kawain-2337 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

195 genes differentially expressed following the kawain-2337 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCG2 ATP-binding cassette, sub-family G (WHITE), member 2 (Junior blood group)
ACTA1 actin, alpha 1, skeletal muscle
AGRN agrin
ALDH7A1 aldehyde dehydrogenase 7 family, member A1
CD47 CD47 molecule
CFP complement factor properdin
COL17A1 collagen, type XVII, alpha 1
COL1A1 collagen, type I, alpha 1
CRK v-crk avian sarcoma virus CT10 oncogene homolog
CTSO cathepsin O
CYP2A6 cytochrome P450, family 2, subfamily A, polypeptide 6
CYP2W1 cytochrome P450, family 2, subfamily W, polypeptide 1
DGKA diacylglycerol kinase, alpha 80kDa
DMRT1 doublesex and mab-3 related transcription factor 1
DOHH deoxyhypusine hydroxylase/monooxygenase
EGR1 early growth response 1
FAM102A family with sequence similarity 102, member A
FAM3A family with sequence similarity 3, member A
FERMT1 fermitin family member 1
FGD1 FYVE, RhoGEF and PH domain containing 1
FLT4 fms-related tyrosine kinase 4
FOXG1 forkhead box G1
GAL3ST4 galactose-3-O-sulfotransferase 4
GBP2 guanylate binding protein 2, interferon-inducible
HCFC1R1 host cell factor C1 regulator 1 (XPO1 dependent)
HIST1H2AK histone cluster 1, H2ak
HIST1H3I histone cluster 1, H3i
HOXA10 homeobox A10
HOXD1 homeobox D1
HPCAL4 hippocalcin like 4
HPS4 Hermansky-Pudlak syndrome 4
HSF1 heat shock transcription factor 1
IGHG1 immunoglobulin heavy constant gamma 1 (G1m marker)
IRF2BP1 interferon regulatory factor 2 binding protein 1
KCTD13 potassium channel tetramerization domain containing 13
KHDRBS1 KH domain containing, RNA binding, signal transduction associated 1
KHSRP KH-type splicing regulatory protein
KIF1B kinesin family member 1B
MAPK7 mitogen-activated protein kinase 7
MARK4 MAP/microtubule affinity-regulating kinase 4
MBTPS2 membrane-bound transcription factor peptidase, site 2
MCCC2 methylcrotonoyl-CoA carboxylase 2 (beta)
MEFV Mediterranean fever
MFAP3L microfibrillar-associated protein 3-like
MSRB2 methionine sulfoxide reductase B2
MVK mevalonate kinase
MYO1C myosin IC
NCOA1 nuclear receptor coactivator 1
NDE1 nudE neurodevelopment protein 1
NEDD9 neural precursor cell expressed, developmentally down-regulated 9
NNAT neuronatin
NUMA1 nuclear mitotic apparatus protein 1
OVGP1 oviductal glycoprotein 1, 120kDa
PATZ1 POZ (BTB) and AT hook containing zinc finger 1
PCBP4 poly(rC) binding protein 4
PCGF3 polycomb group ring finger 3
PCNXL2 pecanex-like 2 (Drosophila)
PLA2G5 phospholipase A2, group V
PMP22 peripheral myelin protein 22
PRMT2 protein arginine methyltransferase 2
PRUNE2 prune homolog 2 (Drosophila)
PTPRA protein tyrosine phosphatase, receptor type, A
RAB11FIP3 RAB11 family interacting protein 3 (class II)
RAB11FIP5 RAB11 family interacting protein 5 (class I)
RBM19 RNA binding motif protein 19
RCAN1 regulator of calcineurin 1
RRN3P1 RNA polymerase I transcription factor homolog (S. cerevisiae) pseudogene 1
SCAMP1 secretory carrier membrane protein 1
SH3BP5 SH3-domain binding protein 5 (BTK-associated)
SIGLEC8 sialic acid binding Ig-like lectin 8
SLC6A9 solute carrier family 6 (neurotransmitter transporter, glycine), member 9
SLC7A8 solute carrier family 7 (amino acid transporter light chain, L system), member 8
SLCO2A1 solute carrier organic anion transporter family, member 2A1
SMARCD1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 1
SOS1 son of sevenless homolog 1 (Drosophila)
SPON2 spondin 2, extracellular matrix protein
SRSF1 serine/arginine-rich splicing factor 1
STBD1 starch binding domain 1
STC2 stanniocalcin 2
STX3 syntaxin 3
TIMELESS timeless circadian clock
TMPRSS15 transmembrane protease, serine 15
TRAF3IP3 TRAF3 interacting protein 3
TRAIP TRAF interacting protein
TRD T cell receptor delta locus
TRIM3 tripartite motif containing 3
UBE3B ubiquitin protein ligase E3B
USB1 U6 snRNA biogenesis 1
YIPF4 Yip1 domain family, member 4
YOD1 YOD1 deubiquitinase
ZFYVE16 zinc finger, FYVE domain containing 16
ZNF276 zinc finger protein 276
ZNF337 zinc finger protein 337
ZNF43 zinc finger protein 43
ZNF609 zinc finger protein 609
ZNF675 zinc finger protein 675

