pramocaine-2198 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the pramocaine-2198 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AAGAB alpha- and gamma-adaptin binding protein
ABCG4 ATP-binding cassette, sub-family G (WHITE), member 4
ABHD6 abhydrolase domain containing 6
ACRV1 acrosomal vesicle protein 1
ADAM5 ADAM metallopeptidase domain 5 (pseudogene)
APP amyloid beta (A4) precursor protein
ARHGEF38 Rho guanine nucleotide exchange factor (GEF) 38
ATP9B ATPase, class II, type 9B
BEST1 bestrophin 1
BGN biglycan
BIN1 bridging integrator 1
BIRC3 baculoviral IAP repeat containing 3
C11ORF16 chromosome 11 open reading frame 16
C7ORF69 chromosome 7 open reading frame 69
CD6 CD6 molecule
CDK10 cyclin-dependent kinase 10
CDKL3 cyclin-dependent kinase-like 3
CEACAM6 carcinoembryonic antigen-related cell adhesion molecule 6 (non-specific cross reacting antigen)
CFAP69 cilia and flagella associated protein 69
CHPF chondroitin polymerizing factor
CIB2 calcium and integrin binding family member 2
CLCA1 chloride channel accessory 1
CNTNAP1 contactin associated protein 1
CREM cAMP responsive element modulator
DBNDD1 dysbindin (dystrobrevin binding protein 1) domain containing 1
DDX3Y DEAD (Asp-Glu-Ala-Asp) box helicase 3, Y-linked
DHX34 DEAH (Asp-Glu-Ala-His) box polypeptide 34
DLGAP4 discs, large (Drosophila) homolog-associated protein 4
DNAJA4 DnaJ (Hsp40) homolog, subfamily A, member 4
ELSPBP1 epididymal sperm binding protein 1
EMID1 EMI domain containing 1
ENTPD1 ectonucleoside triphosphate diphosphohydrolase 1
EPHB1 EPH receptor B1
EPN2 epsin 2
ERBB2 erb-b2 receptor tyrosine kinase 2
FCN2 ficolin (collagen/fibrinogen domain containing lectin) 2
GNRHR gonadotropin-releasing hormone receptor
GOLGA2P5 golgin A2 pseudogene 5
GPC1 glypican 1
GPR137 G protein-coupled receptor 137
GRM3 glutamate receptor, metabotropic 3
HMOX2 heme oxygenase 2
HTR1F 5-hydroxytryptamine (serotonin) receptor 1F, G protein-coupled
IGLL1 immunoglobulin lambda-like polypeptide 1
IL1R2 interleukin 1 receptor, type II
IL24 interleukin 24
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KIAA0319L KIAA0319-like
KIDINS220 kinase D-interacting substrate, 220kDa
KIR2DL5A killer cell immunoglobulin-like receptor, two domains, long cytoplasmic tail, 5A
KLHL35 kelch-like family member 35
KLRG1 killer cell lectin-like receptor subfamily G, member 1
MINOS1P1 mitochondrial inner membrane organizing system 1 pseudogene 1
MLLT4 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 4
MMP14 matrix metallopeptidase 14 (membrane-inserted)
MUC8 mucin 8
MX1 MX dynamin-like GTPase 1
MYL4 myosin, light chain 4, alkali; atrial, embryonic
NAB2 NGFI-A binding protein 2 (EGR1 binding protein 2)
NOL10 nucleolar protein 10
NPY2R neuropeptide Y receptor Y2
PBX1 pre-B-cell leukemia homeobox 1
PDE4DIP phosphodiesterase 4D interacting protein
PDK4 pyruvate dehydrogenase kinase, isozyme 4
PHF7 PHD finger protein 7
PIGQ phosphatidylinositol glycan anchor biosynthesis, class Q
PLCG1 phospholipase C, gamma 1
POLL polymerase (DNA directed), lambda
PSEN2 presenilin 2
RAB40AL RAB40A, member RAS oncogene family-like
RPS6KA6 ribosomal protein S6 kinase, 90kDa, polypeptide 6
SFN stratifin
SIPA1L3 signal-induced proliferation-associated 1 like 3
SIX2 SIX homeobox 2
SLC16A5 solute carrier family 16 (monocarboxylate transporter), member 5
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SPRED2 sprouty-related, EVH1 domain containing 2
STAB2 stabilin 2
STOM stomatin
T T, brachyury homolog (mouse)
TAZ tafazzin
TCN1 transcobalamin I (vitamin B12 binding protein, R binder family)
TFAP2B transcription factor AP-2 beta (activating enhancer binding protein 2 beta)
TFF2 trefoil factor 2
THAP10 THAP domain containing 10
TM4SF5 transmembrane 4 L six family member 5
TMBIM1 transmembrane BAX inhibitor motif containing 1
TULP3 tubby like protein 3
UBOX5 U-box domain containing 5
VPS13A vacuolar protein sorting 13 homolog A (S. cerevisiae)
WDR4 WD repeat domain 4
ZC3H7B zinc finger CCCH-type containing 7B
ZER1 zyg-11 related, cell cycle regulator
ZMIZ2 zinc finger, MIZ-type containing 2
ZNF137P zinc finger protein 137, pseudogene
ZNF428 zinc finger protein 428
ZNF609 zinc finger protein 609
ZNF696 zinc finger protein 696
ZSCAN18 zinc finger and SCAN domain containing 18

