tioguanine-642 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the tioguanine-642 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ABHD5 abhydrolase domain containing 5
ACACA acetyl-CoA carboxylase alpha
ACOT8 acyl-CoA thioesterase 8
ADM2 adrenomedullin 2
AKR1C1 aldo-keto reductase family 1, member C1
AQP6 aquaporin 6, kidney specific
ARNTL aryl hydrocarbon receptor nuclear translocator-like
ARVCF armadillo repeat gene deleted in velocardiofacial syndrome
ATP8B2 ATPase, aminophospholipid transporter, class I, type 8B, member 2
BAIAP2 BAI1-associated protein 2
BAZ2A bromodomain adjacent to zinc finger domain, 2A
BICD1 bicaudal D homolog 1 (Drosophila)
BMP6 bone morphogenetic protein 6
C19ORF40 chromosome 19 open reading frame 40
C1QTNF9B-AS1 C1QTNF9B antisense RNA 1
C4BPA complement component 4 binding protein, alpha
C5ORF30 chromosome 5 open reading frame 30
CACNB1 calcium channel, voltage-dependent, beta 1 subunit
CAMKV CaM kinase-like vesicle-associated
CCDC71 coiled-coil domain containing 71
CCDC93 coiled-coil domain containing 93
CDK10 cyclin-dependent kinase 10
CDYL chromodomain protein, Y-like
CHRM4 cholinergic receptor, muscarinic 4
CIDEB cell death-inducing DFFA-like effector b
COX4I1 cytochrome c oxidase subunit IV isoform 1
CRYBB2P1 crystallin, beta B2 pseudogene 1
DNAJC16 DnaJ (Hsp40) homolog, subfamily C, member 16
DRP2 dystrophin related protein 2
DSCAM Down syndrome cell adhesion molecule
DTNA dystrobrevin, alpha
EFNB3 ephrin-B3
FARP1 FERM, RhoGEF (ARHGEF) and pleckstrin domain protein 1 (chondrocyte-derived)
FBLN1 fibulin 1
GABBR1 gamma-aminobutyric acid (GABA) B receptor, 1
GINS3 GINS complex subunit 3 (Psf3 homolog)
GP2 glycoprotein 2 (zymogen granule membrane)
GRIP2 glutamate receptor interacting protein 2
HERPUD1 homocysteine-inducible, endoplasmic reticulum stress-inducible, ubiquitin-like domain member 1
HINFP histone H4 transcription factor
HOXD9 homeobox D9
HPCAL4 hippocalcin like 4
IRF4 interferon regulatory factor 4
ISCA1 iron-sulfur cluster assembly 1
ITGA3 integrin, alpha 3 (antigen CD49C, alpha 3 subunit of VLA-3 receptor)
KCNMB3 potassium channel subfamily M regulatory beta subunit 3
KIF25 kinesin family member 25
KLHL28 kelch-like family member 28
KLHL35 kelch-like family member 35
LLGL1 lethal giant larvae homolog 1 (Drosophila)
LMF2 lipase maturation factor 2
LYZL6 lysozyme-like 6
MBD1 methyl-CpG binding domain protein 1
MED28 mediator complex subunit 28
MMP17 matrix metallopeptidase 17 (membrane-inserted)
MTMR8 myotubularin related protein 8
NDST2 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 2
NF2 neurofibromin 2 (merlin)
NPEPPS aminopeptidase puromycin sensitive
NREP neuronal regeneration related protein
NRSN2 neurensin 2
OLFM1 olfactomedin 1
PDK2 pyruvate dehydrogenase kinase, isozyme 2
PECR peroxisomal trans-2-enoyl-CoA reductase
PHC1 polyhomeotic homolog 1 (Drosophila)
PIK3C3 phosphatidylinositol 3-kinase, catalytic subunit type 3
PITX1 paired-like homeodomain 1
PPIL2 peptidylprolyl isomerase (cyclophilin)-like 2
PRKRIP1 PRKR interacting protein 1 (IL11 inducible)
PRSS3 protease, serine, 3
PTCRA pre T-cell antigen receptor alpha
PTDSS2 phosphatidylserine synthase 2
RAB32 RAB32, member RAS oncogene family
RND2 Rho family GTPase 2
RUNX1 runt-related transcription factor 1
SEC63 SEC63 homolog (S. cerevisiae)
SEMA3B sema domain, immunoglobulin domain (Ig), short basic domain, secreted, (semaphorin) 3B
SFI1 Sfi1 homolog, spindle assembly associated (yeast)
SFXN3 sideroflexin 3
SGCD sarcoglycan, delta (35kDa dystrophin-associated glycoprotein)
SLC6A3 solute carrier family 6 (neurotransmitter transporter), member 3
SLC7A11 solute carrier family 7 (anionic amino acid transporter light chain, xc- system), member 11
SMO smoothened, frizzled class receptor
SORBS3 sorbin and SH3 domain containing 3
SPTBN5 spectrin, beta, non-erythrocytic 5
SSTR4 somatostatin receptor 4
SUN2 Sad1 and UNC84 domain containing 2
TBL1X transducin (beta)-like 1X-linked
TMEM127 transmembrane protein 127
TMF1 TATA element modulatory factor 1
TNFRSF21 tumor necrosis factor receptor superfamily, member 21
TRIL TLR4 interactor with leucine-rich repeats
TTLL4 tubulin tyrosine ligase-like family member 4
VIPR1 vasoactive intestinal peptide receptor 1
YY1 YY1 transcription factor
ZER1 zyg-11 related, cell cycle regulator
ZFP36L2 ZFP36 ring finger protein-like 2
ZFR zinc finger RNA binding protein

decreased expression

Symbol Name
ABHD3 abhydrolase domain containing 3
AGRP agouti related neuropeptide
