tanespimycin-1006 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

199 genes differentially expressed following the tanespimycin-1006 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABHD3 abhydrolase domain containing 3
ABHD4 abhydrolase domain containing 4
ACVR1B activin A receptor, type IB
ADCY7 adenylate cyclase 7
ARHGAP35 Rho GTPase activating protein 35
B4GALNT1 beta-1,4-N-acetyl-galactosaminyl transferase 1
BAG2 BCL2-associated athanogene 2
BMP4 bone morphogenetic protein 4
BRF2 BRF2, RNA polymerase III transcription initiation factor 50 kDa subunit
BTN2A2 butyrophilin, subfamily 2, member A2
CAMK2G calcium/calmodulin-dependent protein kinase II gamma
CCDC81 coiled-coil domain containing 81
CCDC9 coiled-coil domain containing 9
CCNG2 cyclin G2
CHKB choline kinase beta
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
COL3A1 collagen, type III, alpha 1
CRELD1 cysteine-rich with EGF-like domains 1
CSRP2 cysteine and glycine-rich protein 2
DBP D site of albumin promoter (albumin D-box) binding protein
DDIT4 DNA-damage-inducible transcript 4
DIDO1 death inducer-obliterator 1
DMXL2 Dmx-like 2
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJC3 DnaJ (Hsp40) homolog, subfamily C, member 3
DPYSL4 dihydropyrimidinase-like 4
EDRF1 erythroid differentiation regulatory factor 1
ERP44 endoplasmic reticulum protein 44
FGFR2 fibroblast growth factor receptor 2
FKBP14 FK506 binding protein 14, 22 kDa
GBP2 guanylate binding protein 2, interferon-inducible
GLRX glutaredoxin (thioltransferase)
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HMGCS1 3-hydroxy-3-methylglutaryl-CoA synthase 1 (soluble)
HMOX1 heme oxygenase 1
HOXA1 homeobox A1
HSD17B7 hydroxysteroid (17-beta) dehydrogenase 7
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1
HSPA1A heat shock 70kDa protein 1A
HSPA1L heat shock 70kDa protein 1-like
HSPA4L heat shock 70kDa protein 4-like
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPH1 heat shock 105kDa/110kDa protein 1
HYOU1 hypoxia up-regulated 1
JAG1 jagged 1
KDELR3 KDEL (Lys-Asp-Glu-Leu) endoplasmic reticulum protein retention receptor 3
KDM8 lysine (K)-specific demethylase 8
LPIN1 lipin 1
LZTFL1 leucine zipper transcription factor-like 1
MANF mesencephalic astrocyte-derived neurotrophic factor
MBOAT7 membrane bound O-acyltransferase domain containing 7
MED6 mediator complex subunit 6
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11
N4BP2L2 NEDD4 binding protein 2-like 2
NAP1L2 nucleosome assembly protein 1-like 2
NR3C1 nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor)
OSBPL1A oxysterol binding protein-like 1A
OSGIN1 oxidative stress induced growth inhibitor 1
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PDE4DIP phosphodiesterase 4D interacting protein
PDIA4 protein disulfide isomerase family A, member 4
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PLA2G3 phospholipase A2, group III
POPDC3 popeye domain containing 3
RAB14 RAB14, member RAS oncogene family
RABGGTB Rab geranylgeranyltransferase, beta subunit
RFPL2 ret finger protein-like 2
RGS2 regulator of G-protein signaling 2
SDF2L1 stromal cell-derived factor 2-like 1
SEC24D SEC24 family member D
SEL1L sel-1 suppressor of lin-12-like (C. elegans)
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SH3BGR SH3 domain binding glutamate-rich protein
SIRT5 sirtuin 5
SLC1A4 solute carrier family 1 (glutamate/neutral amino acid transporter), member 4
SLC5A3 solute carrier family 5 (sodium/myo-inositol cotransporter), member 3
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMEK2 SMEK homolog 2, suppressor of mek1 (Dictyostelium)
SNAI2 snail family zinc finger 2
SNAPC3 small nuclear RNA activating complex, polypeptide 3, 50kDa
SSBP1 single-stranded DNA binding protein 1, mitochondrial
TAGLN transgelin
TES testin LIM domain protein
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TRABD TraB domain containing
TRAK1 trafficking protein, kinesin binding 1
TSPYL2 TSPY-like 2
ULBP2 UL16 binding protein 2
XIAP X-linked inhibitor of apoptosis, E3 ubiquitin protein ligase
ZBTB40 zinc finger and BTB domain containing 40
ZMYND8 zinc finger, MYND-type containing 8
ZNF10 zinc finger protein 10
ZNF165 zinc finger protein 165
ZNF227 zinc finger protein 227
ZNF230 zinc finger protein 230
ZNF329 zinc finger protein 329
ZNF76 zinc finger protein 76

