velnacrine-4997 Gene Set

Dataset CMAP Signatures of Differentially Expressed Genes for Small Molecules
Category transcriptomics
Type small molecule perturbation
Description small molecule perturbation identified as [small molecule name]-[perturbation ID] (ChIP-X Enrichment Analysis)
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Genes

197 genes differentially expressed following the velnacrine-4997 small molecule perturbation from the CMAP Signatures of Differentially Expressed Genes for Small Molecules dataset.

increased expression

Symbol Name
ACBD4 acyl-CoA binding domain containing 4
ACVR1B activin A receptor, type IB
ADAP2 ArfGAP with dual PH domains 2
ANKRD2 ankyrin repeat domain 2 (stretch responsive muscle)
ASPH aspartate beta-hydroxylase
BAIAP3 BAI1-associated protein 3
BAX BCL2-associated X protein
C11ORF30 chromosome 11 open reading frame 30
CANX calnexin
CAPN9 calpain 9
CASP1 caspase 1, apoptosis-related cysteine peptidase
CASP10 caspase 10, apoptosis-related cysteine peptidase
CFAP70 cilia and flagella associated protein 70
CLEC3B C-type lectin domain family 3, member B
CLTC clathrin, heavy chain (Hc)
COL16A1 collagen, type XVI, alpha 1
COL19A1 collagen, type XIX, alpha 1
CUL7 cullin 7
CYP4F8 cytochrome P450, family 4, subfamily F, polypeptide 8
DICER1 dicer 1, ribonuclease type III
DLX2 distal-less homeobox 2
DST dystonin
DUSP13 dual specificity phosphatase 13
EML2 echinoderm microtubule associated protein like 2
F2RL2 coagulation factor II (thrombin) receptor-like 2
FLJ11292
GM2A GM2 ganglioside activator
GRM4 glutamate receptor, metabotropic 4
HERC3 HECT and RLD domain containing E3 ubiquitin protein ligase 3
HIPK3 homeodomain interacting protein kinase 3
HIRA histone cell cycle regulator
HIST1H4F histone cluster 1, H4f
HLA-DPA1 major histocompatibility complex, class II, DP alpha 1
ICA1 islet cell autoantigen 1, 69kDa
IFT27 intraflagellar transport 27
IL2 interleukin 2
ING1 inhibitor of growth family, member 1
ITIH2 inter-alpha-trypsin inhibitor heavy chain 2
KANSL1L KAT8 regulatory NSL complex subunit 1-like
KLHL22 kelch-like family member 22
KLK1 kallikrein 1
LAIR1 leukocyte-associated immunoglobulin-like receptor 1
LIFR leukemia inhibitory factor receptor alpha
LOC284244 uncharacterized LOC284244
LRRFIP1 leucine rich repeat (in FLII) interacting protein 1
LTBP4 latent transforming growth factor beta binding protein 4
MAPK8IP2 mitogen-activated protein kinase 8 interacting protein 2
MAST3 microtubule associated serine/threonine kinase 3
MGEA5 meningioma expressed antigen 5 (hyaluronidase)
MON2 MON2 homolog (S. cerevisiae)
MRPL41 mitochondrial ribosomal protein L41
MTHFR methylenetetrahydrofolate reductase (NAD(P)H)
NCKAP1 NCK-associated protein 1
NDST1 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 1
NEAT1 nuclear paraspeckle assembly transcript 1 (non-protein coding)
NF1 neurofibromin 1
OCLM oculomedin
PCDH9 protocadherin 9
PCK1 phosphoenolpyruvate carboxykinase 1 (soluble)
PDCD2 programmed cell death 2
PDE6B phosphodiesterase 6B, cGMP-specific, rod, beta
PEX16 peroxisomal biogenesis factor 16
PHF7 PHD finger protein 7
PIP5K1A phosphatidylinositol-4-phosphate 5-kinase, type I, alpha
POU2F3 POU class 2 homeobox 3
PPP3R1 protein phosphatase 3, regulatory subunit B, alpha
PRKAR1B protein kinase, cAMP-dependent, regulatory, type I, beta
PRSS53 protease, serine, 53
PSG4 pregnancy specific beta-1-glycoprotein 4
PTPN21 protein tyrosine phosphatase, non-receptor type 21
RAD23B RAD23 homolog B (S. cerevisiae)
RBBP9 retinoblastoma binding protein 9
RIF1 replication timing regulatory factor 1
RNF126P1 ring finger protein 126 pseudogene 1
RSPH14 radial spoke head 14 homolog (Chlamydomonas)
SEC23A Sec23 homolog A (S. cerevisiae)
SERGEF secretion regulating guanine nucleotide exchange factor
SH3TC1 SH3 domain and tetratricopeptide repeats 1
SLA Src-like-adaptor
SLC25A37 solute carrier family 25 (mitochondrial iron transporter), member 37
SLC7A1 solute carrier family 7 (cationic amino acid transporter, y+ system), member 1
SMG7 SMG7 nonsense mediated mRNA decay factor
SPINK4 serine peptidase inhibitor, Kazal type 4
SRRM2 serine/arginine repetitive matrix 2
STC1 stanniocalcin 1
TBC1D5 TBC1 domain family, member 5
TBKBP1 TBK1 binding protein 1
TGM2 transglutaminase 2
TIMP3 TIMP metallopeptidase inhibitor 3
TLDC1 TBC/LysM-associated domain containing 1
TMPRSS2 transmembrane protease, serine 2
TUBA3C tubulin, alpha 3c
UCHL1 ubiquitin carboxyl-terminal esterase L1 (ubiquitin thiolesterase)
UTP18 UTP18 small subunit (SSU) processome component homolog (yeast)
VPS13B vacuolar protein sorting 13 homolog B (yeast)
WNT16 wingless-type MMTV integration site family, member 16
YTHDC2 YTH domain containing 2
ZBTB33 zinc finger and BTB domain containing 33
ZFP36L1 ZFP36 ring finger protein-like 1

