tanespimycin-5578 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the tanespimycin-5578 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADCY7 adenylate cyclase 7
ALS2CL ALS2 C-terminal like
BAG2 BCL2-associated athanogene 2
BIN1 bridging integrator 1
BST2 bone marrow stromal cell antigen 2
CASP4 caspase 4, apoptosis-related cysteine peptidase
CCNG2 cyclin G2
CCNJL cyclin J-like
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
CHRM3 cholinergic receptor, muscarinic 3
CNTN5 contactin 5
COBLL1 cordon-bleu WH2 repeat protein-like 1
CPEB3 cytoplasmic polyadenylation element binding protein 3
CSRP2 cysteine and glycine-rich protein 2
DCBLD2 discoidin, CUB and LCCL domain containing 2
DDIT4 DNA-damage-inducible transcript 4
DGAT1 diacylglycerol O-acyltransferase 1
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJB5 DnaJ (Hsp40) homolog, subfamily B, member 5
DTX2 deltex 2, E3 ubiquitin ligase
DYSF dysferlin
EPN1 epsin 1
FGFR2 fibroblast growth factor receptor 2
FGL2 fibrinogen-like 2
FSCN2 fascin actin-bundling protein 2, retinal
GADD45GIP1 growth arrest and DNA-damage-inducible, gamma interacting protein 1
GJA9 gap junction protein, alpha 9, 59kDa
GJB5 gap junction protein, beta 5, 31.1kDa
GP2 glycoprotein 2 (zymogen granule membrane)
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HSPA1A heat shock 70kDa protein 1A
HSPA4L heat shock 70kDa protein 4-like
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPH1 heat shock 105kDa/110kDa protein 1
IL6R interleukin 6 receptor
ING4 inhibitor of growth family, member 4
ITGA9 integrin, alpha 9
KCNJ5 potassium channel, inwardly rectifying subfamily J, member 5
KRT16 keratin 16, type I
LDLR low density lipoprotein receptor
MAN1A2 mannosidase, alpha, class 1A, member 2
MAP1B microtubule-associated protein 1B
MAPK11 mitogen-activated protein kinase 11
MAPRE3 microtubule-associated protein, RP/EB family, member 3
MBNL2 muscleblind-like splicing regulator 2
MDM2 MDM2 proto-oncogene, E3 ubiquitin protein ligase
MED16 mediator complex subunit 16
MKL1 megakaryoblastic leukemia (translocation) 1
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11
MXD4 MAX dimerization protein 4
NAP1L2 nucleosome assembly protein 1-like 2
NBL1 neuroblastoma 1, DAN family BMP antagonist
NPR1 natriuretic peptide receptor 1
NPR3 natriuretic peptide receptor 3
NR3C1 nuclear receptor subfamily 3, group C, member 1 (glucocorticoid receptor)
NUP50 nucleoporin 50kDa
OPLAH 5-oxoprolinase (ATP-hydrolysing)
OSBPL1A oxysterol binding protein-like 1A
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PHLPP2 PH domain and leucine rich repeat protein phosphatase 2
PMAIP1 phorbol-12-myristate-13-acetate-induced protein 1
POPDC3 popeye domain containing 3
PPID peptidylprolyl isomerase D
PSAT1 phosphoserine aminotransferase 1
RBM12B RNA binding motif protein 12B
RFPL2 ret finger protein-like 2
RGS2 regulator of G-protein signaling 2
RNASE4 ribonuclease, RNase A family, 4
RRN3P1 RNA polymerase I transcription factor homolog (S. cerevisiae) pseudogene 1
SEL1L sel-1 suppressor of lin-12-like (C. elegans)
SEMA4G sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4G
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SH3BGR SH3 domain binding glutamate-rich protein
SIRT5 sirtuin 5
SLC5A3 solute carrier family 5 (sodium/myo-inositol cotransporter), member 3
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SNAP23 synaptosomal-associated protein, 23kDa
SORBS1 sorbin and SH3 domain containing 1
SPIB Spi-B transcription factor (Spi-1/PU.1 related)
SRCAP Snf2-related CREBBP activator protein
STIP1 stress-induced phosphoprotein 1
TES testin LIM domain protein
TMEM19 transmembrane protein 19
TNFSF9 tumor necrosis factor (ligand) superfamily, member 9
TNIK TRAF2 and NCK interacting kinase
TPMT thiopurine S-methyltransferase
TPP1 tripeptidyl peptidase I
TRIM2 tripartite motif containing 2
UCHL1 ubiquitin carboxyl-terminal esterase L1 (ubiquitin thiolesterase)
ULBP2 UL16 binding protein 2
WDR59 WD repeat domain 59
ZNF10 zinc finger protein 10
ZNF165 zinc finger protein 165
ZNF227 zinc finger protein 227
ZNF235 zinc finger protein 235
ZNF329 zinc finger protein 329
ZNF419 zinc finger protein 419

decreased expression

Symbol Name
ACKR3 atypical chemokine receptor 3
ACVR2B activin A receptor, type IIB
ADGRG2 adhesion G protein-coupled receptor G2
