pindolol-6834 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the pindolol-6834 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADORA1 adenosine A1 receptor
ADRBK1 adrenergic, beta, receptor kinase 1
AGPAT4 1-acylglycerol-3-phosphate O-acyltransferase 4
AKAP6 A kinase (PRKA) anchor protein 6
AKT2 v-akt murine thymoma viral oncogene homolog 2
AMN amnion associated transmembrane protein
ANGPT4 angiopoietin 4
ARHGEF1 Rho guanine nucleotide exchange factor (GEF) 1
ATAT1 alpha tubulin acetyltransferase 1
ATP5G2 ATP synthase, H+ transporting, mitochondrial Fo complex, subunit C2 (subunit 9)
ATP9A ATPase, class II, type 9A
BAIAP3 BAI1-associated protein 3
BEGAIN brain-enriched guanylate kinase-associated
C14ORF79 chromosome 14 open reading frame 79
C17ORF53 chromosome 17 open reading frame 53
C9ORF9 chromosome 9 open reading frame 9
CASP1 caspase 1, apoptosis-related cysteine peptidase
CD3D CD3d molecule, delta (CD3-TCR complex)
CD48 CD48 molecule
CD83 CD83 molecule
CDK12 cyclin-dependent kinase 12
CEACAM1 carcinoembryonic antigen-related cell adhesion molecule 1 (biliary glycoprotein)
CFAP69 cilia and flagella associated protein 69
CLGN calmegin
CPN2 carboxypeptidase N, polypeptide 2
CYP2C9 cytochrome P450, family 2, subfamily C, polypeptide 9
CYTH4 cytohesin 4
DCAKD dephospho-CoA kinase domain containing
DCBLD2 discoidin, CUB and LCCL domain containing 2
DENND5B DENN/MADD domain containing 5B
DNAJB12 DnaJ (Hsp40) homolog, subfamily B, member 12
DOK4 docking protein 4
DST dystonin
EHBP1L1 EH domain binding protein 1-like 1
ELK3 ELK3, ETS-domain protein (SRF accessory protein 2)
EPHX2 epoxide hydrolase 2, cytoplasmic
FAM188A family with sequence similarity 188, member A
FEZ2 fasciculation and elongation protein zeta 2 (zygin II)
FGF16 fibroblast growth factor 16
FGFR3 fibroblast growth factor receptor 3
FLOT1 flotillin 1
FUBP1 far upstream element (FUSE) binding protein 1
GALR2 galanin receptor 2
GRM7 glutamate receptor, metabotropic 7
HEXIM1 hexamethylene bis-acetamide inducible 1
HEY2 hes-related family bHLH transcription factor with YRPW motif 2
HIST1H3J histone cluster 1, H3j
HIST1H4E histone cluster 1, H4e
HS2ST1 heparan sulfate 2-O-sulfotransferase 1
IFFO1 intermediate filament family orphan 1
IFNA14 interferon, alpha 14
IL5RA interleukin 5 receptor, alpha
ITM2C integral membrane protein 2C
KCNAB2 potassium channel, voltage gated subfamily A regulatory beta subunit 2
KHSRP KH-type splicing regulatory protein
KMT2A lysine (K)-specific methyltransferase 2A
LAMA4 laminin, alpha 4
LOC157562 uncharacterized LOC157562
MFI2 antigen p97 (melanoma associated) identified by monoclonal antibodies 133.2 and 96.5
NF1 neurofibromin 1
NOX5 NADPH oxidase, EF-hand calcium binding domain 5
ONECUT2 one cut homeobox 2
PDE6B phosphodiesterase 6B, cGMP-specific, rod, beta
PER3 period circadian clock 3
PGAM2 phosphoglycerate mutase 2 (muscle)
PLEKHO1 pleckstrin homology domain containing, family O member 1
POU2F3 POU class 2 homeobox 3
PPFIBP1 PTPRF interacting protein, binding protein 1 (liprin beta 1)
PPP4R4 protein phosphatase 4, regulatory subunit 4
PQLC2 PQ loop repeat containing 2
PRDM10 PR domain containing 10
PRKACA protein kinase, cAMP-dependent, catalytic, alpha
PROZ protein Z, vitamin K-dependent plasma glycoprotein
RAB3B RAB3B, member RAS oncogene family
RHBDD3 rhomboid domain containing 3
RIMS3 regulating synaptic membrane exocytosis 3
RPL23AP32 ribosomal protein L23a pseudogene 32
RRH retinal pigment epithelium-derived rhodopsin homolog
RUNX1 runt-related transcription factor 1
SEMA4G sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4G
SLC11A1 solute carrier family 11 (proton-coupled divalent metal ion transporter), member 1
SLC19A1 solute carrier family 19 (folate transporter), member 1
SOX9 SRY (sex determining region Y)-box 9
SPRR1B small proline-rich protein 1B
SYNGR1 synaptogyrin 1
TM4SF1 transmembrane 4 L six family member 1
TMPRSS4 transmembrane protease, serine 4
UHRF1BP1L UHRF1 binding protein 1-like
USP2 ubiquitin specific peptidase 2
VASH2 vasohibin 2
VLDLR very low density lipoprotein receptor
WDR59 WD repeat domain 59
ZC3HAV1 zinc finger CCCH-type, antiviral 1
ZCCHC24 zinc finger, CCHC domain containing 24
ZFPL1 zinc finger protein-like 1
ZMIZ2 zinc finger, MIZ-type containing 2
ZNF440 zinc finger protein 440
ZNF710 zinc finger protein 710
ZZEF1 zinc finger, ZZ-type with EF-hand domain 1

decreased expression

Symbol Name
ADTRP androgen-dependent TFPI-regulating protein