decreased expression

Symbol Name
ACKR3 atypical chemokine receptor 3
AFAP1 actin filament associated protein 1
ARHGAP29 Rho GTPase activating protein 29
ARL15 ADP-ribosylation factor-like 15
BAK1 BCL2-antagonist/killer 1
BAMBI BMP and activin membrane-bound inhibitor
BIK BCL2-interacting killer (apoptosis-inducing)
C9ORF3 chromosome 9 open reading frame 3
CALHM2 calcium homeostasis modulator 2
CCDC88C coiled-coil domain containing 88C
CD302 CD302 molecule
CENPQ centromere protein Q
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CHST10 carbohydrate sulfotransferase 10
CISH cytokine inducible SH2-containing protein
CNNM3 cyclin and CBS domain divalent metal cation transport mediator 3
CRYBG3 beta-gamma crystallin domain containing 3
CTSK cathepsin K
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
CYP20A1 cytochrome P450, family 20, subfamily A, polypeptide 1
DNAAF2 dynein, axonemal, assembly factor 2
DUSP10 dual specificity phosphatase 10
DUSP8 dual specificity phosphatase 8
EGR3 early growth response 3
ERCC4 excision repair cross-complementation group 4
FJX1 four jointed box 1 (Drosophila)
FOXC1 forkhead box C1
GALK1 galactokinase 1
GPATCH3 G patch domain containing 3
GPR19 G protein-coupled receptor 19
GPRC5C G protein-coupled receptor, class C, group 5, member C
GUF1 GUF1 GTPase homolog (S. cerevisiae)
HIVEP1 human immunodeficiency virus type I enhancer binding protein 1
ID1 inhibitor of DNA binding 1, dominant negative helix-loop-helix protein
JUNB jun B proto-oncogene
KIZ kizuna centrosomal protein
KLF10 Kruppel-like factor 10
KLF11 Kruppel-like factor 11
KLF7 Kruppel-like factor 7 (ubiquitous)
KRI1 KRI1 homolog (S. cerevisiae)
LCP1 lymphocyte cytosolic protein 1 (L-plastin)
LIAS lipoic acid synthetase
LYPLA2P1 lysophospholipase II pseudogene 1
MAP1S microtubule-associated protein 1S
MB myoglobin
MED22 mediator complex subunit 22
MITF microphthalmia-associated transcription factor
MMACHC methylmalonic aciduria (cobalamin deficiency) cblC type, with homocystinuria
MT1HL1 metallothionein 1H-like 1
MTA2 metastasis associated 1 family, member 2
MTHFSD methenyltetrahydrofolate synthetase domain containing
MTRF1 mitochondrial translational release factor 1
MYC v-myc avian myelocytomatosis viral oncogene homolog
NABP2 nucleic acid binding protein 2
NFE2L3 nuclear factor, erythroid 2-like 3
NFKBIA nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, alpha
NUPL2 nucleoporin like 2
OXR1 oxidation resistance 1
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
PAQR6 progestin and adipoQ receptor family member VI
PCF11 PCF11 cleavage and polyadenylation factor subunit
PMCH pro-melanin-concentrating hormone
PMM1 phosphomannomutase 1
PMS1 PMS1 postmeiotic segregation increased 1 (S. cerevisiae)
PRKCD protein kinase C, delta
PWP2 PWP2 periodic tryptophan protein homolog (yeast)
RAD54L RAD54-like (S. cerevisiae)
RBM14 RNA binding motif protein 14
RGS16 regulator of G-protein signaling 16
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RHPN1-AS1 RHPN1 antisense RNA 1 (head to head)
RIBC2 RIB43A domain with coiled-coils 2
RPAP1 RNA polymerase II associated protein 1
RPP25 ribonuclease P/MRP 25kDa subunit
RRS1 RRS1 ribosome biogenesis regulator homolog (S. cerevisiae)
SCO2 SCO2 cytochrome c oxidase assembly protein
SECISBP2 SECIS binding protein 2
SEMA4C sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4C
SETMAR SET domain and mariner transposase fusion gene
SH2B2 SH2B adaptor protein 2
SIDT1 SID1 transmembrane family, member 1
SLC25A22 solute carrier family 25 (mitochondrial carrier: glutamate), member 22
SMAD7 SMAD family member 7
SMARCAL1 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a-like 1
SYTL2 synaptotagmin-like 2
TFRC transferrin receptor
TIPIN TIMELESS interacting protein
TMEM104 transmembrane protein 104
TMEM159 transmembrane protein 159
TPST1 tyrosylprotein sulfotransferase 1
TRAPPC12 trafficking protein particle complex 12
TSEN2 TSEN2 tRNA splicing endonuclease subunit
TTF2 transcription termination factor, RNA polymerase II
UAP1L1 UDP-N-acetylglucosamine pyrophosphorylase 1 like 1
UNC119 unc-119 homolog (C. elegans)
ZCCHC6 zinc finger, CCHC domain containing 6
ZNF623 zinc finger protein 623
ZNF669 zinc finger protein 669
ZNF721 zinc finger protein 721
ZXDC ZXD family zinc finger C