ARHGAP5 Rho GTPase activating protein 5
ASTE1 asteroid homolog 1 (Drosophila)
ATG10 autophagy related 10
ATXN8OS ATXN8 opposite strand (non-protein coding)
B4GALNT1 beta-1,4-N-acetyl-galactosaminyl transferase 1
BPIFA1 BPI fold containing family A, member 1
C17ORF80 chromosome 17 open reading frame 80
C1ORF95 chromosome 1 open reading frame 95
CA11 carbonic anhydrase XI
CBLL1 Cbl proto-oncogene-like 1, E3 ubiquitin protein ligase
CCDC170 coiled-coil domain containing 170
CCDC64 coiled-coil domain containing 64
CD79A CD79a molecule, immunoglobulin-associated alpha
CHCHD7 coiled-coil-helix-coiled-coil-helix domain containing 7
CHRNA2 cholinergic receptor, nicotinic, alpha 2 (neuronal)
CHUK conserved helix-loop-helix ubiquitous kinase
COA7 cytochrome c oxidase assembly factor 7 (putative)
COMMD8 COMM domain containing 8
CPOX coproporphyrinogen oxidase
CPSF7 cleavage and polyadenylation specific factor 7, 59kDa
CST8 cystatin 8 (cystatin-related epididymal specific)
CYB5R3 cytochrome b5 reductase 3
DSN1 DSN1, MIS12 kinetochore complex component
ECE2 endothelin converting enzyme 2
EGLN1 egl-9 family hypoxia-inducible factor 1
EHD3 EH-domain containing 3
EPB41L5 erythrocyte membrane protein band 4.1 like 5
ERCC4 excision repair cross-complementation group 4
ESPN espin
FAM171A1 family with sequence similarity 171, member A1
FAM188A family with sequence similarity 188, member A
FPGT fucose-1-phosphate guanylyltransferase
GAN gigaxonin
GFOD1 glucose-fructose oxidoreductase domain containing 1
GMEB1 glucocorticoid modulatory element binding protein 1
GNAI2 guanine nucleotide binding protein (G protein), alpha inhibiting activity polypeptide 2
GPX2 glutathione peroxidase 2
HERC2 HECT and RLD domain containing E3 ubiquitin protein ligase 2
IGFALS insulin-like growth factor binding protein, acid labile subunit
JRKL JRK-like
KCTD3 potassium channel tetramerization domain containing 3
KRT32 keratin 32, type I
LECT1 leukocyte cell derived chemotaxin 1
LGALS4 lectin, galactoside-binding, soluble, 4
LTN1 listerin E3 ubiquitin protein ligase 1
MAFG v-maf avian musculoaponeurotic fibrosarcoma oncogene homolog G
MAPK3 mitogen-activated protein kinase 3
MATK megakaryocyte-associated tyrosine kinase
MIR22HG MIR22 host gene
MUL1 mitochondrial E3 ubiquitin protein ligase 1
MYL1 myosin, light chain 1, alkali; skeletal, fast
MYL12B myosin, light chain 12B, regulatory
NAE1 NEDD8 activating enzyme E1 subunit 1
NELL2 NEL-like 2 (chicken)
NOP14 NOP14 nucleolar protein
NPTX1 neuronal pentraxin I
PARG poly (ADP-ribose) glycohydrolase
PCDHB3 protocadherin beta 3
PCP4 Purkinje cell protein 4
PCTP phosphatidylcholine transfer protein
PIEZO2 piezo-type mechanosensitive ion channel component 2
PIM2 Pim-2 proto-oncogene, serine/threonine kinase
PISD phosphatidylserine decarboxylase
PLA2G10 phospholipase A2, group X
PLD2 phospholipase D2
PLEKHA1 pleckstrin homology domain containing, family A (phosphoinositide binding specific) member 1
PLEKHO1 pleckstrin homology domain containing, family O member 1
PLXNB3 plexin B3
PUS7L pseudouridylate synthase 7 homolog (S. cerevisiae)-like
PWP2 PWP2 periodic tryptophan protein homolog (yeast)
RALBP1 ralA binding protein 1
RAPGEFL1 Rap guanine nucleotide exchange factor (GEF)-like 1
RBMS3 RNA binding motif, single stranded interacting protein 3
RGSL1 regulator of G-protein signaling like 1
RHOH ras homolog family member H
RPS4Y1 ribosomal protein S4, Y-linked 1
S1PR4 sphingosine-1-phosphate receptor 4
SCML1 sex comb on midleg-like 1 (Drosophila)
SEMA4A sema domain, immunoglobulin domain (Ig), transmembrane domain (TM) and short cytoplasmic domain, (semaphorin) 4A
SKAP1 src kinase associated phosphoprotein 1
SLC16A2 solute carrier family 16, member 2 (thyroid hormone transporter)
SLC17A7 solute carrier family 17 (vesicular glutamate transporter), member 7
SLC6A4 solute carrier family 6 (neurotransmitter transporter), member 4
SMARCD3 SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily d, member 3
SRPK3 SRSF protein kinase 3
SURF2 surfeit 2
TCEA2 transcription elongation factor A (SII), 2
TIMM10 translocase of inner mitochondrial membrane 10 homolog (yeast)
TOP2B topoisomerase (DNA) II beta 180kDa
TRIM52 tripartite motif containing 52
TRIM8 tripartite motif containing 8
TSEN2 TSEN2 tRNA splicing endonuclease subunit
UNC93B1 unc-93 homolog B1 (C. elegans)
VASP vasodilator-stimulated phosphoprotein
XPA xeroderma pigmentosum, complementation group A
ZNF280A zinc finger protein 280A
ZNF557 zinc finger protein 557