phthalylsulfathiazole-5249 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the phthalylsulfathiazole-5249 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AAMDC adipogenesis associated, Mth938 domain containing
ADAM22 ADAM metallopeptidase domain 22
ADORA1 adenosine A1 receptor
ALDOAP2 aldolase A, fructose-bisphosphate pseudogene 2
APOE apolipoprotein E
ARFGEF2 ADP-ribosylation factor guanine nucleotide-exchange factor 2 (brefeldin A-inhibited)
ARHGEF4 Rho guanine nucleotide exchange factor (GEF) 4
ARVCF armadillo repeat gene deleted in velocardiofacial syndrome
ATHL1 ATH1, acid trehalase-like 1 (yeast)
BEST2 bestrophin 2
BTN2A2 butyrophilin, subfamily 2, member A2
BTN3A3 butyrophilin, subfamily 3, member A3
CASP1 caspase 1, apoptosis-related cysteine peptidase
CD52 CD52 molecule
CD53 CD53 molecule
CLEC2B C-type lectin domain family 2, member B
COMP cartilage oligomeric matrix protein
CRHR2 corticotropin releasing hormone receptor 2
CRISP2 cysteine-rich secretory protein 2
CSHL1 chorionic somatomammotropin hormone-like 1
CXCL8 chemokine (C-X-C motif) ligand 8
CYP4F11 cytochrome P450, family 4, subfamily F, polypeptide 11
DIAPH2-AS1 DIAPH2 antisense RNA 1
DSPP dentin sialophosphoprotein
EPHB6 EPH receptor B6
ERCC2 excision repair cross-complementation group 2
FGF3 fibroblast growth factor 3
FGF6 fibroblast growth factor 6
FHL1 four and a half LIM domains 1
FLJ11292
GABRA2 gamma-aminobutyric acid (GABA) A receptor, alpha 2
GABRQ gamma-aminobutyric acid (GABA) A receptor, theta
GFER growth factor, augmenter of liver regeneration
GLI2 GLI family zinc finger 2
GPC3 glypican 3
GPR3 G protein-coupled receptor 3
GRIA3 glutamate receptor, ionotropic, AMPA 3
GRM1 glutamate receptor, metabotropic 1
GRM8 glutamate receptor, metabotropic 8
GRPR gastrin-releasing peptide receptor
HLA-DOA major histocompatibility complex, class II, DO alpha
INO80D INO80 complex subunit D
ITGB4 integrin, beta 4
JPH3 junctophilin 3
KCNJ8 potassium channel, inwardly rectifying subfamily J, member 8
KIF1C kinesin family member 1C
KSR1 kinase suppressor of ras 1
LEFTY1 left-right determination factor 1
LPAR4 lysophosphatidic acid receptor 4
LTC4S leukotriene C4 synthase
LY9 lymphocyte antigen 9
MAF v-maf avian musculoaponeurotic fibrosarcoma oncogene homolog
MAPK8IP3 mitogen-activated protein kinase 8 interacting protein 3
MEP1B meprin A, beta
MGAT5 mannosyl (alpha-1,6-)-glycoprotein beta-1,6-N-acetyl-glucosaminyltransferase
MUSK muscle, skeletal, receptor tyrosine kinase
MYLK myosin light chain kinase
NDOR1 NADPH dependent diflavin oxidoreductase 1
NIPAL3 NIPA-like domain containing 3
NNAT neuronatin
NSUN6 NOP2/Sun domain family, member 6
OAS1 2'-5'-oligoadenylate synthetase 1, 40/46kDa
PHLDA1 pleckstrin homology-like domain, family A, member 1
PKP1 plakophilin 1
PLAT plasminogen activator, tissue
PMP2 peripheral myelin protein 2
POLL polymerase (DNA directed), lambda
PPARA peroxisome proliferator-activated receptor alpha
PPP1R2P9 protein phosphatase 1, regulatory (inhibitor) subunit 2 pseudogene 9
PROX1 prospero homeobox 1
PSG3 pregnancy specific beta-1-glycoprotein 3
RARRES2 retinoic acid receptor responder (tazarotene induced) 2
RPL23AP53 ribosomal protein L23a pseudogene 53
RUNX1 runt-related transcription factor 1
S1PR2 sphingosine-1-phosphate receptor 2
SCN10A sodium channel, voltage gated, type X alpha subunit
SDC3 syndecan 3
SFRP4 secreted frizzled-related protein 4
SGK2 serum/glucocorticoid regulated kinase 2
SIGLEC7 sialic acid binding Ig-like lectin 7
SIX3 SIX homeobox 3
SLC11A1 solute carrier family 11 (proton-coupled divalent metal ion transporter), member 1
SLC22A7 solute carrier family 22 (organic anion transporter), member 7
SLC7A8 solute carrier family 7 (amino acid transporter light chain, L system), member 8
SNCA synuclein, alpha (non A4 component of amyloid precursor)
SPARCL1 SPARC-like 1 (hevin)
SPINK1 serine peptidase inhibitor, Kazal type 1
SSX1 synovial sarcoma, X breakpoint 1
SULT2A1 sulfotransferase family, cytosolic, 2A, dehydroepiandrosterone (DHEA)-preferring, member 1
TBC1D2 TBC1 domain family, member 2
TBX3 T-box 3
TCP10 t-complex 10
TMCC2 transmembrane and coiled-coil domain family 2
TNFSF10 tumor necrosis factor (ligand) superfamily, member 10
TRPM3 transient receptor potential cation channel, subfamily M, member 3
UTY ubiquitously transcribed tetratricopeptide repeat containing, Y-linked
