lidoflazine-6278 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the lidoflazine-6278 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCD1 ATP-binding cassette, sub-family D (ALD), member 1
ABHD17B abhydrolase domain containing 17B
ACVR1B activin A receptor, type IB
ADAM5 ADAM metallopeptidase domain 5 (pseudogene)
ADGRG2 adhesion G protein-coupled receptor G2
AGPAT2 1-acylglycerol-3-phosphate O-acyltransferase 2
ANGEL2 angel homolog 2 (Drosophila)
AOX1 aldehyde oxidase 1
APOD apolipoprotein D
APPBP2 amyloid beta precursor protein (cytoplasmic tail) binding protein 2
ARHGAP26 Rho GTPase activating protein 26
ARR3 arrestin 3, retinal (X-arrestin)
BCAS1 breast carcinoma amplified sequence 1
BCL9 B-cell CLL/lymphoma 9
CABIN1 calcineurin binding protein 1
CDH6 cadherin 6, type 2, K-cadherin (fetal kidney)
CEACAM6 carcinoembryonic antigen-related cell adhesion molecule 6 (non-specific cross reacting antigen)
COA1 cytochrome c oxidase assembly factor 1 homolog (S. cerevisiae)
CSF1R colony stimulating factor 1 receptor
CTAGE9 CTAGE family, member 9
CYLD cylindromatosis (turban tumor syndrome)
DCN decorin
DCSTAMP dendrocyte expressed seven transmembrane protein
DIEXF digestive organ expansion factor homolog (zebrafish)
DNAJC17 DnaJ (Hsp40) homolog, subfamily C, member 17
FABP3 fatty acid binding protein 3, muscle and heart
FN1 fibronectin 1
GLRX3 glutaredoxin 3
GMPR guanosine monophosphate reductase
GNAZ guanine nucleotide binding protein (G protein), alpha z polypeptide
HCFC1 host cell factor C1
HERC6 HECT and RLD domain containing E3 ubiquitin protein ligase family member 6
HIPK2 homeodomain interacting protein kinase 2
HMOX1 heme oxygenase 1
HNRNPUL2 heterogeneous nuclear ribonucleoprotein U-like 2
HOXB5 homeobox B5
HOXC10 homeobox C10
HRH1 histamine receptor H1
ICOS inducible T-cell co-stimulator
IFI6 interferon, alpha-inducible protein 6
IFITM1 interferon induced transmembrane protein 1
IL22 interleukin 22
IL6ST interleukin 6 signal transducer
INCENP inner centromere protein antigens 135/155kDa
INPP5B inositol polyphosphate-5-phosphatase, 75kDa
IRS2 insulin receptor substrate 2
KATNB1 katanin p80 (WD repeat containing) subunit B 1
KCNK12 potassium channel, two pore domain subfamily K, member 12
KLF4 Kruppel-like factor 4 (gut)
LOC257152 uncharacterized LOC257152
LYN LYN proto-oncogene, Src family tyrosine kinase
MALT1 MALT1 paracaspase
MANBA mannosidase, beta A, lysosomal
MAP2K2 mitogen-activated protein kinase kinase 2
MAP4 microtubule-associated protein 4
MARK4 MAP/microtubule affinity-regulating kinase 4
MECP2 methyl CpG binding protein 2
MMP25 matrix metallopeptidase 25
MYOC myocilin, trabecular meshwork inducible glucocorticoid response
NFIB nuclear factor I/B
NMT1 N-myristoyltransferase 1
NPFFR1 neuropeptide FF receptor 1
ONECUT2 one cut homeobox 2
OSBPL10 oxysterol binding protein-like 10
PARP3 poly (ADP-ribose) polymerase family, member 3
PDE3B phosphodiesterase 3B, cGMP-inhibited
PLEKHM1 pleckstrin homology domain containing, family M (with RUN domain) member 1
PLSCR3 phospholipid scramblase 3
PMS2P3 postmeiotic segregation increased 2 pseudogene 3
POU5F1B POU class 5 homeobox 1B
PPP2R3A protein phosphatase 2, regulatory subunit B'', alpha
RBFOX1 RNA binding protein, fox-1 homolog (C. elegans) 1
RPLP2 ribosomal protein, large, P2
SCN11A sodium channel, voltage gated, type XI alpha subunit
SEMA3F sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3F
SEMA4A sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4A
SFI1 Sfi1 homolog, spindle assembly associated (yeast)
SFTPA2 surfactant protein A2
SIPA1L3 signal-induced proliferation-associated 1 like 3
SIX2 SIX homeobox 2
SLC15A2 solute carrier family 15 (oligopeptide transporter), member 2
SMC1A structural maintenance of chromosomes 1A
SPATA5L1 spermatogenesis associated 5-like 1
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5
TAP1 transporter 1, ATP-binding cassette, sub-family B (MDR/TAP)
TMEM259 transmembrane protein 259
TOP3B topoisomerase (DNA) III beta
TRIM29 tripartite motif containing 29
TSPAN9 tetraspanin 9
TTC28 tetratricopeptide repeat domain 28
UBOX5 U-box domain containing 5
USP48 ubiquitin specific peptidase 48
UTRN utrophin
VAMP4 vesicle-associated membrane protein 4
VAPB VAMP (vesicle-associated membrane protein)-associated protein B and C
WHSC1L1 Wolf-Hirschhorn syndrome candidate 1-like 1
