tanespimycin-831 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

198 genes differentially expressed following the tanespimycin-831 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ADM adrenomedullin
ALOX15 arachidonate 15-lipoxygenase
ANXA1 annexin A1
ARG2 arginase 2
ARMCX1 armadillo repeat containing, X-linked 1
ATF7IP2 activating transcription factor 7 interacting protein 2
BMP2K BMP2 inducible kinase
C10ORF95 chromosome 10 open reading frame 95
CACYBP calcyclin binding protein
CCNG2 cyclin G2
CCP110 centriolar coiled coil protein 110kDa
CENPO centromere protein O
CHORDC1 cysteine and histidine-rich domain (CHORD) containing 1
CLCN6 chloride channel, voltage-sensitive 6
CLGN calmegin
CPN2 carboxypeptidase N, polypeptide 2
CRELD1 cysteine-rich with EGF-like domains 1
CREM cAMP responsive element modulator
CSRP2 cysteine and glycine-rich protein 2
CYLC1 cylicin, basic protein of sperm head cytoskeleton 1
DDIT3 DNA-damage-inducible transcript 3
DDIT4 DNA-damage-inducible transcript 4
DHRS2 dehydrogenase/reductase (SDR family) member 2
DNAJA1 DnaJ (Hsp40) homolog, subfamily A, member 1
DNAJB1 DnaJ (Hsp40) homolog, subfamily B, member 1
DNAJB4 DnaJ (Hsp40) homolog, subfamily B, member 4
DNAJB9 DnaJ (Hsp40) homolog, subfamily B, member 9
EDRF1 erythroid differentiation regulatory factor 1
EML2 echinoderm microtubule associated protein like 2
ENGASE endo-beta-N-acetylglucosaminidase
ETV5 ets variant 5
EXPH5 exophilin 5
FLT3LG fms-related tyrosine kinase 3 ligand
FNDC3A fibronectin type III domain containing 3A
GRM8 glutamate receptor, metabotropic 8
GTF3C3 general transcription factor IIIC, polypeptide 3, 102kDa
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HMOX1 heme oxygenase 1
HNRNPD heterogeneous nuclear ribonucleoprotein D (AU-rich element RNA binding protein 1, 37kDa)
HSD17B7 hydroxysteroid (17-beta) dehydrogenase 7
HSP90B1 heat shock protein 90kDa beta (Grp94), member 1
HSPA13 heat shock protein 70kDa family, member 13
HSPA1A heat shock 70kDa protein 1A
HSPA4L heat shock 70kDa protein 4-like
HSPA6 heat shock 70kDa protein 6 (HSP70B')
HSPH1 heat shock 105kDa/110kDa protein 1
INHBE inhibin, beta E
KDM6A lysine (K)-specific demethylase 6A
KLF9 Kruppel-like factor 9
LZTFL1 leucine zipper transcription factor-like 1
MANF mesencephalic astrocyte-derived neurotrophic factor
MAP1B microtubule-associated protein 1B
MBNL2 muscleblind-like splicing regulator 2
MFAP3L microfibrillar-associated protein 3-like
MLLT11 myeloid/lymphoid or mixed-lineage leukemia (trithorax homolog, Drosophila); translocated to, 11
MORC4 MORC family CW-type zinc finger 4
N4BP2L2 NEDD4 binding protein 2-like 2
NCR2 natural cytotoxicity triggering receptor 2
NEAT1 nuclear paraspeckle assembly transcript 1 (non-protein coding)
NKX3-2 NK3 homeobox 2
NLGN1 neuroligin 1
NUPR1 nuclear protein, transcriptional regulator, 1
ORC5 origin recognition complex, subunit 5
OSBPL1A oxysterol binding protein-like 1A
OSGIN1 oxidative stress induced growth inhibitor 1
P4HA2 prolyl 4-hydroxylase, alpha polypeptide II
PADI3 peptidyl arginine deiminase, type III
PCM1 pericentriolar material 1
PGF placental growth factor
PLA2G3 phospholipase A2, group III
POFUT1 protein O-fucosyltransferase 1
PPID peptidylprolyl isomerase D
PPM1A protein phosphatase, Mg2+/Mn2+ dependent, 1A
PPM1E protein phosphatase, Mg2+/Mn2+ dependent, 1E
PRSS16 protease, serine, 16 (thymus)
RFTN1 raftlin, lipid raft linker 1
RGS2 regulator of G-protein signaling 2
RPS3A ribosomal protein S3A
SDF2L1 stromal cell-derived factor 2-like 1
SEL1L sel-1 suppressor of lin-12-like (C. elegans)
SENP6 SUMO1/sentrin specific peptidase 6
SERPINH1 serpin peptidase inhibitor, clade H (heat shock protein 47), member 1, (collagen binding protein 1)
SH3BGR SH3 domain binding glutamate-rich protein
SLC1A4 solute carrier family 1 (glutamate/neutral amino acid transporter), member 4
SLC43A1 solute carrier family 43 (amino acid system L transporter), member 1
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
ST3GAL5 ST3 beta-galactoside alpha-2,3-sialyltransferase 5
TES testin LIM domain protein
TSPYL2 TSPY-like 2
UFL1 UFM1-specific ligase 1
VAMP4 vesicle-associated membrane protein 4
VLDLR very low density lipoprotein receptor
ZMYND8 zinc finger, MYND-type containing 8
ZNF165 zinc finger protein 165
ZNF227 zinc finger protein 227
ZNF268 zinc finger protein 268
ZNF350 zinc finger protein 350
ZNF419 zinc finger protein 419