VIPR2 vasoactive intestinal peptide receptor 2
ZNF44 zinc finger protein 44
ZNF440 zinc finger protein 440

decreased expression

Symbol Name
ABHD17B abhydrolase domain containing 17B
ACSL4 acyl-CoA synthetase long-chain family member 4
ACTL8 actin-like 8
AKIP1 A kinase (PRKA) interacting protein 1
ALCAM activated leukocyte cell adhesion molecule
ALDH3B1 aldehyde dehydrogenase 3 family, member B1
ANKFY1 ankyrin repeat and FYVE domain containing 1
ARHGEF5 Rho guanine nucleotide exchange factor (GEF) 5
ASPHD1 aspartate beta-hydroxylase domain containing 1
BCORL1 BCL6 corepressor-like 1
C16ORF59 chromosome 16 open reading frame 59
C17ORF80 chromosome 17 open reading frame 80
CCNJ cyclin J
CENPJ centromere protein J
CHRM3 cholinergic receptor, muscarinic 3
CIC capicua transcriptional repressor
CLCN5 chloride channel, voltage-sensitive 5
COPZ2 coatomer protein complex, subunit zeta 2
CRYBB2P1 crystallin, beta B2 pseudogene 1
CRYBG3 beta-gamma crystallin domain containing 3
CTSD cathepsin D
CYP2R1 cytochrome P450, family 2, subfamily R, polypeptide 1
DSC2 desmocollin 2
DYRK3 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 3
EAF2 ELL associated factor 2
EIF2S3 eukaryotic translation initiation factor 2, subunit 3 gamma, 52kDa
ENO2 enolase 2 (gamma, neuronal)
EPHA2 EPH receptor A2
FBXO5 F-box protein 5
FBXW7 F-box and WD repeat domain containing 7, E3 ubiquitin protein ligase
GALNT12 polypeptide N-acetylgalactosaminyltransferase 12
GATC glutamyl-tRNA(Gln) amidotransferase, subunit C
GBP2 guanylate binding protein 2, interferon-inducible
GDAP1 ganglioside induced differentiation associated protein 1
GINS4 GINS complex subunit 4 (Sld5 homolog)
HAUS6 HAUS augmin-like complex, subunit 6
HIST2H2AA3 histone cluster 2, H2aa3
HLA-J major histocompatibility complex, class I, J (pseudogene)
IFI6 interferon, alpha-inducible protein 6
IMPACT impact RWD domain protein
ITPKB inositol-trisphosphate 3-kinase B
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KDM7A lysine (K)-specific demethylase 7A
LIN7A lin-7 homolog A (C. elegans)
LMCD1 LIM and cysteine-rich domains 1
LRP2 low density lipoprotein receptor-related protein 2
LRRC61 leucine rich repeat containing 61
LZTR1 leucine-zipper-like transcription regulator 1
MAP3K1 mitogen-activated protein kinase kinase kinase 1, E3 ubiquitin protein ligase
MBTPS2 membrane-bound transcription factor peptidase, site 2
MDM4 MDM4, p53 regulator
MTCP1 mature T-cell proliferation 1
MVP major vault protein
NAA50 N(alpha)-acetyltransferase 50, NatE catalytic subunit
NPIPB3 nuclear pore complex interacting protein family, member B3
NR1H3 nuclear receptor subfamily 1, group H, member 3
OSGEPL1 O-sialoglycoprotein endopeptidase-like 1
PGGT1B protein geranylgeranyltransferase type I, beta subunit
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
PLXNA3 plexin A3
POLR3F polymerase (RNA) III (DNA directed) polypeptide F, 39 kDa
PROCR protein C receptor, endothelial
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RANBP17 RAN binding protein 17
RANBP6 RAN binding protein 6
RHBDD3 rhomboid domain containing 3
RIBC2 RIB43A domain with coiled-coils 2
ROBO1 roundabout, axon guidance receptor, homolog 1 (Drosophila)
RPP14 ribonuclease P/MRP 14kDa subunit
S100A9 S100 calcium binding protein A9
SGPP1 sphingosine-1-phosphate phosphatase 1
SLC25A21 solute carrier family 25 (mitochondrial oxoadipate carrier), member 21
SMG1 SMG1 phosphatidylinositol 3-kinase-related kinase
SNX24 sorting nexin 24
SP1 Sp1 transcription factor
SPANXC SPANX family, member C
SRD5A3 steroid 5 alpha-reductase 3
SSFA2 sperm specific antigen 2
STRN striatin, calmodulin binding protein
SUPT3H suppressor of Ty 3 homolog (S. cerevisiae)
TBL1XR1 transducin (beta)-like 1 X-linked receptor 1
TESK1 testis-specific kinase 1
TMEM242 transmembrane protein 242
TMEM53 transmembrane protein 53
TRAF2 TNF receptor-associated factor 2
TRIM36 tripartite motif containing 36
TRMU tRNA 5-methylaminomethyl-2-thiouridylate methyltransferase
TXLNG taxilin gamma
UHRF1BP1L UHRF1 binding protein 1-like
XK X-linked Kx blood group
ZNF136 zinc finger protein 136
ZNF189 zinc finger protein 189
ZNF219 zinc finger protein 219
ZNF329 zinc finger protein 329
ZNF34 zinc finger protein 34
ZNF510 zinc finger protein 510
ZNF573 zinc finger protein 573
ZNF652 zinc finger protein 652