pyrithyldione-6801 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the pyrithyldione-6801 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADCY6 adenylate cyclase 6
ADGRL1 adhesion G protein-coupled receptor L1
ADRBK1 adrenergic, beta, receptor kinase 1
AKAP8L A kinase (PRKA) anchor protein 8-like
ALDH4A1 aldehyde dehydrogenase 4 family, member A1
AMT aminomethyltransferase
C11ORF95 chromosome 11 open reading frame 95
C14ORF79 chromosome 14 open reading frame 79
C1ORF105 chromosome 1 open reading frame 105
CD40 CD40 molecule, TNF receptor superfamily member 5
CD6 CD6 molecule
CHKB choline kinase beta
CLCN6 chloride channel, voltage-sensitive 6
CLIC2 chloride intracellular channel 2
COL11A2 collagen, type XI, alpha 2
COL5A2 collagen, type V, alpha 2
DAPK2 death-associated protein kinase 2
DCTN1 dynactin 1
DNAH17 dynein, axonemal, heavy chain 17
DNAJB12 DnaJ (Hsp40) homolog, subfamily B, member 12
DUSP13 dual specificity phosphatase 13
EDNRA endothelin receptor type A
EHBP1L1 EH domain binding protein 1-like 1
ELK3 ELK3, ETS-domain protein (SRF accessory protein 2)
EMID1 EMI domain containing 1
EXOSC2 exosome component 2
FAM174B family with sequence similarity 174, member B
FGF5 fibroblast growth factor 5
FLOT1 flotillin 1
FN1 fibronectin 1
FRS3 fibroblast growth factor receptor substrate 3
FSCN1 fascin actin-bundling protein 1
GALNT12 polypeptide N-acetylgalactosaminyltransferase 12
GNRHR gonadotropin-releasing hormone receptor
GPER1 G protein-coupled estrogen receptor 1
GSAP gamma-secretase activating protein
GSPT1 G1 to S phase transition 1
HCFC1 host cell factor C1
HIVEP3 human immunodeficiency virus type I enhancer binding protein 3
HLA-E major histocompatibility complex, class I, E
HMGA1 high mobility group AT-hook 1
HOXA4 homeobox A4
HOXB6 homeobox B6
IGHMBP2 immunoglobulin mu binding protein 2
INO80B INO80 complex subunit B
INPP5J inositol polyphosphate-5-phosphatase J
KIAA0040 KIAA0040
KIF26B kinesin family member 26B
KREMEN2 kringle containing transmembrane protein 2
LAT2 linker for activation of T cells family, member 2
LZTR1 leucine-zipper-like transcription regulator 1
MCOLN1 mucolipin 1
MET MET proto-oncogene, receptor tyrosine kinase
MMP16 matrix metallopeptidase 16 (membrane-inserted)
MOCS1 molybdenum cofactor synthesis 1
MST1R macrophage stimulating 1 receptor
NCAPH2 non-SMC condensin II complex, subunit H2
NFATC1 nuclear factor of activated T-cells, cytoplasmic, calcineurin-dependent 1
NPC1 Niemann-Pick disease, type C1
OR7A10 olfactory receptor, family 7, subfamily A, member 10
OXCT2 3-oxoacid CoA transferase 2
PADI3 peptidyl arginine deiminase, type III
PARG poly (ADP-ribose) glycohydrolase
PAX4 paired box 4
PDE4DIP phosphodiesterase 4D interacting protein
PIDD1 p53-induced death domain protein 1
PIGQ phosphatidylinositol glycan anchor biosynthesis, class Q
PIK3CD phosphatidylinositol-4,5-bisphosphate 3-kinase, catalytic subunit delta
PLCD1 phospholipase C, delta 1
PLEKHM2 pleckstrin homology domain containing, family M (with RUN domain) member 2
PLXND1 plexin D1
PMCHL1 pro-melanin-concentrating hormone-like 1, pseudogene
POLR2A polymerase (RNA) II (DNA directed) polypeptide A, 220kDa
PPP1R9A protein phosphatase 1, regulatory subunit 9A
PRDM2 PR domain containing 2, with ZNF domain
RASA3 RAS p21 protein activator 3
RECQL5 RecQ protein-like 5
RNF5 ring finger protein 5, E3 ubiquitin protein ligase
RTEL1 regulator of telomere elongation helicase 1
SAYSD1 SAYSVFN motif domain containing 1
SETD1B SET domain containing 1B
SHOX2 short stature homeobox 2
SIM2 single-minded family bHLH transcription factor 2
SLC39A9 solute carrier family 39, member 9
SOD2 superoxide dismutase 2, mitochondrial
SPTBN1 spectrin, beta, non-erythrocytic 1
STAT5B signal transducer and activator of transcription 5B
TGM2 transglutaminase 2
TICAM1 toll-like receptor adaptor molecule 1
TLDC1 TBC/LysM-associated domain containing 1
TNFAIP3 tumor necrosis factor, alpha-induced protein 3
TNS1 tensin 1
TTC38 tetratricopeptide repeat domain 38
URB1 URB1 ribosome biogenesis 1 homolog (S. cerevisiae)
USP20 ubiquitin specific peptidase 20
USP9Y ubiquitin specific peptidase 9, Y-linked
WDR62 WD repeat domain 62
