pindolol-2238 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the pindolol-2238 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AASS aminoadipate-semialdehyde synthase
ADAM20 ADAM metallopeptidase domain 20
ADAMTS13 ADAM metallopeptidase with thrombospondin type 1 motif, 13
ADGRD2 adhesion G protein-coupled receptor D2
ADM adrenomedullin
AGER advanced glycosylation end product-specific receptor
APOL6 apolipoprotein L, 6
ARAP1 ArfGAP with RhoGAP domain, ankyrin repeat and PH domain 1
ASAP3 ArfGAP with SH3 domain, ankyrin repeat and PH domain 3
ATP1A3 ATPase, Na+/K+ transporting, alpha 3 polypeptide
ATXN3 ataxin 3
BAZ2A bromodomain adjacent to zinc finger domain, 2A
BCAT1 branched chain amino-acid transaminase 1, cytosolic
BRF1 BRF1, RNA polymerase III transcription initiation factor 90 kDa subunit
BST2 bone marrow stromal cell antigen 2
BTRC beta-transducin repeat containing E3 ubiquitin protein ligase
BUB1 BUB1 mitotic checkpoint serine/threonine kinase
C10ORF95 chromosome 10 open reading frame 95
C8ORF44 chromosome 8 open reading frame 44
CACNA1G calcium channel, voltage-dependent, T type, alpha 1G subunit
CACNB1 calcium channel, voltage-dependent, beta 1 subunit
CACNG1 calcium channel, voltage-dependent, gamma subunit 1
CAMK2B calcium/calmodulin-dependent protein kinase II beta
CAPZB capping protein (actin filament) muscle Z-line, beta
CCDC81 coiled-coil domain containing 81
CD70 CD70 molecule
CDRT1 CMT1A duplicated region transcript 1
CFAP45 cilia and flagella associated protein 45
CHM choroideremia (Rab escort protein 1)
CPED1 cadherin-like and PC-esterase domain containing 1
DLX2 distal-less homeobox 2
DNAI2 dynein, axonemal, intermediate chain 2
DNASE1 deoxyribonuclease I
DNASE2B deoxyribonuclease II beta
DPP4 dipeptidyl-peptidase 4
DRD1 dopamine receptor D1
ENOX2 ecto-NOX disulfide-thiol exchanger 2
FAM86C1 family with sequence similarity 86, member C1
FASLG Fas ligand (TNF superfamily, member 6)
FBXW4P1 F-box and WD repeat domain containing 4 pseudogene 1
FGFR1 fibroblast growth factor receptor 1
FLJ11292
FOXG1 forkhead box G1
FOXI1 forkhead box I1
FZR1 fizzy/cell division cycle 20 related 1 (Drosophila)
GGA3 golgi-associated, gamma adaptin ear containing, ARF binding protein 3
GNG3 guanine nucleotide binding protein (G protein), gamma 3
GRK5 G protein-coupled receptor kinase 5
GTDC1 glycosyltransferase-like domain containing 1
HCN2 hyperpolarization activated cyclic nucleotide gated potassium channel 2
HOXC5 homeobox C5
ICOSLG inducible T-cell co-stimulator ligand
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KRT17 keratin 17, type I
LAIR2 leukocyte-associated immunoglobulin-like receptor 2
LAMA4 laminin, alpha 4
LEPR leptin receptor
LTBP2 latent transforming growth factor beta binding protein 2
MAOA monoamine oxidase A
MED25 mediator complex subunit 25
MEF2C myocyte enhancer factor 2C
MMP25 matrix metallopeptidase 25
MS4A1 membrane-spanning 4-domains, subfamily A, member 1
MTCP1 mature T-cell proliferation 1
MUC3B mucin 3B, cell surface associated
NDST1 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 1
NPAS2 neuronal PAS domain protein 2
OVOL2 ovo-like zinc finger 2
PARD6B par-6 family cell polarity regulator beta
PDE5A phosphodiesterase 5A, cGMP-specific
PHC3 polyhomeotic homolog 3 (Drosophila)
PHF20L1 PHD finger protein 20-like 1
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
PLEKHF1 pleckstrin homology domain containing, family F (with FYVE domain) member 1
PLEKHG3 pleckstrin homology domain containing, family G (with RhoGef domain) member 3
PLIN2 perilipin 2
PNPLA3 patatin-like phospholipase domain containing 3
PQLC3 PQ loop repeat containing 3
PTCRA pre T-cell antigen receptor alpha
PTGDR2 prostaglandin D2 receptor 2
PVR poliovirus receptor
RBFOX1 RNA binding protein, fox-1 homolog (C. elegans) 1
RLN1 relaxin 1
RPLP2 ribosomal protein, large, P2
S100A8 S100 calcium binding protein A8
SAG S-antigen; retina and pineal gland (arrestin)
SERHL2 serine hydrolase-like 2
SFI1 Sfi1 homolog, spindle assembly associated (yeast)
SIRT4 sirtuin 4
SLC9A5 solute carrier family 9, subfamily A (NHE5, cation proton antiporter 5), member 5
SMAD1 SMAD family member 1
SORBS1 sorbin and SH3 domain containing 1
SULT4A1 sulfotransferase family 4A, member 1
TAOK2 TAO kinase 2
TFAP2A transcription factor AP-2 alpha (activating enhancer binding protein 2 alpha)
TGFB2 transforming growth factor, beta 2
