repaglinide-7216 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

195 genes differentially expressed following the repaglinide-7216 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AAGAB alpha- and gamma-adaptin binding protein
APLP1 amyloid beta (A4) precursor-like protein 1
APOD apolipoprotein D
ARHGEF1 Rho guanine nucleotide exchange factor (GEF) 1
ARHGEF4 Rho guanine nucleotide exchange factor (GEF) 4
ARMCX4 armadillo repeat containing, X-linked 4
ASAP3 ArfGAP with SH3 domain, ankyrin repeat and PH domain 3
BCL3 B-cell CLL/lymphoma 3
C5AR1 complement component 5a receptor 1
CALML3 calmodulin-like 3
CAMK2B calcium/calmodulin-dependent protein kinase II beta
CASP2 caspase 2, apoptosis-related cysteine peptidase
CBFA2T2 core-binding factor, runt domain, alpha subunit 2; translocated to, 2
CCDC28B coiled-coil domain containing 28B
CCHCR1 coiled-coil alpha-helical rod protein 1
CD58 CD58 molecule
CHST10 carbohydrate sulfotransferase 10
CLCA1 chloride channel accessory 1
CLCN7 chloride channel, voltage-sensitive 7
CPQ carboxypeptidase Q
CRTC1 CREB regulated transcription coactivator 1
DNAJA4 DnaJ (Hsp40) homolog, subfamily A, member 4
DYSF dysferlin
EPHB2 EPH receptor B2
EPS8L1 EPS8-like 1
EXOG endo/exonuclease (5'-3'), endonuclease G-like
EXPH5 exophilin 5
FCN1 ficolin (collagen/fibrinogen domain containing) 1
FUT7 fucosyltransferase 7 (alpha (1,3) fucosyltransferase)
GIMAP5 GTPase, IMAP family member 5
GPR15 G protein-coupled receptor 15
GPR68 G protein-coupled receptor 68
GRK5 G protein-coupled receptor kinase 5
GRM1 glutamate receptor, metabotropic 1
GRM4 glutamate receptor, metabotropic 4
HLCS holocarboxylase synthetase (biotin-(proprionyl-CoA-carboxylase (ATP-hydrolysing)) ligase)
HOXC8 homeobox C8
HSPA1L heat shock 70kDa protein 1-like
IFT122 intraflagellar transport 122
IGLJ3 immunoglobulin lambda joining 3
IL12RB1 interleukin 12 receptor, beta 1
INO80D INO80 complex subunit D
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KDM4C lysine (K)-specific demethylase 4C
KLHL22 kelch-like family member 22
KRT15 keratin 15, type I
LAMB4 laminin, beta 4
LAMP1 lysosomal-associated membrane protein 1
LIMK1 LIM domain kinase 1
LSM14B LSM14B, SCD6 homolog B (S. cerevisiae)
MAP2K5 mitogen-activated protein kinase kinase 5
MED16 mediator complex subunit 16
MGEA5 meningioma expressed antigen 5 (hyaluronidase)
MINK1 misshapen-like kinase 1
MLLT4 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 4
MXD4 MAX dimerization protein 4
NDOR1 NADPH dependent diflavin oxidoreductase 1
NDUFB7 NADH dehydrogenase (ubiquinone) 1 beta subcomplex, 7, 18kDa
NEK9 NIMA-related kinase 9
PGAM2 phosphoglycerate mutase 2 (muscle)
PLK4 polo-like kinase 4
PODNL1 podocan-like 1
PPAP2B phosphatidic acid phosphatase type 2B
PPP4R4 protein phosphatase 4, regulatory subunit 4
PRB1 proline-rich protein BstNI subfamily 1
PRDX2 peroxiredoxin 2
PRKAR1B protein kinase, cAMP-dependent, regulatory, type I, beta
PRODH proline dehydrogenase (oxidase) 1
PSG1 pregnancy specific beta-1-glycoprotein 1
PTBP3 polypyrimidine tract binding protein 3
PTCRA pre T-cell antigen receptor alpha
PTPN14 protein tyrosine phosphatase, non-receptor type 14
RAB40C RAB40C, member RAS oncogene family
RANBP3 RAN binding protein 3
RASGRP2 RAS guanyl releasing protein 2 (calcium and DAG-regulated)
RGS10 regulator of G-protein signaling 10
RGS12 regulator of G-protein signaling 12
RGS9 regulator of G-protein signaling 9
SCN10A sodium channel, voltage gated, type X alpha subunit
SDC3 syndecan 3
SEMA3F sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3F
SERPINB13 serpin peptidase inhibitor, clade B (ovalbumin), member 13
SIPA1L3 signal-induced proliferation-associated 1 like 3
SLC2A3 solute carrier family 2 (facilitated glucose transporter), member 3
SLC6A2 solute carrier family 6 (neurotransmitter transporter), member 2
SOCS1 suppressor of cytokine signaling 1
STC1 stanniocalcin 1
TFF2 trefoil factor 2
THBD thrombomodulin
TNFRSF9 tumor necrosis factor receptor superfamily, member 9
TONSL tonsoku-like, DNA repair protein
TTBK2 tau tubulin kinase 2
UCP1 uncoupling protein 1 (mitochondrial, proton carrier)
VAMP5 vesicle-associated membrane protein 5
VDR vitamin D (1,25- dihydroxyvitamin D3) receptor
WDR61 WD repeat domain 61
YTHDC1 YTH domain containing 1
ZNF749 zinc finger protein 749