ZNF287 zinc finger protein 287
ZNF34 zinc finger protein 34
ZNF350 zinc finger protein 350

decreased expression

Symbol Name
ADGRG2 adhesion G protein-coupled receptor G2
B3GNT3 UDP-GlcNAc:betaGal beta-1,3-N-acetylglucosaminyltransferase 3
BAG4 BCL2-associated athanogene 4
BCOR BCL6 corepressor
BST2 bone marrow stromal cell antigen 2
C11ORF30 chromosome 11 open reading frame 30
C19ORF40 chromosome 19 open reading frame 40
C22ORF46 chromosome 22 open reading frame 46
CCDC25 coiled-coil domain containing 25
CCP110 centriolar coiled coil protein 110kDa
CD83 CD83 molecule
CGA glycoprotein hormones, alpha polypeptide
CNPY3 canopy FGF signaling regulator 3
CORO7 coronin 7
CORT cortistatin
CTAGE9 CTAGE family, member 9
DCAF13 DDB1 and CUL4 associated factor 13
DVL1 dishevelled segment polarity protein 1
DYRK3 dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 3
EAF2 ELL associated factor 2
EHHADH enoyl-CoA, hydratase/3-hydroxyacyl CoA dehydrogenase
ELOVL4 ELOVL fatty acid elongase 4
FAM198B family with sequence similarity 198, member B
FBRS fibrosin
FBXW12 F-box and WD repeat domain containing 12
FLCN folliculin
GALE UDP-galactose-4-epimerase
GAMT guanidinoacetate N-methyltransferase
GPX2 glutathione peroxidase 2
GTF2A1 general transcription factor IIA, 1, 19/37kDa
HDAC5 histone deacetylase 5
HIST1H2AI histone cluster 1, H2ai
HIST1H2AJ histone cluster 1, H2aj
HIST1H4C histone cluster 1, H4c
HS1BP3 HCLS1 binding protein 3
ICK intestinal cell (MAK-like) kinase
IREB2 iron-responsive element binding protein 2
IRF2BP1 interferon regulatory factor 2 binding protein 1
KDM5C lysine (K)-specific demethylase 5C
KRT8P12 keratin 8 pseudogene 12
LIF leukemia inhibitory factor
LOC202181 SUMO-interacting motifs containing 1 pseudogene
LZTS3 leucine zipper, putative tumor suppressor family member 3
MAP9 microtubule-associated protein 9
MAPKBP1 mitogen-activated protein kinase binding protein 1
MEFV Mediterranean fever
MGC12488
MRPL52 mitochondrial ribosomal protein L52
MTERF1 mitochondrial transcription termination factor 1
MUM1 melanoma associated antigen (mutated) 1
NCALD neurocalcin delta
NDUFB6 NADH dehydrogenase (ubiquinone) 1 beta subcomplex, 6, 17kDa
NME5 NME/NM23 family member 5
NOL10 nucleolar protein 10
NUDT18 nudix (nucleoside diphosphate linked moiety X)-type motif 18
PIBF1 progesterone immunomodulatory binding factor 1
PLA2G4C phospholipase A2, group IVC (cytosolic, calcium-independent)
PLXNA3 plexin A3
POM121 POM121 transmembrane nucleoporin
POTEKP POTE ankyrin domain family, member K, pseudogene
RAB30 RAB30, member RAS oncogene family
RASAL1 RAS protein activator like 1 (GAP1 like)
RBL1 retinoblastoma-like 1
RCN1 reticulocalbin 1, EF-hand calcium binding domain
RFTN1 raftlin, lipid raft linker 1
RFXAP regulatory factor X-associated protein
RGS2 regulator of G-protein signaling 2
RIPK4 receptor-interacting serine-threonine kinase 4
S100A9 S100 calcium binding protein A9
SCD5 stearoyl-CoA desaturase 5
SCHIP1 schwannomin interacting protein 1
SECTM1 secreted and transmembrane 1
SEMA4D sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4D
SHARPIN SHANK-associated RH domain interactor
SLC2A8 solute carrier family 2 (facilitated glucose transporter), member 8
SLC9A3R2 solute carrier family 9, subfamily A (NHE3, cation proton antiporter 3), member 3 regulator 2
SLMO1 slowmo homolog 1 (Drosophila)
SPSB1 splA/ryanodine receptor domain and SOCS box containing 1
SPTLC3 serine palmitoyltransferase, long chain base subunit 3
STAG3L4 stromal antigen 3-like 4 (pseudogene)
STMN3 stathmin-like 3
TCHH trichohyalin
TCP10 t-complex 10
TMEM183A transmembrane protein 183A
TRPM4 transient receptor potential cation channel, subfamily M, member 4
TUBA3C tubulin, alpha 3c
UBE2L6 ubiquitin-conjugating enzyme E2L 6
USB1 U6 snRNA biogenesis 1
USP27X ubiquitin specific peptidase 27, X-linked
VCPIP1 valosin containing protein (p97)/p47 complex interacting protein 1
VGF VGF nerve growth factor inducible
VPS33A vacuolar protein sorting 33 homolog A (S. cerevisiae)
ZNF254 zinc finger protein 254
ZNF573 zinc finger protein 573
ZNF675 zinc finger protein 675
ZNF813 zinc finger protein 813
ZNF83 zinc finger protein 83