tanespimycin-1226 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the tanespimycin-1226 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABI3BP ABI family, member 3 (NESH) binding protein
ABL2 ABL proto-oncogene 2, non-receptor tyrosine kinase
ADAM22 ADAM metallopeptidase domain 22
AHSA1 AHA1, activator of heat shock 90kDa protein ATPase homolog 1 (yeast)
ALDH7A1 aldehyde dehydrogenase 7 family, member A1
ARHGAP44 Rho GTPase activating protein 44
B9D1 B9 protein domain 1
BAG3 BCL2-associated athanogene 3
C1ORF54 chromosome 1 open reading frame 54
CBFA2T2 core-binding factor, runt domain, alpha subunit 2; translocated to, 2
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
COL4A6 collagen, type IV, alpha 6
CPEB1 cytoplasmic polyadenylation element binding protein 1
CTGF connective tissue growth factor
CUL5 cullin 5
DHRS9 dehydrogenase/reductase (SDR family) member 9
DIDO1 death inducer-obliterator 1
DIO2 deiodinase, iodothyronine, type II
DMBT1 deleted in malignant brain tumors 1
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DUSP1 dual specificity phosphatase 1
EIF2S2 eukaryotic translation initiation factor 2, subunit 2 beta, 38kDa
ESR1 estrogen receptor 1
FBLN1 fibulin 1
GABARAPL1 GABA(A) receptor-associated protein like 1
GAL3ST4 galactose-3-O-sulfotransferase 4
GAS7 growth arrest-specific 7
GIT2 G protein-coupled receptor kinase interacting ArfGAP 2
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HMOX1 heme oxygenase 1
HSD17B2 hydroxysteroid (17-beta) dehydrogenase 2
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1
HSPA1A heat shock 70kDa protein 1A
HSPA4 heat shock 70kDa protein 4
HSPA4L heat shock 70kDa protein 4-like
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPB1 heat shock 27kDa protein 1
HSPB8 heat shock 22kDa protein 8
HSPH1 heat shock 105kDa/110kDa protein 1
IFT27 intraflagellar transport 27
IL7R interleukin 7 receptor
INO80B INO80 complex subunit B
INPP4A inositol polyphosphate-4-phosphatase, type I, 107kDa
ITIH2 inter-alpha-trypsin inhibitor heavy chain 2
KCNG1 potassium channel, voltage gated modifier subfamily G, member 1
KIF1A kinesin family member 1A
KLHL36 kelch-like family member 36
KRT6A keratin 6A, type II
LRRK1 leucine-rich repeat kinase 1
LY6G6C lymphocyte antigen 6 complex, locus G6C
MANF mesencephalic astrocyte-derived neurotrophic factor
MGEA5 meningioma expressed antigen 5 (hyaluronidase)
MUC5B mucin 5B, oligomeric mucus/gel-forming
NACA nascent polypeptide-associated complex alpha subunit
NCAPH2 non-SMC condensin II complex, subunit H2
NFATC3 nuclear factor of activated T-cells, cytoplasmic, calcineurin-dependent 3
NFYA nuclear transcription factor Y, alpha
NPHS2 nephrosis 2, idiopathic, steroid-resistant (podocin)
NR4A2 nuclear receptor subfamily 4, group A, member 2
NUP214 nucleoporin 214kDa
OASL 2'-5'-oligoadenylate synthetase-like
PDIA4 protein disulfide isomerase family A, member 4
PDZD2 PDZ domain containing 2
PGAP1 post-GPI attachment to proteins 1
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
PPP1R3C protein phosphatase 1, regulatory subunit 3C
PRAMEF11 PRAME family member 11
PSD4 pleckstrin and Sec7 domain containing 4
RABL6 RAB, member RAS oncogene family-like 6
RAD52 RAD52 homolog (S. cerevisiae)
RAPGEF5 Rap guanine nucleotide exchange factor (GEF) 5
RGS10 regulator of G-protein signaling 10
RHAG Rh-associated glycoprotein
RPL10 ribosomal protein L10
RPL23 ribosomal protein L23
RTEL1 regulator of telomere elongation helicase 1
SAT1 spermidine/spermine N1-acetyltransferase 1
SEC63 SEC63 homolog (S. cerevisiae)
SEMA3B sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3B
SERHL2 serine hydrolase-like 2
SERPINA1 serpin peptidase inhibitor, clade A (alpha-1 antiproteinase, antitrypsin), member 1
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SGSH N-sulfoglucosamine sulfohydrolase
SLC5A2 solute carrier family 5 (sodium/glucose cotransporter), member 2
STIP1 stress-induced phosphoprotein 1
TM4SF1 transmembrane 4 L six family member 1
TMEM50B transmembrane protein 50B
TRA2A transformer 2 alpha homolog (Drosophila)
TUT1 terminal uridylyl transferase 1, U6 snRNA-specific
UNKL unkempt family zinc finger-like
ZC3HAV1 zinc finger CCCH-type, antiviral 1
ZFP64 ZFP64 zinc finger protein
ZNF408 zinc finger protein 408
ZNF442 zinc finger protein 442
