meclozine-2424 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the meclozine-2424 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABCG1 ATP-binding cassette, sub-family G (WHITE), member 1
ACSBG2 acyl-CoA synthetase bubblegum family member 2
ACTN2 actinin, alpha 2
ADCY9 adenylate cyclase 9
ADGRB1 adhesion G protein-coupled receptor B1
AFF1 AF4/FMR2 family, member 1
AGGF1 angiogenic factor with G patch and FHA domains 1
ANGEL2 angel homolog 2 (Drosophila)
ANGPT2 angiopoietin 2
ANXA2P3 annexin A2 pseudogene 3
APOC4 apolipoprotein C-IV
ATP10B ATPase, class V, type 10B
AURKA aurora kinase A
CA5B carbonic anhydrase VB, mitochondrial
CASP10 caspase 10, apoptosis-related cysteine peptidase
CBR3 carbonyl reductase 3
CCL27 chemokine (C-C motif) ligand 27
CD34 CD34 molecule
CD84 CD84 molecule
CDC25C cell division cycle 25C
CEBPD CCAAT/enhancer binding protein (C/EBP), delta
CEP170B centrosomal protein 170B
COX11 COX11 cytochrome c oxidase copper chaperone
CREBBP CREB binding protein
CRH corticotropin releasing hormone
CRHR2 corticotropin releasing hormone receptor 2
EDA ectodysplasin A
EIF5A2 eukaryotic translation initiation factor 5A2
EPHB1 EPH receptor B1
FLOT1 flotillin 1
FXYD2 FXYD domain containing ion transport regulator 2
GAL galanin/GMAP prepropeptide
GAS8 growth arrest-specific 8
GLYR1 glyoxylate reductase 1 homolog (Arabidopsis)
HOXA11 homeobox A11
IDS iduronate 2-sulfatase
IFIT2 interferon-induced protein with tetratricopeptide repeats 2
IFT122 intraflagellar transport 122
INPP5J inositol polyphosphate-5-phosphatase J
KAZALD1 Kazal-type serine peptidase inhibitor domain 1
KIF1C kinesin family member 1C
MAOA monoamine oxidase A
MED16 mediator complex subunit 16
MSC musculin
NADK NAD kinase
NKX3-1 NK3 homeobox 1
OASL 2'-5'-oligoadenylate synthetase-like
OR1D2 olfactory receptor, family 1, subfamily D, member 2
OR2H2 olfactory receptor, family 2, subfamily H, member 2
PAX5 paired box 5
PDE4DIP phosphodiesterase 4D interacting protein
PIP4K2B phosphatidylinositol-5-phosphate 4-kinase, type II, beta
PLA2G3 phospholipase A2, group III
PLEKHF1 pleckstrin homology domain containing, family F (with FYVE domain) member 1
PML promyelocytic leukemia
PPP1R12B protein phosphatase 1, regulatory subunit 12B
PPT2 palmitoyl-protein thioesterase 2
PQLC2 PQ loop repeat containing 2
PRKCQ protein kinase C, theta
PRPF18 pre-mRNA processing factor 18
PSG1 pregnancy specific beta-1-glycoprotein 1
PTPRJ protein tyrosine phosphatase, receptor type, J
RAB13 RAB13, member RAS oncogene family
RAB3GAP2 RAB3 GTPase activating protein subunit 2 (non-catalytic)
RAB40B RAB40B, member RAS oncogene family
RASAL2 RAS protein activator like 2
RND1 Rho family GTPase 1
RNF6 ring finger protein (C3H2C3 type) 6
SEMA3A sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3A
SEMA6D sema domain, transmembrane domain (TM), and cytoplasmic domain, (semaphorin) 6D
SGCD sarcoglycan, delta (35kDa dystrophin-associated glycoprotein)
SH3BGR SH3 domain binding glutamate-rich protein
SIRPB1 signal-regulatory protein beta 1
SLC22A5 solute carrier family 22 (organic cation/carnitine transporter), member 5
SLC2A8 solute carrier family 2 (facilitated glucose transporter), member 8
SMARCA4 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 4
SMG7 SMG7 nonsense mediated mRNA decay factor
SOX4 SRY (sex determining region Y)-box 4
ST6GALNAC4 ST6 (alpha-N-acetyl-neuraminyl-2,3-beta-galactosyl-1,3)-N-acetylgalactosaminide alpha-2,6-sialyltransferase 4
STAB2 stabilin 2
TAPT1 transmembrane anterior posterior transformation 1
TAS2R1 taste receptor, type 2, member 1
TBX6 T-box 6
TCP10L t-complex 10-like
TGFBR2 transforming growth factor, beta receptor II (70/80kDa)
TMEM212 transmembrane protein 212
TONSL tonsoku-like, DNA repair protein
TP53I11 tumor protein p53 inducible protein 11
TRIM10 tripartite motif containing 10
TSC22D2 TSC22 domain family, member 2
UBOX5 U-box domain containing 5
VPS33A vacuolar protein sorting 33 homolog A (S. cerevisiae)
YLPM1 YLP motif containing 1
ZFHX4 zinc finger homeobox 4
ZFYVE9 zinc finger, FYVE domain containing 9
ZNF492 zinc finger protein 492
