tanespimycin-2678 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

195 genes differentially expressed following the tanespimycin-2678 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
A1CF APOBEC1 complementation factor
ABHD3 abhydrolase domain containing 3
ACPP acid phosphatase, prostate
AHCYL2 adenosylhomocysteinase-like 2
AHSA1 AHA1, activator of heat shock 90kDa protein ATPase homolog 1 (yeast)
ANGEL2 angel homolog 2 (Drosophila)
ANXA1 annexin A1
ARHGAP35 Rho GTPase activating protein 35
ARIH2 ariadne RBR E3 ubiquitin protein ligase 2
AURKA aurora kinase A
BAG3 BCL2-associated athanogene 3
BLZF1 basic leucine zipper nuclear factor 1
BST2 bone marrow stromal cell antigen 2
C21ORF2 chromosome 21 open reading frame 2
CACYBP calcyclin binding protein
CASP1 caspase 1, apoptosis-related cysteine peptidase
CCDC186 coiled-coil domain containing 186
CCNG2 cyclin G2
CCSER2 coiled-coil serine-rich protein 2
CD84 CD84 molecule
CDKN1C cyclin-dependent kinase inhibitor 1C (p57, Kip2)
CELA2A chymotrypsin-like elastase family, member 2A
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
CNNM4 cyclin and CBS domain divalent metal cation transport mediator 4
CRYZ crystallin, zeta (quinone reductase)
CYTH1 cytohesin 1
DGKG diacylglycerol kinase, gamma 90kDa
DHRS9 dehydrogenase/reductase (SDR family) member 9
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
EMILIN2 elastin microfibril interfacer 2
FAM13A family with sequence similarity 13, member A
FAS Fas cell surface death receptor
FCGR2A Fc fragment of IgG, low affinity IIa, receptor (CD32)
FCGR2C Fc fragment of IgG, low affinity IIc, receptor for (CD32) (gene/pseudogene)
FKBP4 FK506 binding protein 4, 59kDa
FOXO4 forkhead box O4
FZD3 frizzled class receptor 3
GABARAPL1 GABA(A) receptor-associated protein like 1
GLYR1 glyoxylate reductase 1 homolog (Arabidopsis)
GP1BB glycoprotein Ib (platelet), beta polypeptide
GRIN1 glutamate receptor, ionotropic, N-methyl D-aspartate 1
GTF3C3 general transcription factor IIIC, polypeptide 3, 102kDa
H2AFX H2A histone family, member X
HSP90AA1 heat shock protein 90kDa alpha (cytosolic), class A member 1
HSP90AB1 heat shock protein 90kDa alpha (cytosolic), class B member 1
HSPA4 heat shock 70kDa protein 4
HSPA4L heat shock 70kDa protein 4-like
HSPA8 heat shock 70kDa protein 8
HSPB1 heat shock 27kDa protein 1
HSPH1 heat shock 105kDa/110kDa protein 1
HUS1 HUS1 checkpoint homolog (S. pombe)
IL1R1 interleukin 1 receptor, type I
IL6ST interleukin 6 signal transducer
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KCTD20 potassium channel tetramerization domain containing 20
KIAA0513 KIAA0513
LHCGR luteinizing hormone/choriogonadotropin receptor
LILRA2 leukocyte immunoglobulin-like receptor, subfamily A (with TM domain), member 2
LIMK2 LIM domain kinase 2
MAOA monoamine oxidase A
MBNL2 muscleblind-like splicing regulator 2
MBOAT7 membrane bound O-acyltransferase domain containing 7
MCTP2 multiple C2 domains, transmembrane 2
MLXIPL MLX interacting protein-like
MS4A6A membrane-spanning 4-domains, subfamily A, member 6A
NR4A3 nuclear receptor subfamily 4, group A, member 3
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PAPPA2 pappalysin 2
PAPSS2 3'-phosphoadenosine 5'-phosphosulfate synthase 2
PCDHGA8 protocadherin gamma subfamily A, 8
PDE4B phosphodiesterase 4B, cAMP-specific
PDE4DIP phosphodiesterase 4D interacting protein
PDLIM5 PDZ and LIM domain 5
PHACTR1 phosphatase and actin regulator 1
PPID peptidylprolyl isomerase D
PRKACB protein kinase, cAMP-dependent, catalytic, beta
PTPN11 protein tyrosine phosphatase, non-receptor type 11
SCARB2 scavenger receptor class B, member 2
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SIPA1L1 signal-induced proliferation-associated 1 like 1
SLC12A7 solute carrier family 12 (potassium/chloride transporter), member 7
SLC15A2 solute carrier family 15 (oligopeptide transporter), member 2
SLC35D2 solute carrier family 35 (UDP-GlcNAc/UDP-glucose transporter), member D2
SNAP23 synaptosomal-associated protein, 23kDa
SPATS2L spermatogenesis associated, serine-rich 2-like
ST13 suppression of tumorigenicity 13 (colon carcinoma) (Hsp70 interacting protein)
STAM2 signal transducing adaptor molecule (SH3 domain and ITAM motif) 2
STIP1 stress-induced phosphoprotein 1
STX11 syntaxin 11
THAP10 THAP domain containing 10
THBS1 thrombospondin 1
TRD T cell receptor delta locus
TRPS1 trichorhinophalangeal syndrome I
ZBTB38 zinc finger and BTB domain containing 38
ZER1 zyg-11 related, cell cycle regulator
ZSCAN26 zinc finger and SCAN domain containing 26

