pirenzepine-2071 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

194 genes differentially expressed following the pirenzepine-2071 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AFF4 AF4/FMR2 family, member 4
AKAP5 A kinase (PRKA) anchor protein 5
AKAP7 A kinase (PRKA) anchor protein 7
AKR7A3 aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase)
ALDH3A1 aldehyde dehydrogenase 3 family, member A1
ALDH3B1 aldehyde dehydrogenase 3 family, member B1
ARSB arylsulfatase B
BAG4 BCL2-associated athanogene 4
BBC3 BCL2 binding component 3
BCORL1 BCL6 corepressor-like 1
BMP1 bone morphogenetic protein 1
CACYBP calcyclin binding protein
CASZ1 castor zinc finger 1
CCL20 chemokine (C-C motif) ligand 20
CDC42EP2 CDC42 effector protein (Rho GTPase binding) 2
CDH1 cadherin 1, type 1, E-cadherin (epithelial)
CLCN7 chloride channel, voltage-sensitive 7
COL13A1 collagen, type XIII, alpha 1
COL4A2 collagen, type IV, alpha 2
COL9A3 collagen, type IX, alpha 3
CRY2 cryptochrome circadian clock 2
DDX49 DEAD (Asp-Glu-Ala-Asp) box polypeptide 49
DLG3 discs, large homolog 3 (Drosophila)
DNAJB5 DnaJ (Hsp40) homolog, subfamily B, member 5
DSCR3 Down syndrome critical region 3
EIF2S2 eukaryotic translation initiation factor 2, subunit 2 beta, 38kDa
EML3 echinoderm microtubule associated protein like 3
FAM174B family with sequence similarity 174, member B
FAM184A family with sequence similarity 184, member A
GABARAPL1 GABA(A) receptor-associated protein like 1
GGA2 golgi-associated, gamma adaptin ear containing, ARF binding protein 2
GIT2 G protein-coupled receptor kinase interacting ArfGAP 2
GNA13 guanine nucleotide binding protein (G protein), alpha 13
GPR4 G protein-coupled receptor 4
GSDMD gasdermin D
IDH2 isocitrate dehydrogenase 2 (NADP+), mitochondrial
IFNA14 interferon, alpha 14
KIFC3 kinesin family member C3
KLF6 Kruppel-like factor 6
KMO kynurenine 3-monooxygenase (kynurenine 3-hydroxylase)
KRIT1 KRIT1, ankyrin repeat containing
KRT15 keratin 15, type I
KRT17 keratin 17, type I
LPIN2 lipin 2
MAX MYC associated factor X
MED28 mediator complex subunit 28
MIIP migration and invasion inhibitory protein
MYRF myelin regulatory factor
NADK NAD kinase
NMT2 N-myristoyltransferase 2
NUP98 nucleoporin 98kDa
PCYT2 phosphate cytidylyltransferase 2, ethanolamine
PHC1 polyhomeotic homolog 1 (Drosophila)
PIK3CD phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit delta
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
PLEKHF1 pleckstrin homology domain containing, family F (with FYVE domain) member 1
PPBP pro-platelet basic protein (chemokine (C-X-C motif) ligand 7)
PPP1R15A protein phosphatase 1, regulatory subunit 15A
PRKAA2 protein kinase, AMP-activated, alpha 2 catalytic subunit
PRR7 proline rich 7 (synaptic)
RAB3IL1 RAB3A interacting protein (rabin3)-like 1
RAD54B RAD54 homolog B (S. cerevisiae)
RALB v-ral simian leukemia viral oncogene homolog B
RAPGEF5 Rap guanine nucleotide exchange factor (GEF) 5
RB1 retinoblastoma 1
RNASET2 ribonuclease T2
RNF113A ring finger protein 113A
RPL23AP32 ribosomal protein L23a pseudogene 32
RPS6KA6 ribosomal protein S6 kinase, 90kDa, polypeptide 6
S1PR1 sphingosine-1-phosphate receptor 1
SEPP1 selenoprotein P, plasma, 1
SERPINA1 serpin peptidase inhibitor, clade A (alpha-1 antiproteinase, antitrypsin), member 1
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SLC25A37 solute carrier family 25 (mitochondrial iron transporter), member 37
SMPD2 sphingomyelin phosphodiesterase 2, neutral membrane (neutral sphingomyelinase)
SNAP23 synaptosomal-associated protein, 23kDa
SPHK2 sphingosine kinase 2
SS18 synovial sarcoma translocation, chromosome 18
STON1 stonin 1
SULT1A2 sulfotransferase family, cytosolic, 1A, phenol-preferring, member 2
SVEP1 sushi, von Willebrand factor type A, EGF and pentraxin domain containing 1
TFCP2 transcription factor CP2
THBS3 thrombospondin 3
TLN2 talin 2
TMEM47 transmembrane protein 47
TRIM29 tripartite motif containing 29
TSPAN8 tetraspanin 8
UBE3B ubiquitin protein ligase E3B
URB1 URB1 ribosome biogenesis 1 homolog (S. cerevisiae)
WHSC1 Wolf-Hirschhorn syndrome candidate 1
YOD1 YOD1 deubiquitinase
ZNF174 zinc finger protein 174
ZNF197 zinc finger protein 197
ZNF227 zinc finger protein 227
ZNF415 zinc finger protein 415
ZNF589 zinc finger protein 589
ZNF675 zinc finger protein 675
ZNHIT2 zinc finger, HIT-type containing 2

