procaine-5430 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the procaine-5430 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
A4GNT alpha-1,4-N-acetylglucosaminyltransferase
ABCA7 ATP-binding cassette, sub-family A (ABC1), member 7
ABL2 ABL proto-oncogene 2, non-receptor tyrosine kinase
ADD2 adducin 2 (beta)
ADGRG3 adhesion G protein-coupled receptor G3
AP3B2 adaptor-related protein complex 3, beta 2 subunit
ARNT aryl hydrocarbon receptor nuclear translocator
AVPR1A arginine vasopressin receptor 1A
BMP8A bone morphogenetic protein 8a
C18ORF25 chromosome 18 open reading frame 25
C5AR1 complement component 5a receptor 1
CACNG1 calcium channel, voltage-dependent, gamma subunit 1
CADM3 cell adhesion molecule 3
CALD1 caldesmon 1
CD6 CD6 molecule
CD70 CD70 molecule
CEL carboxyl ester lipase
CHRNA3 cholinergic receptor, nicotinic, alpha 3 (neuronal)
CHRNA4 cholinergic receptor, nicotinic, alpha 4 (neuronal)
CLDN17 claudin 17
CLEC4E C-type lectin domain family 4, member E
CLSPN claspin
COMT catechol-O-methyltransferase
CORO2B coronin, actin binding protein, 2B
CR1 complement component (3b/4b) receptor 1 (Knops blood group)
CXORF21 chromosome X open reading frame 21
CYP24A1 cytochrome P450, family 24, subfamily A, polypeptide 1
DDX3Y DEAD (Asp-Glu-Ala-Asp) box helicase 3, Y-linked
DUSP1 dual specificity phosphatase 1
EFEMP2 EGF containing fibulin-like extracellular matrix protein 2
EHD2 EH-domain containing 2
ELL2 elongation factor, RNA polymerase II, 2
EML2 echinoderm microtubule associated protein like 2
FADS3 fatty acid desaturase 3
FBLN1 fibulin 1
FBXW7 F-box and WD repeat domain containing 7, E3 ubiquitin protein ligase
FOXG1 forkhead box G1
GH1 growth hormone 1
GJA4 gap junction protein, alpha 4, 37kDa
HBB hemoglobin, beta
HS3ST2 heparan sulfate (glucosamine) 3-O-sulfotransferase 2
HSD17B3 hydroxysteroid (17-beta) dehydrogenase 3
HSPA12A heat shock 70kDa protein 12A
IL20RA interleukin 20 receptor, alpha
KDM4B lysine (K)-specific demethylase 4B
LMF2 lipase maturation factor 2
LOC100129648 uncharacterized LOC100129648
LOC79999 uncharacterized LOC79999
MADCAM1 mucosal vascular addressin cell adhesion molecule 1
MAP3K13 mitogen-activated protein kinase kinase kinase 13
MRPL20 mitochondrial ribosomal protein L20
MSI1 musashi RNA-binding protein 1
MYH14 myosin, heavy chain 14, non-muscle
MYL10 myosin, light chain 10, regulatory
MYL4 myosin, light chain 4, alkali; atrial, embryonic
N4BP2L1 NEDD4 binding protein 2-like 1
NF1 neurofibromin 1
NFATC1 nuclear factor of activated T-cells, cytoplasmic, calcineurin-dependent 1
NRP2 neuropilin 2
NUP88 nucleoporin 88kDa
OSBP2 oxysterol binding protein 2
OTOR otoraplin
PCDH11Y protocadherin 11 Y-linked
PI15 peptidase inhibitor 15
PLTP phospholipid transfer protein
PLXNC1 plexin C1
PPFIBP2 PTPRF interacting protein, binding protein 2 (liprin beta 2)
PPP4R4 protein phosphatase 4, regulatory subunit 4
PROC protein C (inactivator of coagulation factors Va and VIIIa)
PTGER3 prostaglandin E receptor 3 (subtype EP3)
PTPN11 protein tyrosine phosphatase, non-receptor type 11
PYHIN1 pyrin and HIN domain family, member 1
REM1 RAS (RAD and GEM)-like GTP-binding 1
RIMS3 regulating synaptic membrane exocytosis 3
RUNX1 runt-related transcription factor 1
S100A7 S100 calcium binding protein A7
SERPINA1 serpin peptidase inhibitor, clade A (alpha-1 antiproteinase, antitrypsin), member 1
SERPINF1 serpin peptidase inhibitor, clade F (alpha-2 antiplasmin, pigment epithelium derived factor), member 1
SLC16A5 solute carrier family 16 (monocarboxylate transporter), member 5
SLC22A14 solute carrier family 22, member 14
SLC43A3 solute carrier family 43, member 3
SLCO1C1 solute carrier organic anion transporter family, member 1C1
SPOCK3 sparc/osteonectin, cwcv and kazal-like domains proteoglycan (testican) 3
SPTAN1 spectrin, alpha, non-erythrocytic 1
SZT2 seizure threshold 2 homolog (mouse)
TGM1 transglutaminase 1
TMBIM1 transmembrane BAX inhibitor motif containing 1
TMEM176A transmembrane protein 176A
TMEM212 transmembrane protein 212
TMOD2 tropomodulin 2 (neuronal)
UBXN1 UBX domain protein 1
UPK3B uroplakin 3B
UTRN utrophin
VN1R1 vomeronasal 1 receptor 1
VWA5A von Willebrand factor A domain containing 5A
ZFP2 ZFP2 zinc finger protein
ZFP64 ZFP64 zinc finger protein
