methapyrilene-1588 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the methapyrilene-1588 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AHNAK AHNAK nucleoprotein
AKAP13 A kinase (PRKA) anchor protein 13
AKAP7 A kinase (PRKA) anchor protein 7
ALPK1 alpha-kinase 1
ANXA2P2 annexin A2 pseudogene 2
AP3S2 adaptor-related protein complex 3, sigma 2 subunit
APOBEC3C apolipoprotein B mRNA editing enzyme, catalytic polypeptide-like 3C
ATG13 autophagy related 13
BCLAF1 BCL2-associated transcription factor 1
C22ORF29 chromosome 22 open reading frame 29
CBLB Cbl proto-oncogene B, E3 ubiquitin protein ligase
CCDC40 coiled-coil domain containing 40
CD164 CD164 molecule, sialomucin
CD3EAP CD3e molecule, epsilon associated protein
CNPY3 canopy FGF signaling regulator 3
CNTFR ciliary neurotrophic factor receptor
CREB1 cAMP responsive element binding protein 1
DDX28 DEAD (Asp-Glu-Ala-Asp) box polypeptide 28
ECM1 extracellular matrix protein 1
EEF1D eukaryotic translation elongation factor 1 delta (guanine nucleotide exchange protein)
ELF4 E74-like factor 4 (ets domain transcription factor)
EMD emerin
EPS8L1 EPS8-like 1
FAM162A family with sequence similarity 162, member A
FBLN1 fibulin 1
FBXL18 F-box and leucine-rich repeat protein 18
FOLR1 folate receptor 1 (adult)
FRMD4B FERM domain containing 4B
FZD2 frizzled class receptor 2
GOLGA1 golgin A1
GRM4 glutamate receptor, metabotropic 4
GSK3A glycogen synthase kinase 3 alpha
GSTA4 glutathione S-transferase alpha 4
HADHA hydroxyacyl-CoA dehydrogenase/3-ketoacyl-CoA thiolase/enoyl-CoA hydratase (trifunctional protein), alpha subunit
HSPB11 heat shock protein family B (small), member 11
HYI hydroxypyruvate isomerase (putative)
IMPAD1 inositol monophosphatase domain containing 1
KLHL24 kelch-like family member 24
KPTN kaptin (actin binding protein)
KRT38 keratin 38, type I
LDLRAD4 low density lipoprotein receptor class A domain containing 4
LENEP lens epithelial protein
MACF1 microtubule-actin crosslinking factor 1
MAPK10 mitogen-activated protein kinase 10
MED16 mediator complex subunit 16
METAP2 methionyl aminopeptidase 2
MICALL2 MICAL-like 2
MMP19 matrix metallopeptidase 19
MOSPD2 motile sperm domain containing 2
MR1 major histocompatibility complex, class I-related
MTRF1L mitochondrial translational release factor 1-like
MUC5AC mucin 5AC, oligomeric mucus/gel-forming
MXRA8 matrix-remodelling associated 8
MYL10 myosin, light chain 10, regulatory
MYO1C myosin IC
N4BP2L2 NEDD4 binding protein 2-like 2
NOP16 NOP16 nucleolar protein
NPPA natriuretic peptide A
OR3A3 olfactory receptor, family 3, subfamily A, member 3
PAXBP1 PAX3 and PAX7 binding protein 1
PCIF1 PDX1 C-terminal inhibiting factor 1
PICALM phosphatidylinositol binding clathrin assembly protein
PLCB4 phospholipase C, beta 4
PLD2 phospholipase D2
PLOD1 procollagen-lysine, 2-oxoglutarate 5-dioxygenase 1
POLR3F polymerase (RNA) III (DNA directed) polypeptide F, 39 kDa
PTCRA pre T-cell antigen receptor alpha
PTMA prothymosin, alpha
PTPRU protein tyrosine phosphatase, receptor type, U
RAB6B RAB6B, member RAS oncogene family
RBM19 RNA binding motif protein 19
RECK reversion-inducing-cysteine-rich protein with kazal motifs
RHOT2 ras homolog family member T2
RIOK3 RIO kinase 3
RIPK1 receptor (TNFRSF)-interacting serine-threonine kinase 1
RNF144A ring finger protein 144A
RPS11 ribosomal protein S11
SAFB scaffold attachment factor B
SETD4 SET domain containing 4
SH3BP2 SH3-domain binding protein 2
SLC25A44 solute carrier family 25, member 44
SNAP25 synaptosomal-associated protein, 25kDa
SNTB1 syntrophin, beta 1 (dystrophin-associated protein A1, 59kDa, basic component 1)
SPATA5L1 spermatogenesis associated 5-like 1
SPG7 spastic paraplegia 7 (pure and complicated autosomal recessive)
SPOCK2 sparc/osteonectin, cwcv and kazal-like domains proteoglycan (testican) 2
STX7 syntaxin 7
TBC1D2B TBC1 domain family, member 2B
TK2 thymidine kinase 2, mitochondrial
TOPORS topoisomerase I binding, arginine/serine-rich, E3 ubiquitin protein ligase
TRPM3 transient receptor potential cation channel, subfamily M, member 3
TSR1 TSR1, 20S rRNA accumulation, homolog (S. cerevisiae)
UBQLN4 ubiquilin 4
USP46 ubiquitin specific peptidase 46
VILL villin-like
YBX3 Y box binding protein 3
YIPF2 Yip1 domain family, member 2
ZNF721 zinc finger protein 721
ZNF93 zinc finger protein 93

decreased expression

Symbol Name
AATF apoptosis antagonizing transcription factor
ACADVL acyl-CoA dehydrogenase, very long chain
