tanespimycin-5203 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

196 genes differentially expressed following the tanespimycin-5203 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABHD3 abhydrolase domain containing 3
ADCY7 adenylate cyclase 7
ADM adrenomedullin
ALOXE3 arachidonate lipoxygenase 3
BAG2 BCL2-associated athanogene 2
BBC3 BCL2 binding component 3
BIN1 bridging integrator 1
BLZF1 basic leucine zipper nuclear factor 1
BST2 bone marrow stromal cell antigen 2
BTN2A2 butyrophilin, subfamily 2, member A2
C11ORF73 chromosome 11 open reading frame 73
CACYBP calcyclin binding protein
CASP7 caspase 7, apoptosis-related cysteine peptidase
CCNG2 cyclin G2
CD6 CD6 molecule
CDH6 cadherin 6, type 2, K-cadherin (fetal kidney)
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
CHRM3 cholinergic receptor, muscarinic 3
CLCN6 chloride channel, voltage-sensitive 6
CLU clusterin
CRY2 cryptochrome circadian clock 2
CSRP2 cysteine and glycine-rich protein 2
CUL7 cullin 7
CXCR4 chemokine (C-X-C motif) receptor 4
DAGLA diacylglycerol lipase, alpha
DDIT4 DNA-damage-inducible transcript 4
DHRS2 dehydrogenase/reductase (SDR family) member 2
DIO2 deiodinase, iodothyronine, type II
DIP2C DIP2 disco-interacting protein 2 homolog C (Drosophila)
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJB5 DnaJ (Hsp40) homolog, subfamily B, member 5
EDRF1 erythroid differentiation regulatory factor 1
EFNB3 ephrin-B3
EHD2 EH-domain containing 2
ERP44 endoplasmic reticulum protein 44
FGF18 fibroblast growth factor 18
FGFR2 fibroblast growth factor receptor 2
GEM GTP binding protein overexpressed in skeletal muscle
GTF3C3 general transcription factor IIIC, polypeptide 3, 102kDa
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HMOX1 heme oxygenase 1
HSPA1A heat shock 70kDa protein 1A
HSPA4L heat shock 70kDa protein 4-like
HSPA5 heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPH1 heat shock 105kDa/110kDa protein 1
IFT27 intraflagellar transport 27
IRS2 insulin receptor substrate 2
JAG1 jagged 1
KLK6 kallikrein-related peptidase 6
LAT2 linker for activation of T cells family, member 2
LRRC61 leucine rich repeat containing 61
ME1 malic enzyme 1, NADP(+)-dependent, cytosolic
MED16 mediator complex subunit 16
MICB MHC class I polypeptide-related sequence B
MKNK2 MAP kinase interacting serine/threonine kinase 2
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11
N4BP2L2 NEDD4 binding protein 2-like 2
NAP1L2 nucleosome assembly protein 1-like 2
NBL1 neuroblastoma 1, DAN family BMP antagonist
NOX1 NADPH oxidase 1
NPR3 natriuretic peptide receptor 3
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PLA2G3 phospholipase A2, group III
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1
PON3 paraoxonase 3
PRKD2 protein kinase D2
PRMT2 protein arginine methyltransferase 2
PRSS16 protease, serine, 16 (thymus)
RABGGTB Rab geranylgeranyltransferase, beta subunit
RCAN1 regulator of calcineurin 1
RFPL2 ret finger protein-like 2
RGS2 regulator of G-protein signaling 2
RNASE4 ribonuclease, RNase A family, 4
SEL1L sel-1 suppressor of lin-12-like (C. elegans)
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SH3BGR SH3 domain binding glutamate-rich protein
SIGLEC5 sialic acid binding Ig-like lectin 5
SLC5A3 solute carrier family 5 (sodium/myo-inositol cotransporter), member 3
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMEK2 SMEK homolog 2, suppressor of mek1 (Dictyostelium)
SOCS6 suppressor of cytokine signaling 6
SORBS1 sorbin and SH3 domain containing 1
SOX9 SRY (sex determining region Y)-box 9
STYK1 serine/threonine/tyrosine kinase 1
TES testin LIM domain protein
TMEM97 transmembrane protein 97
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TSPYL4 TSPY-like 4
ZEB1 zinc finger E-box binding homeobox 1
ZNF10 zinc finger protein 10
ZNF155 zinc finger protein 155
ZNF165 zinc finger protein 165
ZNF222 zinc finger protein 222
ZNF227 zinc finger protein 227
ZNF235 zinc finger protein 235
ZNF329 zinc finger protein 329
ZNF862 zinc finger protein 862