ZNF37BP zinc finger protein 37B, pseudogene
ZNF500 zinc finger protein 500

decreased expression

Symbol Name
ABCA11P ATP-binding cassette, sub-family A (ABC1), member 11, pseudogene
ACTR8 ARP8 actin-related protein 8 homolog (yeast)
AHCTF1 AT hook containing transcription factor 1
ANKEF1 ankyrin repeat and EF-hand domain containing 1
AP1AR adaptor-related protein complex 1 associated regulatory protein
ARHGEF5 Rho guanine nucleotide exchange factor (GEF) 5
BAK1 BCL2-antagonist/killer 1
BBS10 Bardet-Biedl syndrome 10
BBS7 Bardet-Biedl syndrome 7
BCL2L2 BCL2-like 2
C11ORF95 chromosome 11 open reading frame 95
C1ORF35 chromosome 1 open reading frame 35
C6ORF47 chromosome 6 open reading frame 47
CAPN15 calpain 15
CCDC15 coiled-coil domain containing 15
CLCN5 chloride channel, voltage-sensitive 5
CLDN4 claudin 4
COCH cochlin
CRY1 cryptochrome circadian clock 1
CYP27B1 cytochrome P450, family 27, subfamily B, polypeptide 1
CYP2J2 cytochrome P450, family 2, subfamily J, polypeptide 2
DCAF10 DDB1 and CUL4 associated factor 10
DNAJC3 DnaJ (Hsp40) homolog, subfamily C, member 3
EIF4ENIF1 eukaryotic translation initiation factor 4E nuclear import factor 1
ERCC4 excision repair cross-complementation group 4
EVPL envoplakin
F8 coagulation factor VIII, procoagulant component
FAM114A2 family with sequence similarity 114, member A2
FAM50B family with sequence similarity 50, member B
FBRS fibrosin
FCHO1 FCH domain only 1
FKBP14 FK506 binding protein 14, 22 kDa
GALT galactose-1-phosphate uridylyltransferase
GLI3 GLI family zinc finger 3
GNG4 guanine nucleotide binding protein (G protein), gamma 4
H2AFY2 H2A histone family, member Y2
HIST1H4J histone cluster 1, H4j
HYAL2 hyaluronoglucosaminidase 2
IFT81 intraflagellar transport 81
IL15RA interleukin 15 receptor, alpha
INF2 inverted formin, FH2 and WH2 domain containing
IREB2 iron-responsive element binding protein 2
KDM5C lysine (K)-specific demethylase 5C
KIAA0355 KIAA0355
KRBOX4 KRAB box domain containing 4
LEMD3 LEM domain containing 3
LRP5 low density lipoprotein receptor-related protein 5
LRRC8E leucine rich repeat containing 8 family, member E
MANEA mannosidase, endo-alpha
MAP4K3 mitogen-activated protein kinase kinase kinase kinase 3
MBTD1 mbt domain containing 1
MGAT1 mannosyl (alpha-1,3-)-glycoprotein beta-1,2-N-acetylglucosaminyltransferase
MKNK2 MAP kinase interacting serine/threonine kinase 2
MMP9 matrix metallopeptidase 9
MYL12A myosin, light chain 12A, regulatory, non-sarcomeric
NAA38 N(alpha)-acetyltransferase 38, NatC auxiliary subunit
NEK11 NIMA-related kinase 11
NPIPB15 nuclear pore complex interacting protein family, member B15
NUDT13 nudix (nucleoside diphosphate linked moiety X)-type motif 13
P3H1 prolyl 3-hydroxylase 1
PC pyruvate carboxylase
POTEKP POTE ankyrin domain family, member K, pseudogene
PRKX protein kinase, X-linked
PTPN13 protein tyrosine phosphatase, non-receptor type 13 (APO-1/CD95 (Fas)-associated phosphatase)
PTPRG protein tyrosine phosphatase, receptor type, G
PYCRL pyrroline-5-carboxylate reductase-like
RAC3 ras-related C3 botulinum toxin substrate 3 (rho family, small GTP binding protein Rac3)
RAD51AP1 RAD51 associated protein 1
RBL1 retinoblastoma-like 1
RECQL4 RecQ protein-like 4
RFTN1 raftlin, lipid raft linker 1
RIPK4 receptor-interacting serine-threonine kinase 4
RNF25 ring finger protein 25
RNF39 ring finger protein 39
SCUBE2 signal peptide, CUB domain, EGF-like 2
SCYL2 SCY1-like 2 (S. cerevisiae)
SECTM1 secreted and transmembrane 1
SERTAD3 SERTA domain containing 3
SETD6 SET domain containing 6
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC41A3 solute carrier family 41, member 3
SLC4A8 solute carrier family 4, sodium bicarbonate cotransporter, member 8
STBD1 starch binding domain 1
TEAD3 TEA domain family member 3
TESK1 testis-specific kinase 1
TMEM254 transmembrane protein 254
TOLLIP toll interacting protein
TRABD TraB domain containing
TRMU tRNA 5-methylaminomethyl-2-thiouridylate methyltransferase
TTC23 tetratricopeptide repeat domain 23
VCPKMT valosin containing protein lysine (K) methyltransferase
WDR19 WD repeat domain 19
WLS wntless Wnt ligand secretion mediator
ZBTB10 zinc finger and BTB domain containing 10
ZKSCAN3 zinc finger with KRAB and SCAN domains 3
ZKSCAN4 zinc finger with KRAB and SCAN domains 4
ZNF205 zinc finger protein 205
ZNF787 zinc finger protein 787