telenzepine-7419 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

195 genes differentially expressed following the telenzepine-7419 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACTR5 ARP5 actin-related protein 5 homolog (yeast)
ADPRM ADP-ribose/CDP-alcohol diphosphatase, manganese-dependent
AKAP17A A kinase (PRKA) anchor protein 17A
AKAP7 A kinase (PRKA) anchor protein 7
AKT2 v-akt murine thymoma viral oncogene homolog 2
ALDH4A1 aldehyde dehydrogenase 4 family, member A1
ANGPTL2 angiopoietin-like 2
ANKZF1 ankyrin repeat and zinc finger domain containing 1
ANTXR1 anthrax toxin receptor 1
APBB2 amyloid beta (A4) precursor protein-binding, family B, member 2
APOM apolipoprotein M
AR androgen receptor
ARHGAP26 Rho GTPase activating protein 26
B4GALT4 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 4
BAZ2A bromodomain adjacent to zinc finger domain, 2A
CAPN10 calpain 10
CD1A CD1a molecule
CHST7 carbohydrate (N-acetylglucosamine 6-O) sulfotransferase 7
COQ7 coenzyme Q7 homolog, ubiquinone (yeast)
CTNND2 catenin (cadherin-associated protein), delta 2
CXXC4 CXXC finger protein 4
DHX57 DEAH (Asp-Glu-Ala-Asp/His) box polypeptide 57
DIO2 deiodinase, iodothyronine, type II
DNAJB2 DnaJ (Hsp40) homolog, subfamily B, member 2
DRP2 dystrophin related protein 2
DSC2 desmocollin 2
DST dystonin
EEF2KMT eukaryotic elongation factor 2 lysine methyltransferase
ENTPD4 ectonucleoside triphosphate diphosphohydrolase 4
EVA1B eva-1 homolog B (C. elegans)
EXD3 exonuclease 3'-5' domain containing 3
FAAH fatty acid amide hydrolase
FADS3 fatty acid desaturase 3
FBXL2 F-box and leucine-rich repeat protein 2
GIT2 G protein-coupled receptor kinase interacting ArfGAP 2
GLG1 golgi glycoprotein 1
HERC4 HECT and RLD domain containing E3 ubiquitin protein ligase 4
HFE hemochromatosis
HIST1H2BJ histone cluster 1, H2bj
HMOX1 heme oxygenase 1
HP1BP3 heterochromatin protein 1, binding protein 3
HSF1 heat shock transcription factor 1
IFT140 intraflagellar transport 140
IL15RA interleukin 15 receptor, alpha
INTS1 integrator complex subunit 1
ITGA6 integrin, alpha 6
KAZN kazrin, periplakin interacting protein
LONP2 lon peptidase 2, peroxisomal
MAP2K7 mitogen-activated protein kinase kinase 7
MAP3K1 mitogen-activated protein kinase kinase kinase 1, E3 ubiquitin protein ligase
MBD1 methyl-CpG binding domain protein 1
MBOAT7 membrane bound O-acyltransferase domain containing 7
MVB12B multivesicular body subunit 12B
MYBPC3 myosin binding protein C, cardiac
NCAPH2 non-SMC condensin II complex, subunit H2
NDE1 nudE neurodevelopment protein 1
NF2 neurofibromin 2 (merlin)
PIK3IP1 phosphoinositide-3-kinase interacting protein 1
PLAGL1 pleiomorphic adenoma gene-like 1
PLEKHG3 pleckstrin homology domain containing, family G (with RhoGef domain) member 3
PLK4 polo-like kinase 4
POLL polymerase (DNA directed), lambda
PPAP2B phosphatidic acid phosphatase type 2B
PPP2R3A protein phosphatase 2, regulatory subunit B'', alpha
PTPRS protein tyrosine phosphatase, receptor type, S
QKI QKI, KH domain containing, RNA binding
RAD51B RAD51 paralog B
RIN2 Ras and Rab interactor 2
RUFY3 RUN and FYVE domain containing 3
SEMA3F sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3F
SEMA4D sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4D
SFXN3 sideroflexin 3
SGSM3 small G protein signaling modulator 3
SIRT3 sirtuin 3
SKP2 S-phase kinase-associated protein 2, E3 ubiquitin protein ligase
SLC16A3 solute carrier family 16 (monocarboxylate transporter), member 3
SLC24A3 solute carrier family 24 (sodium/potassium/calcium exchanger), member 3
SLC7A1 solute carrier family 7 (cationic amino acid transporter, y+ system), member 1
SLC9A3R2 solute carrier family 9, subfamily A (NHE3, cation proton antiporter 3), member 3 regulator 2
SNCA synuclein, alpha (non A4 component of amyloid precursor)
SP1 Sp1 transcription factor
SRD5A3 steroid 5 alpha-reductase 3
STS steroid sulfatase (microsomal), isozyme S
SYMPK symplekin
SYNGR1 synaptogyrin 1
TAGLN transgelin
TCF7L2 transcription factor 7-like 2 (T-cell specific, HMG-box)
TEP1 telomerase-associated protein 1
THBD thrombomodulin
TMEFF1 transmembrane protein with EGF-like and two follistatin-like domains 1
TUBGCP3 tubulin, gamma complex associated protein 3
USP34 ubiquitin specific peptidase 34
WDR19 WD repeat domain 19
WDR48 WD repeat domain 48
YTHDC2 YTH domain containing 2
ZNF276 zinc finger protein 276
ZNF701 zinc finger protein 701

