metacycline-4062 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the metacycline-4062 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADRA1A adrenoceptor alpha 1A
AGTR1 angiotensin II receptor, type 1
AKAP6 A kinase (PRKA) anchor protein 6
ALDH3B2 aldehyde dehydrogenase 3 family, member B2
ANGPT4 angiopoietin 4
AUTS2 autism susceptibility candidate 2
B4GALT1 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 1
BAAT bile acid CoA:amino acid N-acyltransferase
BEGAIN brain-enriched guanylate kinase-associated
BRINP2 bone morphogenetic protein/retinoic acid inducible neural-specific 2
BTNL3 butyrophilin-like 3
C17ORF59 chromosome 17 open reading frame 59
C2CD2L C2CD2-like
C5AR2 complement component 5a receptor 2
CCDC134 coiled-coil domain containing 134
CCDC170 coiled-coil domain containing 170
CCL22 chemokine (C-C motif) ligand 22
CD5 CD5 molecule
CHRNA1 cholinergic receptor, nicotinic, alpha 1 (muscle)
CHRNE cholinergic receptor, nicotinic, epsilon (muscle)
CLPS colipase, pancreatic
COL11A1 collagen, type XI, alpha 1
COL14A1 collagen, type XIV, alpha 1
COL21A1 collagen, type XXI, alpha 1
CSF1R colony stimulating factor 1 receptor
CSF2RB colony stimulating factor 2 receptor, beta, low-affinity (granulocyte-macrophage)
CYTH1 cytohesin 1
CYTH4 cytohesin 4
DCTN1 dynactin 1
DICER1 dicer 1, ribonuclease type III
EXOSC1 exosome component 1
FGF4 fibroblast growth factor 4
FRMD4B FERM domain containing 4B
GAD2 glutamate decarboxylase 2 (pancreatic islets and brain, 65kDa)
GJA8 gap junction protein, alpha 8, 50kDa
GLB1L galactosidase, beta 1-like
GPR157 G protein-coupled receptor 157
GSPT1 G1 to S phase transition 1
HFE hemochromatosis
HHIPL2 HHIP-like 2
HOXD13 homeobox D13
HP haptoglobin
HRH4 histamine receptor H4
HSD3B2 hydroxy-delta-5-steroid dehydrogenase, 3 beta- and steroid delta-isomerase 2
IHH indian hedgehog
INSR insulin receptor
ITGB4 integrin, beta 4
KIF1A kinesin family member 1A
KLHL4 kelch-like family member 4
KRT16 keratin 16, type I
LAMB4 laminin, beta 4
MME membrane metallo-endopeptidase
MTRF1L mitochondrial translational release factor 1-like
NOP14-AS1 NOP14 antisense RNA 1
NR1H4 nuclear receptor subfamily 1, group H, member 4
NRG2 neuregulin 2
OMD osteomodulin
OR2B6 olfactory receptor, family 2, subfamily B, member 6
PCDHA9 protocadherin alpha 9
PDE10A phosphodiesterase 10A
PDE12 phosphodiesterase 12
PDE4D phosphodiesterase 4D, cAMP-specific
PHYHIP phytanoyl-CoA 2-hydroxylase interacting protein
PLA2G3 phospholipase A2, group III
PMFBP1 polyamine modulated factor 1 binding protein 1
POU2F3 POU class 2 homeobox 3
PPARD peroxisome proliferator-activated receptor delta
PPIL2 peptidylprolyl isomerase (cyclophilin)-like 2
PPP1R2P9 protein phosphatase 1, regulatory (inhibitor) subunit 2 pseudogene 9
PPP1R37 protein phosphatase 1, regulatory subunit 37
PRB1 proline-rich protein BstNI subfamily 1
PTBP3 polypyrimidine tract binding protein 3
PTPN1 protein tyrosine phosphatase, non-receptor type 1
RIF1 replication timing regulatory factor 1
RPS14 ribosomal protein S14
SARM1 sterile alpha and TIR motif containing 1
SEC14L4 SEC14-like 4 (S. cerevisiae)
SEMA3E sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3E
SFTPB surfactant protein B
SLC12A4 solute carrier family 12 (potassium/chloride transporter), member 4
SLC6A16 solute carrier family 6, member 16
SPRED2 sprouty-related, EVH1 domain containing 2
SSTR5 somatostatin receptor 5
STOML1 stomatin (EPB72)-like 1
SULT2A1 sulfotransferase family, cytosolic, 2A, dehydroepiandrosterone (DHEA)-preferring, member 1
SULT2B1 sulfotransferase family, cytosolic, 2B, member 1
TBC1D2B TBC1 domain family, member 2B
TFCP2L1 transcription factor CP2-like 1
TMEM257 transmembrane protein 257
TNFRSF9 tumor necrosis factor receptor superfamily, member 9
TPSAB1 tryptase alpha/beta 1
TRIM15 tripartite motif containing 15
VNN2 vanin 2
VPRBP Vpr (HIV-1) binding protein
WNT2B wingless-type MMTV integration site family, member 2B
WT1-AS WT1 antisense RNA
XIST X inactive specific transcript (non-protein coding)
