pentetrazol-2255 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the pentetrazol-2255 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AAGAB alpha- and gamma-adaptin binding protein
ABCD4 ATP-binding cassette, sub-family D (ALD), member 4
ADD2 adducin 2 (beta)
AKAP11 A kinase (PRKA) anchor protein 11
ALCAM activated leukocyte cell adhesion molecule
APC adenomatous polyposis coli
APOL6 apolipoprotein L, 6
ARPIN actin-related protein 2/3 complex inhibitor
BAIAP3 BAI1-associated protein 3
BGN biglycan
BHMT2 betaine--homocysteine S-methyltransferase 2
BMP10 bone morphogenetic protein 10
C21ORF2 chromosome 21 open reading frame 2
C7ORF69 chromosome 7 open reading frame 69
CD3D CD3d molecule, delta (CD3-TCR complex)
CD4 CD4 molecule
CD70 CD70 molecule
CDRT1 CMT1A duplicated region transcript 1
CEP152 centrosomal protein 152kDa
CFAP70 cilia and flagella associated protein 70
CFLAR CASP8 and FADD-like apoptosis regulator
CLDN1 claudin 1
CTAGE1 cutaneous T-cell lymphoma-associated antigen 1
CTBP2 C-terminal binding protein 2
CTNNA1 catenin (cadherin-associated protein), alpha 1, 102kDa
CXCL8 chemokine (C-X-C motif) ligand 8
CYP2C9 cytochrome P450, family 2, subfamily C, polypeptide 9
DICER1 dicer 1, ribonuclease type III
DNAJC28 DnaJ (Hsp40) homolog, subfamily C, member 28
DNASE1L2 deoxyribonuclease I-like 2
EPHB1 EPH receptor B1
ERN2 endoplasmic reticulum to nucleus signaling 2
FAM46C family with sequence similarity 46, member C
FBLN1 fibulin 1
FCGR2C Fc fragment of IgG, low affinity IIc, receptor for (CD32) (gene/pseudogene)
GABRD gamma-aminobutyric acid (GABA) A receptor, delta
GLP1R glucagon-like peptide 1 receptor
GLS glutaminase
GPR182 G protein-coupled receptor 182
HCRP1 hepatocellular carcinoma-related HCRP1
HPGDS hematopoietic prostaglandin D synthase
HTR1D 5-hydroxytryptamine (serotonin) receptor 1D, G protein-coupled
KLK13 kallikrein-related peptidase 13
KRT15 keratin 15, type I
LGALS9 lectin, galactoside-binding, soluble, 9
LRRN3 leucine rich repeat neuronal 3
LTBP4 latent transforming growth factor beta binding protein 4
MED18 mediator complex subunit 18
MEG3 maternally expressed 3 (non-protein coding)
METTL7A methyltransferase like 7A
MTRF1L mitochondrial translational release factor 1-like
MYEF2 myelin expression factor 2
MYO7A myosin VIIA
NR2F1 nuclear receptor subfamily 2, group F, member 1
NR4A1 nuclear receptor subfamily 4, group A, member 1
NUDT7 nudix (nucleoside diphosphate linked moiety X)-type motif 7
NUP54 nucleoporin 54kDa
PCDH1 protocadherin 1
PCDH12 protocadherin 12
PI4K2A phosphatidylinositol 4-kinase type 2 alpha
PML promyelocytic leukemia
PPP2R1B protein phosphatase 2, regulatory subunit A, beta
PRKCE protein kinase C, epsilon
PRKCI protein kinase C, iota
PRMT8 protein arginine methyltransferase 8
PSMB2 proteasome (prosome, macropain) subunit, beta type, 2
PSORS1C1 psoriasis susceptibility 1 candidate 1
PURG purine-rich element binding protein G
RABGAP1 RAB GTPase activating protein 1
RAD52 RAD52 homolog (S. cerevisiae)
RIMBP2 RIMS binding protein 2
RNF126P1 ring finger protein 126 pseudogene 1
RNGTT RNA guanylyltransferase and 5'-phosphatase
RUNX1 runt-related transcription factor 1
SDC2 syndecan 2
SH2D1A SH2 domain containing 1A
SHANK2 SH3 and multiple ankyrin repeat domains 2
SKP2 S-phase kinase-associated protein 2, E3 ubiquitin protein ligase
SLC17A7 solute carrier family 17 (vesicular glutamate transporter), member 7
SLC22A7 solute carrier family 22 (organic anion transporter), member 7
SLC9A3R2 solute carrier family 9, subfamily A (NHE3, cation proton antiporter 3), member 3 regulator 2
SMR3A submaxillary gland androgen regulated protein 3A
SRGN serglycin
SSX3 synovial sarcoma, X breakpoint 3
ST8SIA3 ST8 alpha-N-acetyl-neuraminide alpha-2,8-sialyltransferase 3
STX7 syntaxin 7
SYT2 synaptotagmin II
TAOK2 TAO kinase 2
TIMP3 TIMP metallopeptidase inhibitor 3
TJAP1 tight junction associated protein 1 (peripheral)
TMEM63A transmembrane protein 63A
TNFRSF11B tumor necrosis factor receptor superfamily, member 11b
TP53I11 tumor protein p53 inducible protein 11
TPMT thiopurine S-methyltransferase
VPS13A vacuolar protein sorting 13 homolog A (S. cerevisiae)
WSB1 WD repeat and SOCS box containing 1
YOD1 YOD1 deubiquitinase
ZNF175 zinc finger protein 175
ZNF223 zinc finger protein 223