decreased expression

Symbol Name
ABHD11 abhydrolase domain containing 11
ACTR8 ARP8 actin-related protein 8 homolog (yeast)
ACVR1 activin A receptor, type I
ADGRE5 adhesion G protein-coupled receptor E5
AEN apoptosis enhancing nuclease
AES amino-terminal enhancer of split
AGO1 argonaute RISC catalytic component 1
ANKZF1 ankyrin repeat and zinc finger domain containing 1
APOL6 apolipoprotein L, 6
ARAF A-Raf proto-oncogene, serine/threonine kinase
ASAP1-IT1 ASAP1 intronic transcript 1
ASPSCR1 alveolar soft part sarcoma chromosome region, candidate 1
ATAD2B ATPase family, AAA domain containing 2B
ATF7IP2 activating transcription factor 7 interacting protein 2
ATG16L1 autophagy related 16-like 1 (S. cerevisiae)
B4GALT2 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 2
BCORL1 BCL6 corepressor-like 1
C11ORF68 chromosome 11 open reading frame 68
C16ORF59 chromosome 16 open reading frame 59
C19ORF40 chromosome 19 open reading frame 40
C1GALT1 core 1 synthase, glycoprotein-N-acetylgalactosamine 3-beta-galactosyltransferase 1
CBL Cbl proto-oncogene, E3 ubiquitin protein ligase
CCDC15 coiled-coil domain containing 15
CLN6 ceroid-lipofuscinosis, neuronal 6, late infantile, variant
DNAJC17 DnaJ (Hsp40) homolog, subfamily C, member 17
DSPP dentin sialophosphoprotein
EDAR ectodysplasin A receptor
EFCAB2 EF-hand calcium binding domain 2
EIF2AK2 eukaryotic translation initiation factor 2-alpha kinase 2
ELP3 elongator acetyltransferase complex subunit 3
EPHX1 epoxide hydrolase 1, microsomal (xenobiotic)
ERMAP erythroblast membrane-associated protein (Scianna blood group)
FAM127A family with sequence similarity 127, member A
FGL2 fibrinogen-like 2
FILIP1L filamin A interacting protein 1-like
FJX1 four jointed box 1 (Drosophila)
FKBPL FK506 binding protein like
FOS FBJ murine osteosarcoma viral oncogene homolog
FUT8 fucosyltransferase 8 (alpha (1,6) fucosyltransferase)
GTF2IRD1 GTF2I repeat domain containing 1
HDAC5 histone deacetylase 5
HIST1H2AJ histone cluster 1, H2aj
HIST1H2BE histone cluster 1, H2be
HP haptoglobin
ICK intestinal cell (MAK-like) kinase
ITPKB inositol-trisphosphate 3-kinase B
JADE3 jade family PHD finger 3
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
KIF18A kinesin family member 18A
KLF1 Kruppel-like factor 1 (erythroid)
LINC00339 long intergenic non-protein coding RNA 339
LINS lines homolog (Drosophila)
LYPLA2P1 lysophospholipase II pseudogene 1
MAP7D1 MAP7 domain containing 1
MARCKSL1 MARCKS-like 1
MCM9 minichromosome maintenance complex component 9
MILR1 mast cell immunoglobulin-like receptor 1
MLPH melanophilin
MUL1 mitochondrial E3 ubiquitin protein ligase 1
MUM1 melanoma associated antigen (mutated) 1
NAT6 N-acetyltransferase 6 (GCN5-related)
NIPAL2 NIPA-like domain containing 2
NPFFR1 neuropeptide FF receptor 1
NPM3 nucleophosmin/nucleoplasmin 3
PARPBP PARP1 binding protein
PDE6C phosphodiesterase 6C, cGMP-specific, cone, alpha prime
PHYH phytanoyl-CoA 2-hydroxylase
PIK3C2B phosphatidylinositol-4-phosphate 3-kinase, catalytic subunit type 2 beta
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PLEKHM2 pleckstrin homology domain containing, family M (with RUN domain) member 2
PPIP5K1 diphosphoinositol pentakisphosphate kinase 1
PRAF2 PRA1 domain family, member 2
PRRC1 proline-rich coiled-coil 1
PRRG4 proline rich Gla (G-carboxyglutamic acid) 4 (transmembrane)
QPRT quinolinate phosphoribosyltransferase
RAB8B RAB8B, member RAS oncogene family
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
RFTN1 raftlin, lipid raft linker 1
RGP1 RGP1 retrograde golgi transport homolog (S. cerevisiae)
RPP38 ribonuclease P/MRP 38kDa subunit
SGTA small glutamine-rich tetratricopeptide repeat (TPR)-containing, alpha
SLC25A22 solute carrier family 25 (mitochondrial carrier: glutamate), member 22
SLC25A40 solute carrier family 25, member 40
SMR3A submaxillary gland androgen regulated protein 3A
SPR sepiapterin reductase (7,8-dihydrobiopterin:NADP+ oxidoreductase)
SPRYD7 SPRY domain containing 7
SYNJ2BP synaptojanin 2 binding protein
TIPARP TCDD-inducible poly(ADP-ribose) polymerase
TLR4 toll-like receptor 4
TMEM212 transmembrane protein 212
TUBA3C tubulin, alpha 3c
UPK3A uroplakin 3A
VILL villin-like
ZNF222 zinc finger protein 222
ZNF250 zinc finger protein 250
ZNF37BP zinc finger protein 37B, pseudogene
ZNF552 zinc finger protein 552
ZNF668 zinc finger protein 668
ZNHIT2 zinc finger, HIT-type containing 2