decreased expression

Symbol Name
ACKR3 atypical chemokine receptor 3
AGPAT3 1-acylglycerol-3-phosphate O-acyltransferase 3
ALKBH4 alkB, alkylation repair homolog 4 (E. coli)
ANKRD36B ankyrin repeat domain 36B
APEX2 APEX nuclease (apurinic/apyrimidinic endonuclease) 2
ASF1B anti-silencing function 1B histone chaperone
ASTE1 asteroid homolog 1 (Drosophila)
BAHCC1 BAH domain and coiled-coil containing 1
BIK BCL2-interacting killer (apoptosis-inducing)
C10ORF88 chromosome 10 open reading frame 88
C2CD2 C2 calcium-dependent domain containing 2
C3ORF52 chromosome 3 open reading frame 52
C9ORF3 chromosome 9 open reading frame 3
CCNE1 cyclin E1
CDK8 cyclin-dependent kinase 8
CEBPA CCAAT/enhancer binding protein (C/EBP), alpha
CEP131 centrosomal protein 131kDa
CISH cytokine inducible SH2-containing protein
CLN6 ceroid-lipofuscinosis, neuronal 6, late infantile, variant
CNKSR1 connector enhancer of kinase suppressor of Ras 1
CORO2A coronin, actin binding protein, 2A
CRCP CGRP receptor component
CYP1A1 cytochrome P450, family 1, subfamily A, polypeptide 1
CYP20A1 cytochrome P450, family 20, subfamily A, polypeptide 1
CYP26A1 cytochrome P450, family 26, subfamily A, polypeptide 1
E2F8 E2F transcription factor 8
EPPK1 epiplakin 1
ERMAP erythroblast membrane-associated protein (Scianna blood group)
FA2H fatty acid 2-hydroxylase
FAM179B family with sequence similarity 179, member B
FAN1 FANCD2/FANCI-associated nuclease 1
FOXC1 forkhead box C1
GLTSCR1 glioma tumor suppressor candidate region gene 1
GPR19 G protein-coupled receptor 19
GRWD1 glutamate-rich WD repeat containing 1
H2AFY2 H2A histone family, member Y2
HILPDA hypoxia inducible lipid droplet-associated
HOXC10 homeobox C10
HTR1E 5-hydroxytryptamine (serotonin) receptor 1E, G protein-coupled
ID1 inhibitor of DNA binding 1, dominant negative helix-loop-helix protein
IER2 immediate early response 2
IRX5 iroquois homeobox 5
KCNMB4 potassium channel subfamily M regulatory beta subunit 4
KIF3A kinesin family member 3A
KLF10 Kruppel-like factor 10
KPTN kaptin (actin binding protein)
MANSC1 MANSC domain containing 1
METTL4 methyltransferase like 4
MKNK1 MAP kinase interacting serine/threonine kinase 1
MTA2 metastasis associated 1 family, member 2
MTCL1 microtubule crosslinking factor 1
MUL1 mitochondrial E3 ubiquitin protein ligase 1
NABP2 nucleic acid binding protein 2
NFKBIA nuclear factor of kappa light polypeptide gene enhancer in B-cells inhibitor, alpha
OSGEPL1 O-sialoglycoprotein endopeptidase-like 1
P2RY2 purinergic receptor P2Y, G-protein coupled, 2
PARD6A par-6 family cell polarity regulator alpha
PARP16 poly (ADP-ribose) polymerase family, member 16
PCF11 PCF11 cleavage and polyadenylation factor subunit
PKIA protein kinase (cAMP-dependent, catalytic) inhibitor alpha
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
POLE2 polymerase (DNA directed), epsilon 2, accessory subunit
PPP1R10 protein phosphatase 1, regulatory subunit 10
PRICKLE3 prickle homolog 3 (Drosophila)
PRR7 proline rich 7 (synaptic)
PTCD2 pentatricopeptide repeat domain 2
RBM4B RNA binding motif protein 4B
RGS16 regulator of G-protein signaling 16
RIC8B RIC8 guanine nucleotide exchange factor B
RNF123 ring finger protein 123
RNF170 ring finger protein 170
RPGR retinitis pigmentosa GTPase regulator
SCO2 SCO2 cytochrome c oxidase assembly protein
SH2B2 SH2B adaptor protein 2
SKA1 spindle and kinetochore associated complex subunit 1
SLCO4A1 solute carrier organic anion transporter family, member 4A1
SMAD7 SMAD family member 7
SNX16 sorting nexin 16
SOBP sine oculis binding protein homolog (Drosophila)
SOX12 SRY (sex determining region Y)-box 12
SPATA2L spermatogenesis associated 2-like
STBD1 starch binding domain 1
SYNJ2BP synaptojanin 2 binding protein
TERF2 telomeric repeat binding factor 2
TFAP4 transcription factor AP-4 (activating enhancer binding protein 4)
TMEM11 transmembrane protein 11
TMEM159 transmembrane protein 159
TRIM52 tripartite motif containing 52
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TSEN2 TSEN2 tRNA splicing endonuclease subunit
TSKU tsukushi, small leucine rich proteoglycan
TUBA3C tubulin, alpha 3c
VWA1 von Willebrand factor A domain containing 1
WDR4 WD repeat domain 4
WEE1 WEE1 G2 checkpoint kinase
ZBTB24 zinc finger and BTB domain containing 24
ZMYM3 zinc finger, MYM-type 3
ZNF767P zinc finger family member 767, pseudogene
ZNF813 zinc finger protein 813
ZXDC ZXD family zinc finger C