tamoxifen-2050 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the tamoxifen-2050 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
AKAP9 A kinase (PRKA) anchor protein 9
ALKBH4 alkB, alkylation repair homolog 4 (E. coli)
ANGPTL4 angiopoietin-like 4
ANK3 ankyrin 3, node of Ranvier (ankyrin G)
ARHGAP28 Rho GTPase activating protein 28
BBS9 Bardet-Biedl syndrome 9
BCL2L10 BCL2-like 10 (apoptosis facilitator)
BCORL1 BCL6 corepressor-like 1
C19ORF60 chromosome 19 open reading frame 60
C1QL1 complement component 1, q subcomponent-like 1
CASP1 caspase 1, apoptosis-related cysteine peptidase
CDKN1C cyclin-dependent kinase inhibitor 1C (p57, Kip2)
COA1 cytochrome c oxidase assembly factor 1 homolog (S. cerevisiae)
COL1A2 collagen, type I, alpha 2
COL3A1 collagen, type III, alpha 1
CREM cAMP responsive element modulator
DBT dihydrolipoamide branched chain transacylase E2
DDIT4 DNA-damage-inducible transcript 4
DESI2 desumoylating isopeptidase 2
EDAR ectodysplasin A receptor
EFNA3 ephrin-A3
ELK4 ELK4, ETS-domain protein (SRF accessory protein 1)
EPS8L1 EPS8-like 1
ERN2 endoplasmic reticulum to nucleus signaling 2
FCMR Fc fragment of IgM receptor
FKBP10 FK506 binding protein 10, 65 kDa
FOXG1 forkhead box G1
GHRHR growth hormone releasing hormone receptor
GK glycerol kinase
GLI2 GLI family zinc finger 2
GLYR1 glyoxylate reductase 1 homolog (Arabidopsis)
GPR19 G protein-coupled receptor 19
GPR85 G protein-coupled receptor 85
HABP4 hyaluronan binding protein 4
HLCS holocarboxylase synthetase (biotin-(proprionyl-CoA-carboxylase (ATP-hydrolysing)) ligase)
HMOX1 heme oxygenase 1
HOMER3 homer scaffolding protein 3
HTT huntingtin
IQCE IQ motif containing E
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KIAA1644 KIAA1644
KIF5C kinesin family member 5C
KLHL36 kelch-like family member 36
LINC00094 long intergenic non-protein coding RNA 94
LIPE lipase, hormone-sensitive
LRFN3 leucine rich repeat and fibronectin type III domain containing 3
LRP3 low density lipoprotein receptor-related protein 3
MAFF v-maf avian musculoaponeurotic fibrosarcoma oncogene homolog F
MAGOH2P mago-nashi homolog 2, pseudogene
MAPK12 mitogen-activated protein kinase 12
MOCS1 molybdenum cofactor synthesis 1
MTF1 metal-regulatory transcription factor 1
MUC1 mucin 1, cell surface associated
MYO9B myosin IXB
NAB2 NGFI-A binding protein 2 (EGR1 binding protein 2)
NADK NAD kinase
NEK3 NIMA-related kinase 3
OGT O-linked N-acetylglucosamine (GlcNAc) transferase
OR7E47P olfactory receptor, family 7, subfamily E, member 47 pseudogene
OVOL2 ovo-like zinc finger 2
PDGFRA platelet-derived growth factor receptor, alpha polypeptide
PGLYRP4 peptidoglycan recognition protein 4
PLXNB3 plexin B3
PODNL1 podocan-like 1
POLG polymerase (DNA directed), gamma
PPP1R13B protein phosphatase 1, regulatory subunit 13B
PTCH1 patched 1
PYHIN1 pyrin and HIN domain family, member 1
RAB27B RAB27B, member RAS oncogene family
RAB3B RAB3B, member RAS oncogene family
RGS4 regulator of G-protein signaling 4
RNF126P1 ring finger protein 126 pseudogene 1
ROR1 receptor tyrosine kinase-like orphan receptor 1
RPS4Y1 ribosomal protein S4, Y-linked 1
S1PR1 sphingosine-1-phosphate receptor 1
SCNN1B sodium channel, non voltage gated 1 beta subunit
SLC16A1 solute carrier family 16 (monocarboxylate transporter), member 1
SLC1A4 solute carrier family 1 (glutamate/neutral amino acid transporter), member 4
SLC7A7 solute carrier family 7 (amino acid transporter light chain, y+L system), member 7
SOX12 SRY (sex determining region Y)-box 12
STX6 syntaxin 6
STXBP6 syntaxin binding protein 6 (amisyn)
SUPT20H suppressor of Ty 20 homolog (S. cerevisiae)
SYNGR3 synaptogyrin 3
TAF13 TAF13 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 18kDa
TAF6L TAF6-like RNA polymerase II, p300/CBP-associated factor (PCAF)-associated factor, 65kDa
TAT tyrosine aminotransferase
TLR2 toll-like receptor 2
TM4SF1 transmembrane 4 L six family member 1
TNFSF10 tumor necrosis factor (ligand) superfamily, member 10
TRIM29 tripartite motif containing 29
TSNAXIP1 translin-associated factor X interacting protein 1
TUBG2 tubulin, gamma 2
USP12 ubiquitin specific peptidase 12
ZBTB20 zinc finger and BTB domain containing 20
ZMYM5 zinc finger, MYM-type 5
ZNF222 zinc finger protein 222
ZNF34 zinc finger protein 34