ACP2 acid phosphatase 2, lysosomal
ADAT1 adenosine deaminase, tRNA-specific 1
APOBR apolipoprotein B receptor
BCKDK branched chain ketoacid dehydrogenase kinase
C1ORF54 chromosome 1 open reading frame 54
CASZ1 castor zinc finger 1
CCNT1 cyclin T1
CD151 CD151 molecule (Raph blood group)
CD248 CD248 molecule, endosialin
CD69 CD69 molecule
CDKN1A cyclin-dependent kinase inhibitor 1A (p21, Cip1)
CFAP74 cilia and flagella associated protein 74
CLPB ClpB homolog, mitochondrial AAA ATPase chaperonin
CPNE1 copine I
CPOX coproporphyrinogen oxidase
CSAD cysteine sulfinic acid decarboxylase
CSTF3 cleavage stimulation factor, 3' pre-RNA, subunit 3, 77kDa
CTDNEP1 CTD nuclear envelope phosphatase 1
CTNNAL1 catenin (cadherin-associated protein), alpha-like 1
DNAJC3 DnaJ (Hsp40) homolog, subfamily C, member 3
DOLK dolichol kinase
EFTUD1 elongation factor Tu GTP binding domain containing 1
EMP3 epithelial membrane protein 3
FAM114A1 family with sequence similarity 114, member A1
FAM160B2 family with sequence similarity 160, member B2
FBXL14 F-box and leucine-rich repeat protein 14
FTH1P5 ferritin, heavy polypeptide 1 pseudogene 5
FTO fat mass and obesity associated
FURIN furin (paired basic amino acid cleaving enzyme)
GABARAPL2 GABA(A) receptor-associated protein-like 2
GDAP2 ganglioside induced differentiation associated protein 2
GNG3 guanine nucleotide binding protein (G protein), gamma 3
GPR137B G protein-coupled receptor 137B
HACD2 3-hydroxyacyl-CoA dehydratase 2
HP haptoglobin
HSPA4L heat shock 70kDa protein 4-like
IFIT1 interferon-induced protein with tetratricopeptide repeats 1
IFITM3 interferon induced transmembrane protein 3
KIF13B kinesin family member 13B
LIN37 lin-37 DREAM MuvB core complex component
LSP1 lymphocyte-specific protein 1
MADCAM1 mucosal vascular addressin cell adhesion molecule 1
MFSD11 major facilitator superfamily domain containing 11
MGAT1 mannosyl (alpha-1,3-)-glycoprotein beta-1,2-N-acetylglucosaminyltransferase
MSL2 male-specific lethal 2 homolog (Drosophila)
MUTYH mutY homolog
NARS2 asparaginyl-tRNA synthetase 2, mitochondrial (putative)
NHLRC2 NHL repeat containing 2
NME3 NME/NM23 nucleoside diphosphate kinase 3
NSF N-ethylmaleimide-sensitive factor
NTHL1 nth endonuclease III-like 1 (E. coli)
OCEL1 occludin/ELL domain containing 1
PCDHGB5 protocadherin gamma subfamily B, 5
PELI2 pellino E3 ubiquitin protein ligase family member 2
PEMT phosphatidylethanolamine N-methyltransferase
PIBF1 progesterone immunomodulatory binding factor 1
PODNL1 podocan-like 1
POLA2 polymerase (DNA directed), alpha 2, accessory subunit
PRCC papillary renal cell carcinoma (translocation-associated)
PUS7 pseudouridylate synthase 7 (putative)
PVRL2 poliovirus receptor-related 2 (herpesvirus entry mediator B)
QTRTD1 queuine tRNA-ribosyltransferase domain containing 1
RAB4B RAB4B, member RAS oncogene family
RAPGEF6 Rap guanine nucleotide exchange factor (GEF) 6
REPIN1 replication initiator 1
RIC8A RIC8 guanine nucleotide exchange factor A
RMDN3 regulator of microtubule dynamics 3
SASH3 SAM and SH3 domain containing 3
SCD5 stearoyl-CoA desaturase 5
SEMA4A sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4A
SHPK sedoheptulokinase
SLC12A2 solute carrier family 12 (sodium/potassium/chloride transporter), member 2
SLC12A7 solute carrier family 12 (potassium/chloride transporter), member 7
SLC22A18 solute carrier family 22, member 18
SLC25A28 solute carrier family 25 (mitochondrial iron transporter), member 28
SLC7A7 solute carrier family 7 (amino acid transporter light chain, y+L system), member 7
STK39 serine threonine kinase 39
TAF4B TAF4b RNA polymerase II, TATA box binding protein (TBP)-associated factor, 105kDa
TBL3 transducin (beta)-like 3
TESK2 testis-specific kinase 2
TMEM177 transmembrane protein 177
TRIM22 tripartite motif containing 22
TRMT12 tRNA methyltransferase 12 homolog (S. cerevisiae)
TTI1 TELO2 interacting protein 1
TYW1 tRNA-yW synthesizing protein 1 homolog (S. cerevisiae)
UGDH UDP-glucose 6-dehydrogenase
USB1 U6 snRNA biogenesis 1
VASP vasodilator-stimulated phosphoprotein
WBSCR16 Williams-Beuren syndrome chromosome region 16
WDR41 WD repeat domain 41
WDR46 WD repeat domain 46
WDR82 WD repeat domain 82
XRCC1 X-ray repair complementing defective repair in Chinese hamster cells 1
ZEB2 zinc finger E-box binding homeobox 2
ZNF107 zinc finger protein 107
ZNF16 zinc finger protein 16
ZNF804A zinc finger protein 804A
ZSCAN5A zinc finger and SCAN domain containing 5A