phenoxybenzamine-5613 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the phenoxybenzamine-5613 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADM adrenomedullin
ALDH8A1 aldehyde dehydrogenase 8 family, member A1
ARVCF armadillo repeat gene deleted in velocardiofacial syndrome
ATF3 activating transcription factor 3
ATF7IP2 activating transcription factor 7 interacting protein 2
BDKRB2 bradykinin receptor B2
BTG2 BTG family, member 2
C1ORF54 chromosome 1 open reading frame 54
CAMKK2 calcium/calmodulin-dependent protein kinase kinase 2, beta
CDKN1A cyclin-dependent kinase inhibitor 1A (p21, Cip1)
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
COL2A1 collagen, type II, alpha 1
CREM cAMP responsive element modulator
CSRP2 cysteine and glycine-rich protein 2
CYP26A1 cytochrome P450, family 26, subfamily A, polypeptide 1
DCTN1 dynactin 1
DDIT3 DNA-damage-inducible transcript 3
DDIT4 DNA-damage-inducible transcript 4
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJB9 DnaJ (Hsp40) homolog, subfamily B, member 9
DUSP1 dual specificity phosphatase 1
DUSP4 dual specificity phosphatase 4
EGR1 early growth response 1
ENGASE endo-beta-N-acetylglucosaminidase
EPHA2 EPH receptor A2
ETS2 v-ets avian erythroblastosis virus E26 oncogene homolog 2
FAS Fas cell surface death receptor
FCER1G Fc fragment of IgE, high affinity I, receptor for; gamma polypeptide
FLJ42627 uncharacterized LOC645644
FOS FBJ murine osteosarcoma viral oncogene homolog
FOSL1 FOS-like antigen 1
GADD45A growth arrest and DNA-damage-inducible, alpha
GEM GTP binding protein overexpressed in skeletal muscle
GUCA1B guanylate cyclase activator 1B (retina)
HBEGF heparin-binding EGF-like growth factor
HBP1 HMG-box transcription factor 1
HLA-E major histocompatibility complex, class I, E
HMOX1 heme oxygenase 1
HSPA6 heat shock 70kDa protein 6 (HSP70B')
IDI2-AS1 IDI2 antisense RNA 1
IER5 immediate early response 5
IFT27 intraflagellar transport 27
INHBE inhibin, beta E
IRS2 insulin receptor substrate 2
JMJD6 jumonji domain containing 6
KCNAB1 potassium channel, voltage gated subfamily A regulatory beta subunit 1
KHDRBS1 KH domain containing, RNA binding, signal transduction associated 1
KIAA0125 KIAA0125
KLHL25 kelch-like family member 25
LARP6 La ribonucleoprotein domain family, member 6
LOC157562 uncharacterized LOC157562
MAFF v-maf avian musculoaponeurotic fibrosarcoma oncogene homolog F
MAP1LC3B microtubule-associated protein 1 light chain 3 beta
MDM2 MDM2 proto-oncogene, E3 ubiquitin protein ligase
MT1E metallothionein 1E
MT1F metallothionein 1F
MT1G metallothionein 1G
MT1H metallothionein 1H
MT1HL1 metallothionein 1H-like 1
MT1X metallothionein 1X
MT2A metallothionein 2A
N4BP2L1 NEDD4 binding protein 2-like 1
N4BP2L2 NEDD4 binding protein 2-like 2
NEK9 NIMA-related kinase 9
NHLH2 nescient helix loop helix 2
NR4A1 nuclear receptor subfamily 4, group A, member 1
NR4A2 nuclear receptor subfamily 4, group A, member 2
NUP88 nucleoporin 88kDa
OSGIN1 oxidative stress induced growth inhibitor 1
PGF placental growth factor
PHLDA1 pleckstrin homology-like domain, family A, member 1
PLLP plasmolipin
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1
POPDC3 popeye domain containing 3
PPP1R15A protein phosphatase 1, regulatory subunit 15A
PRKRIP1 PRKR interacting protein 1 (IL11 inducible)
RFPL2 ret finger protein-like 2
RGS2 regulator of G-protein signaling 2
RGS20 regulator of G-protein signaling 20
RND1 Rho family GTPase 1
RSL1D1 ribosomal L1 domain containing 1
SAT1 spermidine/spermine N1-acetyltransferase 1
SERPINB8 serpin peptidase inhibitor, clade B (ovalbumin), member 8
SERPINB9 serpin peptidase inhibitor, clade B (ovalbumin), member 9
SESN1 sestrin 1
SLC30A1 solute carrier family 30 (zinc transporter), member 1
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMIM7 small integral membrane protein 7
SNAI2 snail family zinc finger 2
SOX9 SRY (sex determining region Y)-box 9
SQSTM1 sequestosome 1
TES testin LIM domain protein
TMEM97 transmembrane protein 97
TSPYL2 TSPY-like 2
YPEL5 yippee-like 5 (Drosophila)
ZNF473 zinc finger protein 473
ZNF682 zinc finger protein 682
ZRSR1 zinc finger (CCCH type), RNA-binding motif and serine/arginine rich 1

decreased expression

Symbol Name
ACKR3 atypical chemokine receptor 3