ZNF132 zinc finger protein 132
ZXDB zinc finger, X-linked, duplicated B
ZZEF1 zinc finger, ZZ-type with EF-hand domain 1

decreased expression

Symbol Name
A2M alpha-2-macroglobulin
AKR1B1 aldo-keto reductase family 1, member B1 (aldose reductase)
ANP32A-IT1 ANP32A intronic transcript 1
ARMC4 armadillo repeat containing 4
ARRB1 arrestin, beta 1
ATP8B1 ATPase, aminophospholipid transporter, class I, type 8B, member 1
C10ORF95 chromosome 10 open reading frame 95
C1QTNF9B-AS1 C1QTNF9B antisense RNA 1
C2ORF68 chromosome 2 open reading frame 68
C8ORF60 chromosome 8 open reading frame 60
CA11 carbonic anhydrase XI
CCDC121 coiled-coil domain containing 121
CCP110 centriolar coiled coil protein 110kDa
CD82 CD82 molecule
CDK3 cyclin-dependent kinase 3
CFD complement factor D (adipsin)
CLCF1 cardiotrophin-like cytokine factor 1
DSE dermatan sulfate epimerase
FAM188A family with sequence similarity 188, member A
FMO4 flavin containing monooxygenase 4
GBP2 guanylate binding protein 2, interferon-inducible
GLRA1 glycine receptor, alpha 1
GPATCH2L G patch domain containing 2-like
GPR143 G protein-coupled receptor 143
GPR19 G protein-coupled receptor 19
HERC5 HECT and RLD domain containing E3 ubiquitin protein ligase 5
HIRA histone cell cycle regulator
HIST1H2AJ histone cluster 1, H2aj
HIST1H3B histone cluster 1, H3b
HIST1H3E histone cluster 1, H3e
HIST1H4A histone cluster 1, H4a
HIST1H4C histone cluster 1, H4c
IGFBP6 insulin-like growth factor binding protein 6
INPP5J inositol polyphosphate-5-phosphatase J
IRF2BP1 interferon regulatory factor 2 binding protein 1
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCNK12 potassium channel, two pore domain subfamily K, member 12
KIAA0754 KIAA0754
KLHL26 kelch-like family member 26
KLHL28 kelch-like family member 28
LINC00597 long intergenic non-protein coding RNA 597
LOC100286895 cell division cycle 27 homolog pseudogene
MAGI1 membrane associated guanylate kinase, WW and PDZ domain containing 1
MAGOHB mago-nashi homolog B (Drosophila)
MAP3K1 mitogen-activated protein kinase kinase kinase 1, E3 ubiquitin protein ligase
MAP3K14 mitogen-activated protein kinase kinase kinase 14
MAPK12 mitogen-activated protein kinase 12
MBTD1 mbt domain containing 1
METTL16 methyltransferase like 16
MICAL3 microtubule associated monooxygenase, calponin and LIM domain containing 3
MITF microphthalmia-associated transcription factor
MRPL41 mitochondrial ribosomal protein L41
MRPS18C mitochondrial ribosomal protein S18C
MYO1F myosin IF
N4BP3 NEDD4 binding protein 3
NIPAL2 NIPA-like domain containing 2
NOD1 nucleotide-binding oligomerization domain containing 1
NPFFR1 neuropeptide FF receptor 1
NR1D2 nuclear receptor subfamily 1, group D, member 2
PDE12 phosphodiesterase 12
PHC1 polyhomeotic homolog 1 (Drosophila)
PKD2 polycystic kidney disease 2 (autosomal dominant)
PLA2G3 phospholipase A2, group III
POLL polymerase (DNA directed), lambda
PRKCE protein kinase C, epsilon
PRRG2 proline rich Gla (G-carboxyglutamic acid) 2
RAB30 RAB30, member RAS oncogene family
RIN1 Ras and Rab interactor 1
RPGRIP1L RPGRIP1-like
RPL10L ribosomal protein L10-like
SAYSD1 SAYSVFN motif domain containing 1
SEMA4D sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4D
SENP7 SUMO1/sentrin specific peptidase 7
SH2B3 SH2B adaptor protein 3
SLC12A5 solute carrier family 12 (potassium/chloride transporter), member 5
SLC44A1 solute carrier family 44 (choline transporter), member 1
SLC8B1 solute carrier family 8 (sodium/lithium/calcium exchanger), member B1
SMARCD1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 1
SP1 Sp1 transcription factor
STAG3L1 stromal antigen 3-like 1 (pseudogene)
STEAP4 STEAP family member 4
STK16 serine/threonine kinase 16
TBC1D19 TBC1 domain family, member 19
TMEM53 transmembrane protein 53
TRIM36 tripartite motif containing 36
TRPV6 transient receptor potential cation channel, subfamily V, member 6
TSPAN5 tetraspanin 5
TTC30A tetratricopeptide repeat domain 30A
TTC33 tetratricopeptide repeat domain 33
TWISTNB TWIST neighbor
UBQLN4 ubiquilin 4
VEGFC vascular endothelial growth factor C
YEATS4 YEATS domain containing 4
ZC3H3 zinc finger CCCH-type containing 3
ZNF134 zinc finger protein 134
ZNF324 zinc finger protein 324
ZNF586 zinc finger protein 586