ZNF747 zinc finger protein 747
ZNF778 zinc finger protein 778
ZSCAN26 zinc finger and SCAN domain containing 26

decreased expression

Symbol Name
ABTB2 ankyrin repeat and BTB (POZ) domain containing 2
ANAPC2 anaphase promoting complex subunit 2
ARHGEF16 Rho guanine nucleotide exchange factor (GEF) 16
ARHGEF28 Rho guanine nucleotide exchange factor (GEF) 28
BDH1 3-hydroxybutyrate dehydrogenase, type 1
BLM Bloom syndrome, RecQ helicase-like
C11ORF68 chromosome 11 open reading frame 68
C16ORF59 chromosome 16 open reading frame 59
C1ORF56 chromosome 1 open reading frame 56
C9ORF114 chromosome 9 open reading frame 114
CABYR calcium binding tyrosine-(Y)-phosphorylation regulated
CDCA4 cell division cycle associated 4
CDKN1A cyclin-dependent kinase inhibitor 1A (p21, Cip1)
CENPT centromere protein T
CFAP44 cilia and flagella associated protein 44
CHPF chondroitin polymerizing factor
CLCN2 chloride channel, voltage-sensitive 2
CLCN5 chloride channel, voltage-sensitive 5
CNIH3 cornichon family AMPA receptor auxiliary protein 3
CSTF3 cleavage stimulation factor, 3' pre-RNA, subunit 3, 77kDa
CUEDC1 CUE domain containing 1
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
DAPP1 dual adaptor of phosphotyrosine and 3-phosphoinositides
DSN1 DSN1, MIS12 kinetochore complex component
DTL denticleless E3 ubiquitin protein ligase homolog (Drosophila)
E2F8 E2F transcription factor 8
EDC3 enhancer of mRNA decapping 3
EDC4 enhancer of mRNA decapping 4
EFNA3 ephrin-A3
EPPK1 epiplakin 1
ERF Ets2 repressor factor
ERN2 endoplasmic reticulum to nucleus signaling 2
ESRP2 epithelial splicing regulatory protein 2
FADS2 fatty acid desaturase 2
FAM57A family with sequence similarity 57, member A
FBXL7 F-box and leucine-rich repeat protein 7
FJX1 four jointed box 1 (Drosophila)
FSD1 fibronectin type III and SPRY domain containing 1
GABBR1 gamma-aminobutyric acid (GABA) B receptor, 1
HDAC3 histone deacetylase 3
HIST1H1D histone cluster 1, H1d
HIST1H2AM histone cluster 1, H2am
IMPDH1 IMP (inosine 5'-monophosphate) dehydrogenase 1
JUNB jun B proto-oncogene
KCNMB4 potassium channel subfamily M regulatory beta subunit 4
KIFC1 kinesin family member C1
KRT15 keratin 15, type I
LONRF3 LON peptidase N-terminal domain and ring finger 3
MAP3K14 mitogen-activated protein kinase kinase kinase 14
MAPK3 mitogen-activated protein kinase 3
MCM10 minichromosome maintenance complex component 10
MCOLN1 mucolipin 1
MICALL2 MICAL-like 2
MOXD1 monooxygenase, DBH-like 1
MPP3 membrane protein, palmitoylated 3 (MAGUK p55 subfamily member 3)
MXD3 MAX dimerization protein 3
NACC2 NACC family member 2, BEN and BTB (POZ) domain containing
NDRG1 N-myc downstream regulated 1
ORC1 origin recognition complex, subunit 1
OVGP1 oviductal glycoprotein 1, 120kDa
PAQR4 progestin and adipoQ receptor family member IV
PARP16 poly (ADP-ribose) polymerase family, member 16
PCF11 PCF11 cleavage and polyadenylation factor subunit
PCYT2 phosphate cytidylyltransferase 2, ethanolamine
POMT2 protein-O-mannosyltransferase 2
PPARG peroxisome proliferator-activated receptor gamma
PPRC1 peroxisome proliferator-activated receptor gamma, coactivator-related 1
PRR15L proline rich 15-like
PSKH1 protein serine kinase H1
PYCRL pyrroline-5-carboxylate reductase-like
RASSF8 Ras association (RalGDS/AF-6) domain family (N-terminal) member 8
RBM14 RNA binding motif protein 14
RBM15 RNA binding motif protein 15
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
RPL13P5 ribosomal protein L13 pseudogene 5
SETBP1 SET binding protein 1
SLC26A6 solute carrier family 26 (anion exchanger), member 6
SNPH syntaphilin
SOWAHC sosondowah ankyrin repeat domain family member C
SPATA2L spermatogenesis associated 2-like
SREK1IP1 SREK1-interacting protein 1
STAG3L1 stromal antigen 3-like 1 (pseudogene)
STIM1 stromal interaction molecule 1
TBX19 T-box 19
TEAD3 TEA domain family member 3
TICAM1 toll-like receptor adaptor molecule 1
TMEM104 transmembrane protein 104
TMEM156 transmembrane protein 156
TRIM21 tripartite motif containing 21
TUBB2B tubulin, beta 2B class IIb
TUFT1 tuftelin 1
TXNL4B thioredoxin-like 4B
ULK1 unc-51 like autophagy activating kinase 1
URM1 ubiquitin related modifier 1
USP6 ubiquitin specific peptidase 6
WASF1 WAS protein family, member 1
ZDHHC14 zinc finger, DHHC-type containing 14
ZNF143 zinc finger protein 143