decreased expression

Symbol Name
ACTN4 actinin, alpha 4
ACTR3B ARP3 actin-related protein 3 homolog B (yeast)
ACYP1 acylphosphatase 1, erythrocyte (common) type
ATAD5 ATPase family, AAA domain containing 5
BAHD1 bromo adjacent homology domain containing 1
BATF basic leucine zipper transcription factor, ATF-like
BCL9 B-cell CLL/lymphoma 9
C16ORF59 chromosome 16 open reading frame 59
CAMKMT calmodulin-lysine N-methyltransferase
CARM1 coactivator-associated arginine methyltransferase 1
CASZ1 castor zinc finger 1
CCDC88C coiled-coil domain containing 88C
CCNJ cyclin J
CCNO cyclin O
CFD complement factor D (adipsin)
CPPED1 calcineurin-like phosphoesterase domain containing 1
CUEDC1 CUE domain containing 1
DDX31 DEAD (Asp-Glu-Ala-Asp) box polypeptide 31
DHX35 DEAH (Asp-Glu-Ala-His) box polypeptide 35
DSCAM Down syndrome cell adhesion molecule
EGLN3 egl-9 family hypoxia-inducible factor 3
ELMO3 engulfment and cell motility 3
ELOVL4 ELOVL fatty acid elongase 4
EOGT EGF domain-specific O-linked N-acetylglucosamine (GlcNAc) transferase
EPB41L5 erythrocyte membrane protein band 4.1 like 5
FANCE Fanconi anemia, complementation group E
FBXL14 F-box and leucine-rich repeat protein 14
FBXO31 F-box protein 31
GAN gigaxonin
GNE glucosamine (UDP-N-acetyl)-2-epimerase/N-acetylmannosamine kinase
HEATR3 HEAT repeat containing 3
HGSNAT heparan-alpha-glucosaminide N-acetyltransferase
HPSE heparanase
INF2 inverted formin, FH2 and WH2 domain containing
IPPK inositol 1,3,4,5,6-pentakisphosphate 2-kinase
KCNN4 potassium channel, calcium activated intermediate/small conductance subfamily N alpha, member 4
KIAA0125 KIAA0125
KLHL12 kelch-like family member 12
LAMB3 laminin, beta 3
LOC202181 SUMO-interacting motifs containing 1 pseudogene
MAMLD1 mastermind-like domain containing 1
MAP3K6 mitogen-activated protein kinase kinase kinase 6
MAST3 microtubule associated serine/threonine kinase 3
MCOLN3 mucolipin 3
MEX3C mex-3 RNA binding family member C
MTHFSD methenyltetrahydrofolate synthetase domain containing
NABP2 nucleic acid binding protein 2
NACA2 nascent polypeptide-associated complex alpha subunit 2
NDE1 nudE neurodevelopment protein 1
OCEL1 occludin/ELL domain containing 1
OFD1 oral-facial-digital syndrome 1
OGDH oxoglutarate (alpha-ketoglutarate) dehydrogenase (lipoamide)
PARP16 poly (ADP-ribose) polymerase family, member 16
PC pyruvate carboxylase
PDP1 pyruvate dehyrogenase phosphatase catalytic subunit 1
PLA2G15 phospholipase A2, group XV
PTK6 protein tyrosine kinase 6
RASAL1 RAS protein activator like 1 (GAP1 like)
RBL1 retinoblastoma-like 1
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
RNF126P1 ring finger protein 126 pseudogene 1
RNF19A ring finger protein 19A, RBR E3 ubiquitin protein ligase
S100A4 S100 calcium binding protein A4
SCAI suppressor of cancer cell invasion
SCML2 sex comb on midleg-like 2 (Drosophila)
SECISBP2 SECIS binding protein 2
SH2B3 SH2B adaptor protein 3
SH2D4A SH2 domain containing 4A
SIK1 salt-inducible kinase 1
SLC17A5 solute carrier family 17 (acidic sugar transporter), member 5
SLC20A2 solute carrier family 20 (phosphate transporter), member 2
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SLC9A1 solute carrier family 9, subfamily A (NHE1, cation proton antiporter 1), member 1
SNAPC2 small nuclear RNA activating complex, polypeptide 2, 45kDa
SNIP1 Smad nuclear interacting protein 1
SPSB1 splA/ryanodine receptor domain and SOCS box containing 1
SREBF1 sterol regulatory element binding transcription factor 1
SUV39H2 suppressor of variegation 3-9 homolog 2 (Drosophila)
TBX19 T-box 19
THBS3 thrombospondin 3
TMEM115 transmembrane protein 115
TMEM184B transmembrane protein 184B
TNRC6B trinucleotide repeat containing 6B
TRAIP TRAF interacting protein
TRAPPC2 trafficking protein particle complex 2
TSC1 tuberous sclerosis 1
TUT1 terminal uridylyl transferase 1, U6 snRNA-specific
TWF2 twinfilin actin binding protein 2
UBQLN4 ubiquilin 4
UPP1 uridine phosphorylase 1
VWA1 von Willebrand factor A domain containing 1
XRCC1 X-ray repair complementing defective repair in Chinese hamster cells 1
ZC3H12A zinc finger CCCH-type containing 12A
ZNF280D zinc finger protein 280D
ZNF492 zinc finger protein 492
ZNF552 zinc finger protein 552
ZNF573 zinc finger protein 573