ALG12 ALG12, alpha-1,6-mannosyltransferase
ARHGDIB Rho GDP dissociation inhibitor (GDI) beta
ARHGEF26 Rho guanine nucleotide exchange factor (GEF) 26
ARID5B AT rich interactive domain 5B (MRF1-like)
ATAD5 ATPase family, AAA domain containing 5
B3GNT1
BCL11B B-cell CLL/lymphoma 11B (zinc finger protein)
BRINP3 bone morphogenetic protein/retinoic acid inducible neural-specific 3
BUB1B BUB1 mitotic checkpoint serine/threonine kinase B
C14ORF93 chromosome 14 open reading frame 93
C1ORF106 chromosome 1 open reading frame 106
CAMKMT calmodulin-lysine N-methyltransferase
CBX8 chromobox homolog 8
CCDC85C coiled-coil domain containing 85C
CD82 CD82 molecule
CTDP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1
CTDSP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) small phosphatase 1
DAG1 dystroglycan 1 (dystrophin-associated glycoprotein 1)
DDAH1 dimethylarginine dimethylaminohydrolase 1
DDX58 DEAD (Asp-Glu-Ala-Asp) box polypeptide 58
DNAJA4 DnaJ (Hsp40) homolog, subfamily A, member 4
DYNC2H1 dynein, cytoplasmic 2, heavy chain 1
E2F8 E2F transcription factor 8
EGR3 early growth response 3
ERCC6L excision repair cross-complementation group 6-like
ESRP2 epithelial splicing regulatory protein 2
FAM155A family with sequence similarity 155, member A
FBXO22 F-box protein 22
FBXO5 F-box protein 5
FCHSD2 FCH and double SH3 domains 2
FER fer (fps/fes related) tyrosine kinase
FOXRED2 FAD-dependent oxidoreductase domain containing 2
GHR growth hormone receptor
GLI3 GLI family zinc finger 3
GNA12 guanine nucleotide binding protein (G protein) alpha 12
GPHN gephyrin
H1F0 H1 histone family, member 0
HIST1H1D histone cluster 1, H1d
HMGB3 high mobility group box 3
IGSF3 immunoglobulin superfamily, member 3
IRX5 iroquois homeobox 5
JAK2 Janus kinase 2
LGR4 leucine-rich repeat containing G protein-coupled receptor 4
LMNB1 lamin B1
MAP3K4 mitogen-activated protein kinase kinase kinase 4
MBD5 methyl-CpG binding domain protein 5
MEIS1 Meis homeobox 1
MKL2 MKL/myocardin-like 2
MPPED2 metallophosphoesterase domain containing 2
MSL1 male-specific lethal 1 homolog (Drosophila)
MXD3 MAX dimerization protein 3
NBEA neurobeachin
NCAPH non-SMC condensin I complex, subunit H
NDST2 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 2
NPY1R neuropeptide Y receptor Y1
OLFML2A olfactomedin-like 2A
OSMR oncostatin M receptor
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
PAGR1 PAXIP1 associated glutamate-rich protein 1
PBX3 pre-B-cell leukemia homeobox 3
PDE8B phosphodiesterase 8B
PHLPP1 PH domain and leucine rich repeat protein phosphatase 1
PIK3R1 phosphoinositide-3-kinase, regulatory subunit 1 (alpha)
PKIA protein kinase (cAMP-dependent, catalytic) inhibitor alpha
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
PPT2 palmitoyl-protein thioesterase 2
PRR15L proline rich 15-like
PSRC1 proline/serine-rich coiled-coil 1
PTPN13 protein tyrosine phosphatase, non-receptor type 13 (APO-1/CD95 (Fas)-associated phosphatase)
PTPRA protein tyrosine phosphatase, receptor type, A
PVRL3 poliovirus receptor-related 3
RBM12 RNA binding motif protein 12
RFTN1 raftlin, lipid raft linker 1
RHOB ras homolog family member B
RHPN1-AS1 RHPN1 antisense RNA 1 (head to head)
RIN2 Ras and Rab interactor 2
SEMA4D sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4D
SIRAL2 SIR2 antiphage like 2
SLC25A12 solute carrier family 25 (aspartate/glutamate carrier), member 12
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SLC6A14 solute carrier family 6 (amino acid transporter), member 14
SLC9A2 solute carrier family 9, subfamily A (NHE2, cation proton antiporter 2), member 2
SMAD7 SMAD family member 7
SSBP2 single-stranded DNA binding protein 2
SYTL2 synaptotagmin-like 2
TET3 tet methylcytosine dioxygenase 3
THNSL1 threonine synthase-like 1 (S. cerevisiae)
THRAP3 thyroid hormone receptor associated protein 3
TMEM223 transmembrane protein 223
TMPRSS3 transmembrane protease, serine 3
TRIB2 tribbles pseudokinase 2
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TRPS1 trichorhinophalangeal syndrome I
TTC28 tetratricopeptide repeat domain 28
UNC119 unc-119 homolog (C. elegans)
USB1 U6 snRNA biogenesis 1
VANGL1 VANGL planar cell polarity protein 1
VAV3 vav 3 guanine nucleotide exchange factor
WDR7 WD repeat domain 7