AHDC1 AT hook, DNA binding motif, containing 1
ANKRD36B ankyrin repeat domain 36B
ANKZF1 ankyrin repeat and zinc finger domain containing 1
ANP32A-IT1 ANP32A intronic transcript 1
AXIN1 axin 1
BAHCC1 BAH domain and coiled-coil containing 1
BIK BCL2-interacting killer (apoptosis-inducing)
C1ORF106 chromosome 1 open reading frame 106
C1QTNF3 C1q and tumor necrosis factor related protein 3
C5AR2 complement component 5a receptor 2
CCNT1 cyclin T1
CD82 CD82 molecule
CDADC1 cytidine and dCMP deaminase domain containing 1
CHAC1 ChaC glutathione-specific gamma-glutamylcyclotransferase 1
CLMN calmin (calponin-like, transmembrane)
CTNNBIP1 catenin, beta interacting protein 1
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
CYP26A1 cytochrome P450, family 26, subfamily A, polypeptide 1
DBNDD1 dysbindin (dystrobrevin binding protein 1) domain containing 1
DDX43 DEAD (Asp-Glu-Ala-Asp) box polypeptide 43
DNAAF2 dynein, axonemal, assembly factor 2
DUSP2 dual specificity phosphatase 2
EGR3 early growth response 3
EXD3 exonuclease 3'-5' domain containing 3
FAM102A family with sequence similarity 102, member A
FAM120C family with sequence similarity 120C
FAM155B family with sequence similarity 155, member B
GNAZ guanine nucleotide binding protein (G protein), alpha z polypeptide
GPR19 G protein-coupled receptor 19
HIVEP1 human immunodeficiency virus type I enhancer binding protein 1
HOXA4 homeobox A4
HOXC13 homeobox C13
HS1BP3 HCLS1 binding protein 3
ID1 inhibitor of DNA binding 1, dominant negative helix-loop-helix protein
IER2 immediate early response 2
IPO13 importin 13
ITGA10 integrin, alpha 10
JUNB jun B proto-oncogene
KIAA0125 KIAA0125
KLF10 Kruppel-like factor 10
KLF11 Kruppel-like factor 11
LIN7A lin-7 homolog A (C. elegans)
LOC390998 ribosomal protein L10 pseudogene
LRFN4 leucine rich repeat and fibronectin type III domain containing 4
LRRC49 leucine rich repeat containing 49
MAPKBP1 mitogen-activated protein kinase binding protein 1
MATK megakaryocyte-associated tyrosine kinase
MCOLN1 mucolipin 1
MID1IP1 MID1 interacting protein 1
MMP15 matrix metallopeptidase 15 (membrane-inserted)
MYC v-myc avian myelocytomatosis viral oncogene homolog
NCAM2 neural cell adhesion molecule 2
NFKBIA nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, alpha
ONECUT2 one cut homeobox 2
OR7E47P olfactory receptor, family 7, subfamily E, member 47 pseudogene
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
PCF11 PCF11 cleavage and polyadenylation factor subunit
PGBD5 piggyBac transposable element derived 5
PIK3R2 phosphoinositide-3-kinase, regulatory subunit 2 (beta)
PLXNA3 plexin A3
PMS1 PMS1 postmeiotic segregation increased 1 (S. cerevisiae)
PODXL2 podocalyxin-like 2
PPM1F protein phosphatase, Mg2+/Mn2+ dependent, 1F
PPRC1 peroxisome proliferator-activated receptor gamma, coactivator-related 1
PRKCD protein kinase C, delta
PTPRU protein tyrosine phosphatase, receptor type, U
RAB33B RAB33B, member RAS oncogene family
RAPGEFL1 Rap guanine nucleotide exchange factor (GEF)-like 1
RASSF8 Ras association (RalGDS/AF-6) domain family (N-terminal) member 8
RBM14 RNA binding motif protein 14
RFNG RFNG O-fucosylpeptide 3-beta-N-acetylglucosaminyltransferase
RGS16 regulator of G-protein signaling 16
RHPN1-AS1 RHPN1 antisense RNA 1 (head to head)
RNPEPL1 arginyl aminopeptidase (aminopeptidase B)-like 1
RPL23AP32 ribosomal protein L23a pseudogene 32
RPS6KA5 ribosomal protein S6 kinase, 90kDa, polypeptide 5
SCO2 SCO2 cytochrome c oxidase assembly protein
SEMA4C sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4C
SETD6 SET domain containing 6
SLC26A6 solute carrier family 26 (anion exchanger), member 6
SLC9A1 solute carrier family 9, subfamily A (NHE1, cation proton antiporter 1), member 1
SMAD7 SMAD family member 7
SNAPC2 small nuclear RNA activating complex, polypeptide 2, 45kDa
SNAPC4 small nuclear RNA activating complex, polypeptide 4, 190kDa
SPHK1 sphingosine kinase 1
ST3GAL1 ST3 beta-galactoside alpha-2,3-sialyltransferase 1
STX1A syntaxin 1A (brain)
SYTL2 synaptotagmin-like 2
TERF2 telomeric repeat binding factor 2
TICAM1 toll-like receptor adaptor molecule 1
TMEM120B transmembrane protein 120B
TRPV1 transient receptor potential cation channel, subfamily V, member 1
TWISTNB TWIST neighbor
WDR76 WD repeat domain 76
XRCC3 X-ray repair complementing defective repair in Chinese hamster cells 3
ZXDC ZXD family zinc finger C