ZNF93 zinc finger protein 93

decreased expression

Symbol Name
AIM2 absent in melanoma 2
ASB7 ankyrin repeat and SOCS box containing 7
ATHL1 ATH1, acid trehalase-like 1 (yeast)
B3GNT1
BAG4 BCL2-associated athanogene 4
CDK6 cyclin-dependent kinase 6
CHMP7 charged multivesicular body protein 7
CHPF chondroitin polymerizing factor
CHRNA10 cholinergic receptor, nicotinic, alpha 10 (neuronal)
CRELD1 cysteine-rich with EGF-like domains 1
CRY2 cryptochrome circadian clock 2
DGKG diacylglycerol kinase, gamma 90kDa
DOK3 docking protein 3
DTX4 deltex 4, E3 ubiquitin ligase
DZANK1 double zinc ribbon and ankyrin repeat domains 1
EFNA3 ephrin-A3
EMILIN2 elastin microfibril interfacer 2
FAM127B family with sequence similarity 127, member B
FAM204A family with sequence similarity 204, member A
FBRS fibrosin
FSTL3 follistatin-like 3 (secreted glycoprotein)
GPR85 G protein-coupled receptor 85
HERC6 HECT and RLD domain containing E3 ubiquitin protein ligase family member 6
IGFLR1 IGF-like family receptor 1
INO80D INO80 complex subunit D
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
KLHL21 kelch-like family member 21
KLHL28 kelch-like family member 28
LOC257152 uncharacterized LOC257152
LPAR6 lysophosphatidic acid receptor 6
LYPLA2P1 lysophospholipase II pseudogene 1
LZTS3 leucine zipper, putative tumor suppressor family member 3
MCOLN1 mucolipin 1
METTL21B methyltransferase like 21B
MICAL3 microtubule associated monooxygenase, calponin and LIM domain containing 3
MKL2 MKL/myocardin-like 2
MPZ myelin protein zero
MREG melanoregulin
MRPL44 mitochondrial ribosomal protein L44
MYBBP1A MYB binding protein (P160) 1a
NECAB3 N-terminal EF-hand calcium binding protein 3
NINJ2 ninjurin 2
OPLAH 5-oxoprolinase (ATP-hydrolysing)
OTUD3 OTU deubiquitinase 3
OXCT2 3-oxoacid CoA transferase 2
PADI2 peptidyl arginine deiminase, type II
PBLD phenazine biosynthesis-like protein domain containing
PCYT2 phosphate cytidylyltransferase 2, ethanolamine
PEX26 peroxisomal biogenesis factor 26
PGGT1B protein geranylgeranyltransferase type I, beta subunit
PHC1 polyhomeotic homolog 1 (Drosophila)
PIK3R2 phosphoinositide-3-kinase, regulatory subunit 2 (beta)
PLA2G12A phospholipase A2, group XIIA
PMFBP1 polyamine modulated factor 1 binding protein 1
PPFIA4 protein tyrosine phosphatase, receptor type, f polypeptide (PTPRF), interacting protein (liprin), alpha 4
PVRL2 poliovirus receptor-related 2 (herpesvirus entry mediator B)
PWAR5 Prader Willi/Angelman region RNA 5
RAB17 RAB17, member RAS oncogene family
RAB3A RAB3A, member RAS oncogene family
RHBDF1 rhomboid 5 homolog 1 (Drosophila)
RIN1 Ras and Rab interactor 1
RNF122 ring finger protein 122
RPA4 replication protein A4, 30kDa
SETD1A SET domain containing 1A
SH2D4A SH2 domain containing 4A
SHARPIN SHANK-associated RH domain interactor
SLC20A2 solute carrier family 20 (phosphate transporter), member 2
SLC27A3 solute carrier family 27 (fatty acid transporter), member 3
SLC31A2 solute carrier family 31 (copper transporter), member 2
SLC38A10 solute carrier family 38, member 10
SLCO4A1 solute carrier organic anion transporter family, member 4A1
SPR sepiapterin reductase (7,8-dihydrobiopterin:NADP+ oxidoreductase)
TAGLN transgelin
TCTN2 tectonic family member 2
TESK1 testis-specific kinase 1
TIMP2 TIMP metallopeptidase inhibitor 2
TRAIP TRAF interacting protein
TRANK1 tetratricopeptide repeat and ankyrin repeat containing 1
TRDMT1 tRNA aspartic acid methyltransferase 1
TRIM36 tripartite motif containing 36
TSC22D4 TSC22 domain family, member 4
TSPAN32 tetraspanin 32
TTLL1 tubulin tyrosine ligase-like family member 1
TTPAL tocopherol (alpha) transfer protein-like
TUBA4B tubulin, alpha 4b
VEGFB vascular endothelial growth factor B
WDR62 WD repeat domain 62
ZBED8 zinc finger, BED-type containing 8
ZDHHC24 zinc finger, DHHC-type containing 24
ZMAT5 zinc finger, matrin-type 5
ZNF155 zinc finger protein 155
ZNF219 zinc finger protein 219
ZNF226 zinc finger protein 226
ZNF354A zinc finger protein 354A
ZNF493 zinc finger protein 493
ZNF528 zinc finger protein 528
ZNF580 zinc finger protein 580
ZNF816 zinc finger protein 816