decreased expression

Symbol Name
ACKR3 atypical chemokine receptor 3
ADAM15 ADAM metallopeptidase domain 15
ANKRD36 ankyrin repeat domain 36
ANKRD36B ankyrin repeat domain 36B
ANP32A-IT1 ANP32A intronic transcript 1
ATAD5 ATPase family, AAA domain containing 5
BLM Bloom syndrome, RecQ helicase-like
C11ORF68 chromosome 11 open reading frame 68
C1ORF35 chromosome 1 open reading frame 35
C9ORF3 chromosome 9 open reading frame 3
CCNT1 cyclin T1
CDK5 cyclin-dependent kinase 5
CLCN2 chloride channel, voltage-sensitive 2
CLDN9 claudin 9
COA7 cytochrome c oxidase assembly factor 7 (putative)
CORO2A coronin, actin binding protein, 2A
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
DDX58 DEAD (Asp-Glu-Ala-Asp) box polypeptide 58
DLEU1 deleted in lymphocytic leukemia 1 (non-protein coding)
DZANK1 double zinc ribbon and ankyrin repeat domains 1
EEF2KMT eukaryotic elongation factor 2 lysine methyltransferase
EGR3 early growth response 3
ELP3 elongator acetyltransferase complex subunit 3
ENTPD5 ectonucleoside triphosphate diphosphohydrolase 5
ERCC4 excision repair cross-complementation group 4
ERF Ets2 repressor factor
FAN1 FANCD2/FANCI-associated nuclease 1
FKBP5 FK506 binding protein 5
GLS2 glutaminase 2 (liver, mitochondrial)
GPR19 G protein-coupled receptor 19
HLA-DRB1 major histocompatibility complex, class II, DR beta 1
ID1 inhibitor of DNA binding 1, dominant negative helix-loop-helix protein
IER2 immediate early response 2
IL17RB interleukin 17 receptor B
IRX5 iroquois homeobox 5
JUNB jun B proto-oncogene
KLF10 Kruppel-like factor 10
KLF11 Kruppel-like factor 11
LOC390998 ribosomal protein L10 pseudogene
METTL8 methyltransferase like 8
MICALL2 MICAL-like 2
MMP9 matrix metallopeptidase 9
MYC v-myc avian myelocytomatosis viral oncogene homolog
NFKBIA nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, alpha
NRIP1 nuclear receptor interacting protein 1
NUPL2 nucleoporin like 2
NXT1 nuclear transport factor 2-like export factor 1
OSGEPL1 O-sialoglycoprotein endopeptidase-like 1
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
PAGR1 PAXIP1 associated glutamate-rich protein 1
PALB2 partner and localizer of BRCA2
PARD6A par-6 family cell polarity regulator alpha
PCF11 PCF11 cleavage and polyadenylation factor subunit
PMS1 PMS1 postmeiotic segregation increased 1 (S. cerevisiae)
POLR1B polymerase (RNA) I polypeptide B, 128kDa
POLR1E polymerase (RNA) I polypeptide E, 53kDa
POLR3D polymerase (RNA) III (DNA directed) polypeptide D, 44kDa
PPRC1 peroxisome proliferator-activated receptor gamma, coactivator-related 1
PRKCD protein kinase C, delta
PYCRL pyrroline-5-carboxylate reductase-like
RAB27B RAB27B, member RAS oncogene family
RAB4B RAB4B, member RAS oncogene family
RASSF1 Ras association (RalGDS/AF-6) domain family member 1
RGS16 regulator of G-protein signaling 16
RHBDF2 rhomboid 5 homolog 2 (Drosophila)
RIBC2 RIB43A domain with coiled-coils 2
RIPK1 receptor (TNFRSF)-interacting serine-threonine kinase 1
RPAP2 RNA polymerase II associated protein 2
RPGR retinitis pigmentosa GTPase regulator
RPP25 ribonuclease P/MRP 25kDa subunit
RRS1 RRS1 ribosome biogenesis regulator homolog (S. cerevisiae)
SCO2 SCO2 cytochrome c oxidase assembly protein
SETMAR SET domain and mariner transposase fusion gene
SIX1 SIX homeobox 1
SLC25A28 solute carrier family 25 (mitochondrial iron transporter), member 28
SLC27A3 solute carrier family 27 (fatty acid transporter), member 3
SLC29A3 solute carrier family 29 (equilibrative nucleoside transporter), member 3
SMAD7 SMAD family member 7
SMU1 smu-1 suppressor of mec-8 and unc-52 homolog (C. elegans)
SOWAHC sosondowah ankyrin repeat domain family member C
SPATA2L spermatogenesis associated 2-like
SYTL2 synaptotagmin-like 2
TAF15 TAF15 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 68kDa
TAF4B TAF4b RNA polymerase II, TATA box binding protein (TBP)-associated factor, 105kDa
TIPIN TIMELESS interacting protein
TMEM180 transmembrane protein 180
UAP1L1 UDP-N-acetylglucosamine pyrophosphorylase 1 like 1
UBE2G2 ubiquitin-conjugating enzyme E2G 2
WDR4 WD repeat domain 4
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZBTB39 zinc finger and BTB domain containing 39
ZBTB48 zinc finger and BTB domain containing 48
ZNF124 zinc finger protein 124
ZNF276 zinc finger protein 276
ZNF573 zinc finger protein 573
ZXDC ZXD family zinc finger C