ZNF552 zinc finger protein 552

decreased expression

Symbol Name
ABTB2 ankyrin repeat and BTB (POZ) domain containing 2
ACYP2 acylphosphatase 2, muscle type
ADCY6 adenylate cyclase 6
ADPRM ADP-ribose/CDP-alcohol diphosphatase, manganese-dependent
AKR1B10 aldo-keto reductase family 1, member B10 (aldose reductase)
APH1B APH1B gamma secretase subunit
ARID4A AT rich interactive domain 4A (RBP1-like)
AUH AU RNA binding protein/enoyl-CoA hydratase
BAMBI BMP and activin membrane-bound inhibitor
C11ORF73 chromosome 11 open reading frame 73
C16ORF45 chromosome 16 open reading frame 45
C4ORF19 chromosome 4 open reading frame 19
CCDC130 coiled-coil domain containing 130
CCDC85C coiled-coil domain containing 85C
CCNA1 cyclin A1
CDK5RAP2 CDK5 regulatory subunit associated protein 2
CDKN2D cyclin-dependent kinase inhibitor 2D (p19, inhibits CDK4)
CEP131 centrosomal protein 131kDa
CHEK2 checkpoint kinase 2
CHST2 carbohydrate (N-acetylglucosamine-6-O) sulfotransferase 2
CLCN5 chloride channel, voltage-sensitive 5
CLIP4 CAP-GLY domain containing linker protein family, member 4
COMMD10 COMM domain containing 10
CRADD CASP2 and RIPK1 domain containing adaptor with death domain
CTSO cathepsin O
E4F1 E4F transcription factor 1
ECHDC1 ethylmalonyl-CoA decarboxylase 1
EDC3 enhancer of mRNA decapping 3
EDN1 endothelin 1
EGF epidermal growth factor
FAM222B family with sequence similarity 222, member B
FURIN furin (paired basic amino acid cleaving enzyme)
GSTZ1 glutathione S-transferase zeta 1
H2BFS H2B histone family, member S (pseudogene)
HIRA histone cell cycle regulator
HIST1H2BI histone cluster 1, H2bi
HPS6 Hermansky-Pudlak syndrome 6
HSD17B14 hydroxysteroid (17-beta) dehydrogenase 14
HSPA4L heat shock 70kDa protein 4-like
IFT81 intraflagellar transport 81
JMJD4 jumonji domain containing 4
KCTD7 potassium channel tetramerization domain containing 7
KIAA0753 KIAA0753
KLHL3 kelch-like family member 3
KPNA4 karyopherin alpha 4 (importin alpha 3)
KRT86 keratin 86, type II
LMNB1 lamin B1
LONRF3 LON peptidase N-terminal domain and ring finger 3
LSM2 LSM2 homolog, U6 small nuclear RNA associated (S. cerevisiae)
MFSD12 major facilitator superfamily domain containing 12
MRPL28 mitochondrial ribosomal protein L28
MYNN myoneurin
MYO19 myosin XIX
NME3 NME/NM23 nucleoside diphosphate kinase 3
NOL12 nucleolar protein 12
NPDC1 neural proliferation, differentiation and control, 1
NPY1R neuropeptide Y receptor Y1
NUBP2 nucleotide binding protein 2
NUDT2 nudix (nucleoside diphosphate linked moiety X)-type motif 2
OLFML2A olfactomedin-like 2A
PCSK7 proprotein convertase subtilisin/kexin type 7
PDGFD platelet derived growth factor D
PECR peroxisomal trans-2-enoyl-CoA reductase
PELI1 pellino E3 ubiquitin protein ligase 1
PEX26 peroxisomal biogenesis factor 26
PLA2G15 phospholipase A2, group XV
PLCB3 phospholipase C, beta 3 (phosphatidylinositol-specific)
PLEKHO2 pleckstrin homology domain containing, family O member 2
PRAME preferentially expressed antigen in melanoma
RAB8B RAB8B, member RAS oncogene family
RBM38 RNA binding motif protein 38
RBM41 RNA binding motif protein 41
SCNM1 sodium channel modifier 1
SCRN3 secernin 3
SLC37A1 solute carrier family 37 (glucose-6-phosphate transporter), member 1
SLC4A1AP solute carrier family 4 (anion exchanger), member 1, adaptor protein
SNX5 sorting nexin 5
SPATA7 spermatogenesis associated 7
SPECC1L sperm antigen with calponin homology and coiled-coil domains 1-like
SPEG SPEG complex locus
STIM1 stromal interaction molecule 1
TM7SF2 transmembrane 7 superfamily member 2
TMC5 transmembrane channel-like 5
TRIM21 tripartite motif containing 21
TSKU tsukushi, small leucine rich proteoglycan
USB1 U6 snRNA biogenesis 1
XRCC1 X-ray repair complementing defective repair in Chinese hamster cells 1
XRCC2 X-ray repair complementing defective repair in Chinese hamster cells 2
ZBTB3 zinc finger and BTB domain containing 3
ZBTB48 zinc finger and BTB domain containing 48
ZDHHC18 zinc finger, DHHC-type containing 18
ZFYVE16 zinc finger, FYVE domain containing 16
ZKSCAN3 zinc finger with KRAB and SCAN domains 3
ZNF350 zinc finger protein 350
ZNF574 zinc finger protein 574
ZNF665 zinc finger protein 665
ZNF8 zinc finger protein 8
ZNF804A zinc finger protein 804A
ZXDC ZXD family zinc finger C