ZNF155 zinc finger protein 155
ZNF391 zinc finger protein 391
ZNF484 zinc finger protein 484

decreased expression

Symbol Name
ABCC6 ATP-binding cassette, sub-family C (CFTR/MRP), member 6
ADAM23 ADAM metallopeptidase domain 23
ANP32A-IT1 ANP32A intronic transcript 1
APOLD1 apolipoprotein L domain containing 1
ARHGEF16 Rho guanine nucleotide exchange factor (GEF) 16
ARHGEF38 Rho guanine nucleotide exchange factor (GEF) 38
BIRC3 baculoviral IAP repeat containing 3
BTC betacellulin
C3AR1 complement component 3a receptor 1
CA11 carbonic anhydrase XI
CAMTA2 calmodulin binding transcription activator 2
CDADC1 cytidine and dCMP deaminase domain containing 1
CFAP45 cilia and flagella associated protein 45
CHRNA9 cholinergic receptor, nicotinic, alpha 9 (neuronal)
CLIC3 chloride intracellular channel 3
CYB5R2 cytochrome b5 reductase 2
DGCR11 DiGeorge syndrome critical region gene 11 (non-protein coding)
DMTN dematin actin binding protein
DNM3 dynamin 3
DPYS dihydropyrimidinase
EFNA3 ephrin-A3
EFNB1 ephrin-B1
EN1 engrailed homeobox 1
EPPK1 epiplakin 1
ERCC2 excision repair cross-complementation group 2
FAM110B family with sequence similarity 110, member B
FBXO22 F-box protein 22
FBXO31 F-box protein 31
GNA14 guanine nucleotide binding protein (G protein), alpha 14
GPC3 glypican 3
GPRIN2 G protein regulated inducer of neurite outgrowth 2
GRM4 glutamate receptor, metabotropic 4
HOXA6 homeobox A6
HSF2BP heat shock transcription factor 2 binding protein
HTR1D 5-hydroxytryptamine (serotonin) receptor 1D, G protein-coupled
IFT140 intraflagellar transport 140
IFT54 intraflagellar transport 54
IL12A interleukin 12A
IL22 interleukin 22
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNS1 potassium voltage-gated channel, modifier subfamily S, member 1
KCNS3 potassium voltage-gated channel, modifier subfamily S, member 3
KIFC3 kinesin family member C3
KLF13 Kruppel-like factor 13
LIME1 Lck interacting transmembrane adaptor 1
LRP5L low density lipoprotein receptor-related protein 5-like
LRRC2 leucine rich repeat containing 2
MAN2C1 mannosidase, alpha, class 2C, member 1
MATN3 matrilin 3
MED15 mediator complex subunit 15
MTCP1 mature T-cell proliferation 1
MTSS1L metastasis suppressor 1-like
NAT6 N-acetyltransferase 6 (GCN5-related)
NGF nerve growth factor (beta polypeptide)
NKX3-2 NK3 homeobox 2
NOD1 nucleotide-binding oligomerization domain containing 1
NRTN neurturin
OR1D2 olfactory receptor, family 1, subfamily D, member 2
OSMR oncostatin M receptor
OXCT2 3-oxoacid CoA transferase 2
PID1 phosphotyrosine interaction domain containing 1
PLA2G1B phospholipase A2, group IB (pancreas)
PLD3 phospholipase D family, member 3
PLXNB3 plexin B3
PRSS12 protease, serine, 12 (neurotrypsin, motopsin)
PTK6 protein tyrosine kinase 6
RGCC regulator of cell cycle
RSPH14 radial spoke head 14 homolog (Chlamydomonas)
S1PR1 sphingosine-1-phosphate receptor 1
SCN1B sodium channel, voltage gated, type I beta subunit
SLC16A6 solute carrier family 16, member 6
SLC18A2 solute carrier family 18 (vesicular monoamine transporter), member 2
SMPDL3B sphingomyelin phosphodiesterase, acid-like 3B
SOD3 superoxide dismutase 3, extracellular
SSTR4 somatostatin receptor 4
STEAP4 STEAP family member 4
TAS2R10 taste receptor, type 2, member 10
TBC1D17 TBC1 domain family, member 17
TBKBP1 TBK1 binding protein 1
THSD4 thrombospondin, type I, domain containing 4
TINAGL1 tubulointerstitial nephritis antigen-like 1
TNFRSF14 tumor necrosis factor receptor superfamily, member 14
TRAF2 TNF receptor-associated factor 2
TRIM45 tripartite motif containing 45
TRPM4 transient receptor potential cation channel, subfamily M, member 4
VWA1 von Willebrand factor A domain containing 1
WDR62 WD repeat domain 62
XAB2 XPA binding protein 2
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZFP30 ZFP30 zinc finger protein
ZNF219 zinc finger protein 219
ZNF37BP zinc finger protein 37B, pseudogene
ZNF549 zinc finger protein 549
ZNF749 zinc finger protein 749
ZNF76 zinc finger protein 76
ZNF768 zinc finger protein 768