decreased expression

Symbol Name
ADRB2 adrenoceptor beta 2, surface
AEN apoptosis enhancing nuclease
ATF3 activating transcription factor 3
BATF3 basic leucine zipper transcription factor, ATF-like 3
BHLHE41 basic helix-loop-helix family, member e41
C10ORF2 chromosome 10 open reading frame 2
C7ORF69 chromosome 7 open reading frame 69
CCBL1 cysteine conjugate-beta lyase, cytoplasmic
CCDC86 coiled-coil domain containing 86
CD3EAP CD3e molecule, epsilon associated protein
CDR2L cerebellar degeneration-related protein 2-like
CEL carboxyl ester lipase
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CHST12 carbohydrate (chondroitin 4) sulfotransferase 12
CLEC2D C-type lectin domain family 2, member D
CPTP ceramide-1-phosphate transfer protein
DDN dendrin
DSPP dentin sialophosphoprotein
DUSP2 dual specificity phosphatase 2
DUSP8 dual specificity phosphatase 8
DVL1 dishevelled segment polarity protein 1
EEF2KMT eukaryotic elongation factor 2 lysine methyltransferase
ENDOG endonuclease G
ENTPD5 ectonucleoside triphosphate diphosphohydrolase 5
EXOSC5 exosome component 5
F3 coagulation factor III (thromboplastin, tissue factor)
FAM86B1 family with sequence similarity 86, member B1
FGF23 fibroblast growth factor 23
FICD FIC domain containing
FJX1 four jointed box 1 (Drosophila)
FLT4 fms-related tyrosine kinase 4
FOSL1 FOS-like antigen 1
GSTZ1 glutathione S-transferase zeta 1
HAMP hepcidin antimicrobial peptide
HDAC9 histone deacetylase 9
HOMER1 homer scaffolding protein 1
INHBE inhibin, beta E
KIAA1024 KIAA1024
KIAA1456 KIAA1456
KIF21B kinesin family member 21B
KLF13 Kruppel-like factor 13
KPTN kaptin (actin binding protein)
LRRC20 leucine rich repeat containing 20
LY6D lymphocyte antigen 6 complex, locus D
MBL1P mannose-binding lectin (protein A) 1, pseudogene
MNT MAX network transcriptional repressor
MRPS18C mitochondrial ribosomal protein S18C
MTSS1L metastasis suppressor 1-like
MXD3 MAX dimerization protein 3
MYC v-myc avian myelocytomatosis viral oncogene homolog
MYL5 myosin, light chain 5, regulatory
NAG18 NAG18 mRNA
NARFL nuclear prelamin A recognition factor-like
NOL6 nucleolar protein 6 (RNA-associated)
NR1D2 nuclear receptor subfamily 1, group D, member 2
NSMF NMDA receptor synaptonuclear signaling and neuronal migration factor
NT5E 5'-nucleotidase, ecto (CD73)
NTSR1 neurotensin receptor 1 (high affinity)
NXT1 nuclear transport factor 2-like export factor 1
P2RY6 pyrimidinergic receptor P2Y, G-protein coupled, 6
PAQR6 progestin and adipoQ receptor family member VI
PGP phosphoglycolate phosphatase
PIGH phosphatidylinositol glycan anchor biosynthesis, class H
PKD2L2 polycystic kidney disease 2-like 2
POLH polymerase (DNA directed), eta
POTEKP POTE ankyrin domain family, member K, pseudogene
PPRC1 peroxisome proliferator-activated receptor gamma, coactivator-related 1
PRDM13 PR domain containing 13
PUS1 pseudouridylate synthase 1
PYCR1 pyrroline-5-carboxylate reductase 1
RCL1 RNA terminal phosphate cyclase-like 1
RFXAP regulatory factor X-associated protein
RGS16 regulator of G-protein signaling 16
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RPS6KA4 ribosomal protein S6 kinase, 90kDa, polypeptide 4
RRP9 ribosomal RNA processing 9, small subunit (SSU) processome component, homolog (yeast)
RUSC2 RUN and SH3 domain containing 2
SIGIRR single immunoglobulin and toll-interleukin 1 receptor (TIR) domain
SLC1A5 solute carrier family 1 (neutral amino acid transporter), member 5
SLCO4A1 solute carrier organic anion transporter family, member 4A1
SMAD7 SMAD family member 7
SMR3A submaxillary gland androgen regulated protein 3A
SOX12 SRY (sex determining region Y)-box 12
STAG3L1 stromal antigen 3-like 1 (pseudogene)
STC2 stanniocalcin 2
TERT telomerase reverse transcriptase
TFAP4 transcription factor AP-4 (activating enhancer binding protein 4)
TIMM8A translocase of inner mitochondrial membrane 8 homolog A (yeast)
TMEM120B transmembrane protein 120B
TMEM159 transmembrane protein 159
TNF tumor necrosis factor
TRAIP TRAF interacting protein
TRIB3 tribbles pseudokinase 3
USP36 ubiquitin specific peptidase 36
ZNF250 zinc finger protein 250
ZNF580 zinc finger protein 580
ZNF696 zinc finger protein 696