ALDH4A1 aldehyde dehydrogenase 4 family, member A1
APOLD1 apolipoprotein L domain containing 1
ARHGEF5 Rho guanine nucleotide exchange factor (GEF) 5
ARSB arylsulfatase B
ASCC2 activating signal cointegrator 1 complex subunit 2
B3GNT3 UDP-GlcNAc:betaGal beta-1,3-N-acetylglucosaminyltransferase 3
BBC3 BCL2 binding component 3
BCL9 B-cell CLL/lymphoma 9
BTF3P11 basic transcription factor 3 pseudogene 11
C19ORF73 chromosome 19 open reading frame 73
C8ORF60 chromosome 8 open reading frame 60
CAMK1 calcium/calmodulin-dependent protein kinase I
CGA glycoprotein hormones, alpha polypeptide
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CNKSR1 connector enhancer of kinase suppressor of Ras 1
CNNM4 cyclin and CBS domain divalent metal cation transport mediator 4
CUL9 cullin 9
CYP2R1 cytochrome P450, family 2, subfamily R, polypeptide 1
EEF2KMT eukaryotic elongation factor 2 lysine methyltransferase
ERCC4 excision repair cross-complementation group 4
ERN1 endoplasmic reticulum to nucleus signaling 1
EXD3 exonuclease 3'-5' domain containing 3
FAM131A family with sequence similarity 131, member A
FAM169A family with sequence similarity 169, member A
FBXO22 F-box protein 22
FRS2 fibroblast growth factor receptor substrate 2
GNB1L guanine nucleotide binding protein (G protein), beta polypeptide 1-like
GNG4 guanine nucleotide binding protein (G protein), gamma 4
GNG7 guanine nucleotide binding protein (G protein), gamma 7
GPRASP1 G protein-coupled receptor associated sorting protein 1
GTPBP2 GTP binding protein 2
HDAC7 histone deacetylase 7
HIST1H4D histone cluster 1, H4d
IFI6 interferon, alpha-inducible protein 6
IFT54 intraflagellar transport 54
IL20RA interleukin 20 receptor, alpha
INO80D INO80 complex subunit D
IQCG IQ motif containing G
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
KIAA0125 KIAA0125
KIAA0355 KIAA0355
KLF2 Kruppel-like factor 2
KREMEN2 kringle containing transmembrane protein 2
KRT15 keratin 15, type I
LGALS4 lectin, galactoside-binding, soluble, 4
LHX6 LIM homeobox 6
LIF leukemia inhibitory factor
LIN7B lin-7 homolog B (C. elegans)
LMBR1L limb development membrane protein 1-like
LOC729164 hCG1732469
LRCH1 leucine-rich repeats and calponin homology (CH) domain containing 1
MC1R melanocortin 1 receptor (alpha melanocyte stimulating hormone receptor)
NCALD neurocalcin delta
NEK11 NIMA-related kinase 11
NPIPB3 nuclear pore complex interacting protein family, member B3
NRGN neurogranin (protein kinase C substrate, RC3)
OTUB2 OTU deubiquitinase, ubiquitin aldehyde binding 2
OTUD3 OTU deubiquitinase 3
PADI3 peptidyl arginine deiminase, type III
PHEX phosphate regulating endopeptidase homolog, X-linked
PIGZ phosphatidylinositol glycan anchor biosynthesis, class Z
POLL polymerase (DNA directed), lambda
POM121 POM121 transmembrane nucleoporin
PPP2R3B protein phosphatase 2, regulatory subunit B'', beta
PRODH proline dehydrogenase (oxidase) 1
PTP4A3 protein tyrosine phosphatase type IVA, member 3
RAB3A RAB3A, member RAS oncogene family
RASAL1 RAS protein activator like 1 (GAP1 like)
RGS2 regulator of G-protein signaling 2
ROM1 retinal outer segment membrane protein 1
RRAGB Ras-related GTP binding B
S100A4 S100 calcium binding protein A4
S100A9 S100 calcium binding protein A9
SAMSN1 SAM domain, SH3 domain and nuclear localization signals 1
SCD5 stearoyl-CoA desaturase 5
SEMA4A sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4A
SLC22A18AS solute carrier family 22 (organic cation transporter), member 18 antisense
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC26A6 solute carrier family 26 (anion exchanger), member 6
SLC9A1 solute carrier family 9, subfamily A (NHE1, cation proton antiporter 1), member 1
SOWAHC sosondowah ankyrin repeat domain family member C
SOX3 SRY (sex determining region Y)-box 3
STAG3L4 stromal antigen 3-like 4 (pseudogene)
TAF4B TAF4b RNA polymerase II, TATA box binding protein (TBP)-associated factor, 105kDa
TICAM1 toll-like receptor adaptor molecule 1
TLR5 toll-like receptor 5
TMEM209 transmembrane protein 209
TMEM212 transmembrane protein 212
TMEM53 transmembrane protein 53
UPK3B uroplakin 3B
VEZT vezatin, adherens junctions transmembrane protein
VWA1 von Willebrand factor A domain containing 1
YIF1B Yip1 interacting factor homolog B (S. cerevisiae)
ZAK sterile alpha motif and leucine zipper containing kinase AZK
ZBED1 zinc finger, BED-type containing 1
ZNF552 zinc finger protein 552
ZNF665 zinc finger protein 665
ZNF747 zinc finger protein 747