decreased expression

Symbol Name
ABLIM3 actin binding LIM protein family, member 3
ATG9A autophagy related 9A
B4GALT2 UDP-Gal:betaGlcNAc beta 1,4- galactosyltransferase, polypeptide 2
BCL9 B-cell CLL/lymphoma 9
BRPF1 bromodomain and PHD finger containing, 1
C16ORF59 chromosome 16 open reading frame 59
CALCOCO1 calcium binding and coiled-coil domain 1
CENPT centromere protein T
CHST11 carbohydrate (chondroitin 4) sulfotransferase 11
CLSPN claspin
CRYL1 crystallin, lambda 1
DAP death-associated protein
DCAF13 DDB1 and CUL4 associated factor 13
DHDDS dehydrodolichyl diphosphate synthase
DNM1 dynamin 1
ETHE1 ethylmalonic encephalopathy 1
EVPL envoplakin
FAM160B2 family with sequence similarity 160, member B2
FAM193B family with sequence similarity 193, member B
FAM63A family with sequence similarity 63, member A
FBRS fibrosin
FBXO31 F-box protein 31
FBXW7 F-box and WD repeat domain containing 7, E3 ubiquitin protein ligase
FGD6 FYVE, RhoGEF and PH domain containing 6
FHOD1 formin homology 2 domain containing 1
FOXRED2 FAD-dependent oxidoreductase domain containing 2
FURIN furin (paired basic amino acid cleaving enzyme)
FUT1 fucosyltransferase 1 (galactoside 2-alpha-L-fucosyltransferase, H blood group)
FUZ fuzzy planar cell polarity protein
GLB1L2 galactosidase, beta 1-like 2
GLI3 GLI family zinc finger 3
GPHN gephyrin
HIRIP3 HIRA interacting protein 3
HIST1H2AJ histone cluster 1, H2aj
HIST1H4D histone cluster 1, H4d
HIST1H4J histone cluster 1, H4j
IER3IP1 immediate early response 3 interacting protein 1
INF2 inverted formin, FH2 and WH2 domain containing
IRX4 iroquois homeobox 4
LINC00115 long intergenic non-protein coding RNA 115
LRFN3 leucine rich repeat and fibronectin type III domain containing 3
MBNL3 muscleblind-like splicing regulator 3
MECR mitochondrial trans-2-enoyl-CoA reductase
MFSD11 major facilitator superfamily domain containing 11
MICALL2 MICAL-like 2
MITF microphthalmia-associated transcription factor
MXD3 MAX dimerization protein 3
NARFL nuclear prelamin A recognition factor-like
NINL ninein-like
NPIPB15 nuclear pore complex interacting protein family, member B15
NSMF NMDA receptor synaptonuclear signaling and neuronal migration factor
OGFRL1 opioid growth factor receptor-like 1
PCDHB3 protocadherin beta 3
PEX26 peroxisomal biogenesis factor 26
PGP phosphoglycolate phosphatase
PIGH phosphatidylinositol glycan anchor biosynthesis, class H
PIGL phosphatidylinositol glycan anchor biosynthesis, class L
PLD2 phospholipase D2
PLD3 phospholipase D family, member 3
PLXNA3 plexin A3
POP1 processing of precursor 1, ribonuclease P/MRP subunit (S. cerevisiae)
PRMT7 protein arginine methyltransferase 7
PTCD2 pentatricopeptide repeat domain 2
PYCRL pyrroline-5-carboxylate reductase-like
QTRT1 queuine tRNA-ribosyltransferase 1
RAB8B RAB8B, member RAS oncogene family
RAC3 ras-related C3 botulinum toxin substrate 3 (rho family, small GTP binding protein Rac3)
RAPGEFL1 Rap guanine nucleotide exchange factor (GEF)-like 1
RNF126P1 ring finger protein 126 pseudogene 1
RPAP1 RNA polymerase II associated protein 1
RRAS related RAS viral (r-ras) oncogene homolog
RRNAD1 ribosomal RNA adenine dimethylase domain containing 1
SETD1A SET domain containing 1A
SLC12A7 solute carrier family 12 (potassium/chloride transporter), member 7
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SMPD2 sphingomyelin phosphodiesterase 2, neutral membrane (neutral sphingomyelinase)
SPSB1 splA/ryanodine receptor domain and SOCS box containing 1
SREK1IP1 SREK1-interacting protein 1
STXBP1 syntaxin binding protein 1
TFAP4 transcription factor AP-4 (activating enhancer binding protein 4)
TMEM134 transmembrane protein 134
TMEM160 transmembrane protein 160
TMEM53 transmembrane protein 53
TRIP10 thyroid hormone receptor interactor 10
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TSPAN5 tetraspanin 5
TUBA3C tubulin, alpha 3c
VGF VGF nerve growth factor inducible
VWA1 von Willebrand factor A domain containing 1
WARS2 tryptophanyl tRNA synthetase 2, mitochondrial
XPC xeroderma pigmentosum, complementation group C
ZBED1 zinc finger, BED-type containing 1
ZBTB25 zinc finger and BTB domain containing 25
ZNF180 zinc finger protein 180
ZNF205 zinc finger protein 205
ZNF212 zinc finger protein 212
ZNF586 zinc finger protein 586
ZNF767P zinc finger family member 767, pseudogene