decreased expression

Symbol Name
ABCC6 ATP-binding cassette, sub-family C (CFTR/MRP), member 6
ADAM23 ADAM metallopeptidase domain 23
ADGRE3 adhesion G protein-coupled receptor E3
AEN apoptosis enhancing nuclease
ANKRD2 ankyrin repeat domain 2 (stretch responsive muscle)
ARHGEF10L Rho guanine nucleotide exchange factor (GEF) 10-like
ARMC7 armadillo repeat containing 7
BTBD18 BTB (POZ) domain containing 18
C16ORF59 chromosome 16 open reading frame 59
C7ORF43 chromosome 7 open reading frame 43
CALCOCO1 calcium binding and coiled-coil domain 1
CAMK4 calcium/calmodulin-dependent protein kinase IV
CBY1 chibby homolog 1 (Drosophila)
CCDC132 coiled-coil domain containing 132
CCDC186 coiled-coil domain containing 186
CDA cytidine deaminase
CDR2L cerebellar degeneration-related protein 2-like
CEP41 centrosomal protein 41kDa
CHML choroideremia-like (Rab escort protein 2)
CHRNB1 cholinergic receptor, nicotinic, beta 1 (muscle)
CPTP ceramide-1-phosphate transfer protein
CRY2 cryptochrome circadian clock 2
CTAGE9 CTAGE family, member 9
DGAT1 diacylglycerol O-acyltransferase 1
DGKG diacylglycerol kinase, gamma 90kDa
EPHA4 EPH receptor A4
EPX eosinophil peroxidase
ERCC6L excision repair cross-complementation group 6-like
FAM204A family with sequence similarity 204, member A
FMOD fibromodulin
FZD6 frizzled class receptor 6
GEMIN8 gem (nuclear organelle) associated protein 8
GPR19 G protein-coupled receptor 19
GPR21 G protein-coupled receptor 21
GPR22 G protein-coupled receptor 22
GRPR gastrin-releasing peptide receptor
GRWD1 glutamate-rich WD repeat containing 1
GTF3C5 general transcription factor IIIC, polypeptide 5, 63kDa
HERC3 HECT and RLD domain containing E3 ubiquitin protein ligase 3
HIST1H1E histone cluster 1, H1e
HIST1H2AI histone cluster 1, H2ai
IL1RAPL2 interleukin 1 receptor accessory protein-like 2
INO80D INO80 complex subunit D
IQCC IQ motif containing C
KCNS1 potassium voltage-gated channel, modifier subfamily S, member 1
LAIR2 leukocyte-associated immunoglobulin-like receptor 2
LIMS2 LIM and senescent cell antigen-like domains 2
LRCH1 leucine-rich repeats and calponin homology (CH) domain containing 1
LTBP2 latent transforming growth factor beta binding protein 2
LZTS3 leucine zipper, putative tumor suppressor family member 3
MDM4 MDM4, p53 regulator
MEFV Mediterranean fever
METTL16 methyltransferase like 16
MFSD6 major facilitator superfamily domain containing 6
MKRN3 makorin ring finger protein 3
NAG18 NAG18 mRNA
NFKBIL1 nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor-like 1
OR7E47P olfactory receptor, family 7, subfamily E, member 47 pseudogene
PADI2 peptidyl arginine deiminase, type II
PARG poly (ADP-ribose) glycohydrolase
PDGFD platelet derived growth factor D
PER3 period circadian clock 3
PLP1 proteolipid protein 1
PORCN porcupine homolog (Drosophila)
PRKCE protein kinase C, epsilon
PRR7 proline rich 7 (synaptic)
PRSS12 protease, serine, 12 (neurotrypsin, motopsin)
QTRT1 queuine tRNA-ribosyltransferase 1
RAB13 RAB13, member RAS oncogene family
RAB3A RAB3A, member RAS oncogene family
RFPL3 ret finger protein-like 3
RNASE3 ribonuclease, RNase A family, 3
RNF121 ring finger protein 121
RNF126P1 ring finger protein 126 pseudogene 1
SAA4 serum amyloid A4, constitutive
SGCE sarcoglycan, epsilon
SLC12A8 solute carrier family 12, member 8
SLC22A5 solute carrier family 22 (organic cation/carnitine transporter), member 5
SLC7A2 solute carrier family 7 (cationic amino acid transporter, y+ system), member 2
SNAI1 snail family zinc finger 1
SP1 Sp1 transcription factor
SPR sepiapterin reductase (7,8-dihydrobiopterin:NADP+ oxidoreductase)
SYNDIG1 synapse differentiation inducing 1
TMEM212 transmembrane protein 212
TNFRSF13B tumor necrosis factor receptor superfamily, member 13B
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TP53I3 tumor protein p53 inducible protein 3
TRAIP TRAF interacting protein
TTC4 tetratricopeptide repeat domain 4
UAP1L1 UDP-N-acetylglucosamine pyrophosphorylase 1 like 1
VASH2 vasohibin 2
VASP vasodilator-stimulated phosphoprotein
VSIG10 V-set and immunoglobulin domain containing 10
XDH xanthine dehydrogenase
ZNF155 zinc finger protein 155
ZNF219 zinc finger protein 219
ZNF250 zinc finger protein 250
ZNF32 zinc finger protein 32
ZNF667 zinc finger protein 667