ZZEF1 zinc finger, ZZ-type with EF-hand domain 1

decreased expression

Symbol Name
ADCY7 adenylate cyclase 7
AHNAK2 AHNAK nucleoprotein 2
AMT aminomethyltransferase
ARHGAP4 Rho GTPase activating protein 4
ARID3B AT rich interactive domain 3B (BRIGHT-like)
ARMC4 armadillo repeat containing 4
B3GNT3 UDP-GlcNAc:betaGal beta-1,3-N-acetylglucosaminyltransferase 3
BAG4 BCL2-associated athanogene 4
BEGAIN brain-enriched guanylate kinase-associated
C2ORF27A chromosome 2 open reading frame 27A
CILP cartilage intermediate layer protein, nucleotide pyrophosphohydrolase
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
DDX51 DEAD (Asp-Glu-Ala-Asp) box polypeptide 51
DDX54 DEAD (Asp-Glu-Ala-Asp) box polypeptide 54
DFFB DNA fragmentation factor, 40kDa, beta polypeptide (caspase-activated DNase)
DGAT1 diacylglycerol O-acyltransferase 1
DMTN dematin actin binding protein
DNAJA4 DnaJ (Hsp40) homolog, subfamily A, member 4
DNMT3A DNA (cytosine-5-)-methyltransferase 3 alpha
DUSP8 dual specificity phosphatase 8
EVA1B eva-1 homolog B (C. elegans)
EXD3 exonuclease 3'-5' domain containing 3
EXO5 exonuclease 5
FADS2 fatty acid desaturase 2
FBXO2 F-box protein 2
FKBP10 FK506 binding protein 10, 65 kDa
FLCN folliculin
FRK fyn-related Src family tyrosine kinase
GABRR2 gamma-aminobutyric acid (GABA) A receptor, rho 2
GFOD1 glucose-fructose oxidoreductase domain containing 1
GLB1L2 galactosidase, beta 1-like 2
GLRA1 glycine receptor, alpha 1
GNG3 guanine nucleotide binding protein (G protein), gamma 3
HLA-DMA major histocompatibility complex, class II, DM alpha
IRF2BP1 interferon regulatory factor 2 binding protein 1
ITGA10 integrin, alpha 10
ITGA3 integrin, alpha 3 (antigen CD49C, alpha 3 subunit of VLA-3 receptor)
KCNK12 potassium channel, two pore domain subfamily K, member 12
KCNN2 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 2
KIF13B kinesin family member 13B
KLK5 kallikrein-related peptidase 5
KREMEN2 kringle containing transmembrane protein 2
KRT24 keratin 24, type I
LIN7A lin-7 homolog A (C. elegans)
LMBR1L limb development membrane protein 1-like
LOXL3 lysyl oxidase-like 3
MAP4K2 mitogen-activated protein kinase kinase kinase kinase 2
MYO1E myosin IE
NLRX1 NLR family member X1
NOL12 nucleolar protein 12
NPFFR1 neuropeptide FF receptor 1
NRSN2 neurensin 2
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18
OTUB2 OTU deubiquitinase, ubiquitin aldehyde binding 2
P2RY6 pyrimidinergic receptor P2Y, G-protein coupled, 6
PCDHB13 protocadherin beta 13
PDPR pyruvate dehydrogenase phosphatase regulatory subunit
PIP5K1C phosphatidylinositol-4-phosphate 5-kinase, type I, gamma
PLA2G3 phospholipase A2, group III
POLL polymerase (DNA directed), lambda
PRAMEF11 PRAME family member 11
RASL11B RAS-like, family 11, member B
RASSF2 Ras association (RalGDS/AF-6) domain family member 2
RNASEL ribonuclease L (2',5'-oligoisoadenylate synthetase-dependent)
SCHIP1 schwannomin interacting protein 1
SERPINE2 serpin peptidase inhibitor, clade E (nexin, plasminogen activator inhibitor type 1), member 2
SLC12A8 solute carrier family 12, member 8
SLC22A4 solute carrier family 22 (organic cation/zwitterion transporter), member 4
SLC25A21 solute carrier family 25 (mitochondrial oxoadipate carrier), member 21
SLC30A3 solute carrier family 30 (zinc transporter), member 3
SLPI secretory leukocyte peptidase inhibitor
SMIM14 small integral membrane protein 14
SNTA1 syntrophin, alpha 1
STIM1 stromal interaction molecule 1
TAOK1 TAO kinase 1
TBC1D17 TBC1 domain family, member 17
TBC1D19 TBC1 domain family, member 19
TBKBP1 TBK1 binding protein 1
TM6SF1 transmembrane 6 superfamily member 1
TMEM242 transmembrane protein 242
TNFSF13 tumor necrosis factor (ligand) superfamily, member 13
TOM1 target of myb1 (chicken)
TRMT13 tRNA methyltransferase 13 homolog (S. cerevisiae)
TUBA4A tubulin, alpha 4a
TUT1 terminal uridylyl transferase 1, U6 snRNA-specific
USB1 U6 snRNA biogenesis 1
USP20 ubiquitin specific peptidase 20
VEGFB vascular endothelial growth factor B
VPS33A vacuolar protein sorting 33 homolog A (S. cerevisiae)
WLS wntless Wnt ligand secretion mediator
ZDHHC14 zinc finger, DHHC-type containing 14
ZNF34 zinc finger protein 34
ZNF350 zinc finger protein 350
ZNF37BP zinc finger protein 37B, pseudogene
ZNF442 zinc finger protein 442
ZNF552 zinc finger protein 552