decreased expression

Symbol Name
AGPAT3 1-acylglycerol-3-phosphate O-acyltransferase 3
AMT aminomethyltransferase
ANKRD40 ankyrin repeat domain 40
APOLD1 apolipoprotein L domain containing 1
ARHGAP10 Rho GTPase activating protein 10
ATP10D ATPase, class V, type 10D
BMP15 bone morphogenetic protein 15
C16ORF59 chromosome 16 open reading frame 59
C7ORF43 chromosome 7 open reading frame 43
C7ORF69 chromosome 7 open reading frame 69
CAMTA2 calmodulin binding transcription activator 2
CFD complement factor D (adipsin)
CHMP6 charged multivesicular body protein 6
CLCN5 chloride channel, voltage-sensitive 5
COG4 component of oligomeric golgi complex 4
CSGALNACT1 chondroitin sulfate N-acetylgalactosaminyltransferase 1
CUEDC1 CUE domain containing 1
DCLRE1A DNA cross-link repair 1A
DDX31 DEAD (Asp-Glu-Ala-Asp) box polypeptide 31
DMTF1 cyclin D binding myb-like transcription factor 1
DTWD1 DTW domain containing 1
EDC3 enhancer of mRNA decapping 3
EDN1 endothelin 1
EIF2AK2 eukaryotic translation initiation factor 2-alpha kinase 2
F3 coagulation factor III (thromboplastin, tissue factor)
FAM169A family with sequence similarity 169, member A
FBRS fibrosin
FLRT3 fibronectin leucine rich transmembrane protein 3
GPATCH2L G patch domain containing 2-like
GPR1 G protein-coupled receptor 1
GTF2H2B general transcription factor IIH, polypeptide 2B (pseudogene)
HSPA4L heat shock 70kDa protein 4-like
IFT88 intraflagellar transport 88
INPP5E inositol polyphosphate-5-phosphatase, 72 kDa
INPPL1 inositol polyphosphate phosphatase-like 1
KDM5C lysine (K)-specific demethylase 5C
KIAA0895 KIAA0895
KIAA1551 KIAA1551
KIFC1 kinesin family member C1
L2HGDH L-2-hydroxyglutarate dehydrogenase
LMNB1 lamin B1
LOC100272216 uncharacterized LOC100272216
MAGEH1 melanoma antigen family H1
MFGE8 milk fat globule-EGF factor 8 protein
NDUFAF7 NADH dehydrogenase (ubiquinone) complex I, assembly factor 7
NEIL3 nei endonuclease VIII-like 3 (E. coli)
NME6 NME/NM23 nucleoside diphosphate kinase 6
NPY1R neuropeptide Y receptor Y1
NR1D2 nuclear receptor subfamily 1, group D, member 2
NT5M 5',3'-nucleotidase, mitochondrial
OSMR oncostatin M receptor
PAN2 PAN2 poly(A) specific ribonuclease subunit
PBLD phenazine biosynthesis-like protein domain containing
PDGFRL platelet-derived growth factor receptor-like
PDLIM2 PDZ and LIM domain 2 (mystique)
PDZK1 PDZ domain containing 1
PILRB paired immunoglobin-like type 2 receptor beta
PTPRR protein tyrosine phosphatase, receptor type, R
PTTG3P pituitary tumor-transforming 3, pseudogene
RANBP17 RAN binding protein 17
RNASEH2B ribonuclease H2, subunit B
RSRC1 arginine/serine-rich coiled-coil 1
SCARA3 scavenger receptor class A, member 3
SCEL sciellin
SDC3 syndecan 3
SEC14L2 SEC14-like 2 (S. cerevisiae)
SHPK sedoheptulokinase
SLC12A8 solute carrier family 12, member 8
SLC2A6 solute carrier family 2 (facilitated glucose transporter), member 6
SLC39A7 solute carrier family 39 (zinc transporter), member 7
SNHG3 small nucleolar RNA host gene 3
SPSB1 splA/ryanodine receptor domain and SOCS box containing 1
SREK1IP1 SREK1-interacting protein 1
STAG3L4 stromal antigen 3-like 4 (pseudogene)
TCTN1 tectonic family member 1
TCTN2 tectonic family member 2
TGS1 trimethylguanosine synthase 1
TINAGL1 tubulointerstitial nephritis antigen-like 1
TMEM183A transmembrane protein 183A
TMEM209 transmembrane protein 209
TMEM260 transmembrane protein 260
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TRPM4 transient receptor potential cation channel, subfamily M, member 4
USF2 upstream transcription factor 2, c-fos interacting
VEGFB vascular endothelial growth factor B
WWC2 WW and C2 domain containing 2
XRCC1 X-ray repair complementing defective repair in Chinese hamster cells 1
YEATS2 YEATS domain containing 2
ZC3H12A zinc finger CCCH-type containing 12A
ZNF124 zinc finger protein 124
ZNF177 zinc finger protein 177
ZNF254 zinc finger protein 254
ZNF304 zinc finger protein 304
ZNF408 zinc finger protein 408
ZNF629 zinc finger protein 629
ZSCAN26 zinc finger and SCAN domain containing 26