TREX1 three prime repair exonuclease 1
VPS13D vacuolar protein sorting 13 homolog D (S. cerevisiae)
XYLB xylulokinase homolog (H. influenzae)
YPEL1 yippee-like 1 (Drosophila)

decreased expression

Symbol Name
ALPK1 alpha-kinase 1
APOLD1 apolipoprotein L domain containing 1
ATAD5 ATPase family, AAA domain containing 5
ATAT1 alpha tubulin acetyltransferase 1
BEX4 brain expressed, X-linked 4
BMP15 bone morphogenetic protein 15
C17ORF53 chromosome 17 open reading frame 53
C1ORF159 chromosome 1 open reading frame 159
CA5BP1 carbonic anhydrase VB pseudogene 1
CCDC132 coiled-coil domain containing 132
CCRN4L CCR4 carbon catabolite repression 4-like (S. cerevisiae)
CD83 CD83 molecule
CDK3 cyclin-dependent kinase 3
CDKN2D cyclin-dependent kinase inhibitor 2D (p19, inhibits CDK4)
CERS4 ceramide synthase 4
CTDP1 CTD (carboxy-terminal domain, RNA polymerase II, polypeptide A) phosphatase, subunit 1
CYP2B7P cytochrome P450, family 2, subfamily B, polypeptide 7, pseudogene
DDX54 DEAD (Asp-Glu-Ala-Asp) box polypeptide 54
DNAJA4 DnaJ (Hsp40) homolog, subfamily A, member 4
DNAJB2 DnaJ (Hsp40) homolog, subfamily B, member 2
EHD3 EH-domain containing 3
ENTPD7 ectonucleoside triphosphate diphosphohydrolase 7
EPB41L5 erythrocyte membrane protein band 4.1 like 5
FAM46C family with sequence similarity 46, member C
FBXL8 F-box and leucine-rich repeat protein 8
FLJ11710 uncharacterized protein FLJ11710
GATA4 GATA binding protein 4
GPRC5D G protein-coupled receptor, class C, group 5, member D
GSTA4 glutathione S-transferase alpha 4
HIST1H3E histone cluster 1, H3e
HIST1H4A histone cluster 1, H4a
HIST1H4D histone cluster 1, H4d
HPX hemopexin
IDI2-AS1 IDI2 antisense RNA 1
IFT140 intraflagellar transport 140
IGSF1 immunoglobulin superfamily, member 1
IRF2BP1 interferon regulatory factor 2 binding protein 1
ITGA3 integrin, alpha 3 (antigen CD49C, alpha 3 subunit of VLA-3 receptor)
JUNB jun B proto-oncogene
KIF13B kinesin family member 13B
KLHL25 kelch-like family member 25
KREMEN2 kringle containing transmembrane protein 2
KRT15 keratin 15, type I
KRT6B keratin 6B, type II
LAMP3 lysosomal-associated membrane protein 3
LHX1 LIM homeobox 1
LHX6 LIM homeobox 6
LMO2 LIM domain only 2 (rhombotin-like 1)
LOC729164 hCG1732469
LRP2 low density lipoprotein receptor-related protein 2
LYRM9 LYR motif containing 9
LZTS3 leucine zipper, putative tumor suppressor family member 3
MAGEB2 melanoma antigen family B2
MBTD1 mbt domain containing 1
MCC mutated in colorectal cancers
MRPL41 mitochondrial ribosomal protein L41
MSI1 musashi RNA-binding protein 1
NPFFR1 neuropeptide FF receptor 1
NPIPB3 nuclear pore complex interacting protein family, member B3
OSMR oncostatin M receptor
PADI1 peptidyl arginine deiminase, type I
PEX26 peroxisomal biogenesis factor 26
PHC1 polyhomeotic homolog 1 (Drosophila)
PHEX phosphate regulating endopeptidase homolog, X-linked
PLA2G4C phospholipase A2, group IVC (cytosolic, calcium-independent)
PLAC1 placenta-specific 1
PLIN3 perilipin 3
PMEL premelanosome protein
POLL polymerase (DNA directed), lambda
PQLC2 PQ loop repeat containing 2
PRPH peripherin
RNASEL ribonuclease L (2',5'-oligoisoadenylate synthetase-dependent)
RNF39 ring finger protein 39
RPGRIP1L RPGRIP1-like
SEC14L5 SEC14-like 5 (S. cerevisiae)
SERPINE2 serpin peptidase inhibitor, clade E (nexin, plasminogen activator inhibitor type 1), member 2
SH3BGR SH3 domain binding glutamate-rich protein
SKA1 spindle and kinetochore associated complex subunit 1
SLC43A1 solute carrier family 43 (amino acid system L transporter), member 1
SLC47A1 solute carrier family 47 (multidrug and toxin extrusion), member 1
SMARCD3 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 3
SMPDL3B sphingomyelin phosphodiesterase, acid-like 3B
SUGP1 SURP and G patch domain containing 1
TBC1D17 TBC1 domain family, member 17
TMEM120B transmembrane protein 120B
TNS2 tensin 2
TOPORS topoisomerase I binding, arginine/serine-rich, E3 ubiquitin protein ligase
TRPC5 transient receptor potential cation channel, subfamily C, member 5
TYRP1 tyrosinase-related protein 1
VAX2 ventral anterior homeobox 2
VWA5A von Willebrand factor A domain containing 5A
XRCC2 X-ray repair complementing defective repair in Chinese hamster cells 2
ZFP69B ZFP69 zinc finger protein B
ZNF37BP zinc finger protein 37B, pseudogene
ZNF747 zinc finger protein 747
ZSCAN2 zinc finger and SCAN domain containing 2