
| RHEB | Ras homolog enriched in brain |
| RNASE2 | ribonuclease, RNase A family, 2 (liver, eosinophil-derived neurotoxin) |
| RUNX1T1 | runt-related transcription factor 1; translocated to, 1 (cyclin D-related) |
| SAYSD1 | SAYSVFN motif domain containing 1 |
| SCN3B | sodium channel, voltage gated, type III beta subunit |
| SEC14L4 | SEC14-like 4 (S. cerevisiae) |
| SERPINA7 | serpin peptidase inhibitor, clade A (alpha-1 antiproteinase, antitrypsin), member 7 |
| SFTPB | surfactant protein B |
| SHOX2 | short stature homeobox 2 |
| SIRT4 | sirtuin 4 |
| SOX2 | SRY (sex determining region Y)-box 2 |
| SUGP1 | SURP and G patch domain containing 1 |
| TAPBP | TAP binding protein (tapasin) |
| TBR1 | T-box, brain, 1 |
| TFR2 | transferrin receptor 2 |
| TMPO | thymopoietin |
| TNNT2 | troponin T type 2 (cardiac) |
| TP53I11 | tumor protein p53 inducible protein 11 |
| TRIM25 | tripartite motif containing 25 |
| VDR | vitamin D (1,25- dihydroxyvitamin D3) receptor |
| VPS53 | vacuolar protein sorting 53 homolog (S. cerevisiae) |
| ZNF280B | zinc finger protein 280B |
| ZNF507 | zinc finger protein 507 |
| Symbol | Name |
|---|---|
| ACSS3 | acyl-CoA synthetase short-chain family member 3 |
| AGPAT4 | 1-acylglycerol-3-phosphate O-acyltransferase 4 |
| AHDC1 | AT hook, DNA binding motif, containing 1 |
| ALOX12 | arachidonate 12-lipoxygenase |
| ALOX12P2 | arachidonate 12-lipoxygenase pseudogene 2 |
| ANKFY1 | ankyrin repeat and FYVE domain containing 1 |
| ANP32A-IT1 | ANP32A intronic transcript 1 |
| APOL6 | apolipoprotein L, 6 |
| ARMCX2 | armadillo repeat containing, X-linked 2 |
| AXIN1 | axin 1 |
| BAP1 | BRCA1 associated protein-1 (ubiquitin carboxy-terminal hydrolase) |
| C11ORF30 | chromosome 11 open reading frame 30 |
| C4ORF29 | chromosome 4 open reading frame 29 |
| CAPN15 | calpain 15 |
| CBX8 | chromobox homolog 8 |
| CCDC7 | coiled-coil domain containing 7 |
| CCT6B | chaperonin containing TCP1, subunit 6B (zeta 2) |
| CD82 | CD82 molecule |
| CDH7 | cadherin 7, type 2 |
| CEP41 | centrosomal protein 41kDa |
| CFAP45 | cilia and flagella associated protein 45 |
| CHM | choroideremia (Rab escort protein 1) |
| CHST10 | carbohydrate sulfotransferase 10 |
| CHST11 | carbohydrate (chondroitin 4) sulfotransferase 11 |
| CNGA1 | cyclic nucleotide gated channel alpha 1 |
| CTDP1 | CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1 |
| CWF19L1 | CWF19-like 1, cell cycle control (S. pombe) |
| DHX35 | DEAH (Asp-Glu-Ala-His) box polypeptide 35 |
| DLK2 | delta-like 2 homolog (Drosophila) |
| DMBT1 | deleted in malignant brain tumors 1 |
| DMTN | dematin actin binding protein |
| ERMAP | erythroblast membrane-associated protein (Scianna blood group) |
| ERN2 | endoplasmic reticulum to nucleus signaling 2 |
| EYA4 | EYA transcriptional coactivator and phosphatase 4 |
| FCER1G | Fc fragment of IgE, high affinity I, receptor for; gamma polypeptide |
| GRAMD1C | GRAM domain containing 1C |
| HHLA3 | HERV-H LTR-associating 3 |
| HOXA7 | homeobox A7 |
| KCNB1 | potassium channel, voltage gated Shab related subfamily B, member 1 |
| KIAA0319L | KIAA0319-like |
| KIF13A | kinesin family member 13A |
| KLHL36 | kelch-like family member 36 |
| LIG4 | ligase IV, DNA, ATP-dependent |
| LPPR4 | lipid phosphate phosphatase-related protein type 4 |
| LSM14B | LSM14B, SCD6 homolog B (S. cerevisiae) |
| MANBA | mannosidase, beta A, lysosomal |
| MAST3 | microtubule associated serine/threonine kinase 3 |
| MFGE8 | milk fat globule-EGF factor 8 protein |
| MTCP1 | mature T-cell proliferation 1 |
| MUC7 | mucin 7, secreted |
| MYLK | myosin light chain kinase |
| NABP2 | nucleic acid binding protein 2 |
| NCALD | neurocalcin delta |
| NTSR1 | neurotensin receptor 1 (high affinity) |
| OSMR | oncostatin M receptor |
| P2RY4 | pyrimidinergic receptor P2Y, G-protein coupled, 4 |
| PALM | paralemmin |
| PDPR | pyruvate dehydrogenase phosphatase regulatory subunit |
| PITPNM1 | phosphatidylinositol transfer protein, membrane-associated 1 |
| PLEKHB1 | pleckstrin homology domain containing, family B (evectins) member 1 |
| PLEKHG6 | pleckstrin homology domain containing, family G (with RhoGef domain) member 6 |
| PLXNB3 | plexin B3 |
| POLR3D | polymerase (RNA) III (DNA directed) polypeptide D, 44kDa |
| PRB3 | proline-rich protein BstNI subfamily 3 |
| PREX2 | phosphatidylinositol-3,4,5-trisphosphate-dependent Rac exchange factor 2 |
| RAB3IL1 | RAB3A interacting protein (rabin3)-like 1 |
| RAI2 | retinoic acid induced 2 |
| RASL11B | RAS-like, family 11, member B |
| RPA4 | replication protein A4, 30kDa |
| RSPH14 | radial spoke head 14 homolog (Chlamydomonas) |
| SCN1B | sodium channel, voltage gated, type I beta subunit |
| SERGEF | secretion regulating guanine nucleotide exchange factor |
| SETD1A | SET domain containing 1A |
| SOX21 | SRY (sex determining region Y)-box 21 |
| SP1 | Sp1 transcription factor |
| STRN4 | striatin, calmodulin binding protein 4 |
| SYT17 | synaptotagmin XVII |
| TFAP4 | transcription factor AP-4 (activating enhancer binding protein 4) |
| TNS2 | tensin 2 |
| TOM1 | target of myb1 (chicken) |
| TPST2 | tyrosylprotein sulfotransferase 2 |
| UNC93B1 | unc-93 homolog B1 (C. elegans) |
| UNKL | unkempt family zinc finger-like |
| USB1 | U6 snRNA biogenesis 1 |
| WDR62 | WD repeat domain 62 |
| WFDC2 | WAP four-disulfide core domain 2 |
| WNT10B | wingless-type MMTV integration site family, member 10B |
| XAF1 | XIAP associated factor 1 |
| XDH | xanthine dehydrogenase |
| ZNF222 | zinc finger protein 222 |
| ZNF230 | zinc finger protein 230 |
| ZNF426 | zinc finger protein 426 |
| ZNF492 | zinc finger protein 492 |
| ZNF573 | zinc finger protein 573 |
| ZNF639 | zinc finger protein 639 |
| ZNF768 | zinc finger protein 768 |
| ZNF862 | zinc finger protein 862 |