decreased expression

Symbol Name
ADAM15 ADAM metallopeptidase domain 15
ADCK3 aarF domain containing kinase 3
ADM adrenomedullin
AES amino-terminal enhancer of split
AKIP1 A kinase (PRKA) interacting protein 1
ANKRD28 ankyrin repeat domain 28
BAGE B melanoma antigen
BCORL1 BCL6 corepressor-like 1
BTBD7 BTB (POZ) domain containing 7
C14ORF132 chromosome 14 open reading frame 132
C14ORF93 chromosome 14 open reading frame 93
C16ORF59 chromosome 16 open reading frame 59
C1ORF35 chromosome 1 open reading frame 35
CA5BP1 carbonic anhydrase VB pseudogene 1
CDC42SE1 CDC42 small effector 1
CHMP6 charged multivesicular body protein 6
CHRM3 cholinergic receptor, muscarinic 3
CIDEC cell death-inducing DFFA-like effector c
CLK3 CDC-like kinase 3
CNPY3 canopy FGF signaling regulator 3
CYP2R1 cytochrome P450, family 2, subfamily R, polypeptide 1
DCAF13 DDB1 and CUL4 associated factor 13
DLEU2 deleted in lymphocytic leukemia 2 (non-protein coding)
DNM1 dynamin 1
DOCK4 dedicator of cytokinesis 4
EFNA3 ephrin-A3
FAM155B family with sequence similarity 155, member B
FBXO22 F-box protein 22
FER fer (fps/fes related) tyrosine kinase
FSTL3 follistatin-like 3 (secreted glycoprotein)
GDI1 GDP dissociation inhibitor 1
GMPPA GDP-mannose pyrophosphorylase A
GPRC5C G protein-coupled receptor, class C, group 5, member C
GPX2 glutathione peroxidase 2
GRB2 growth factor receptor-bound protein 2
HS1BP3 HCLS1 binding protein 3
IDI2-AS1 IDI2 antisense RNA 1
INO80D INO80 complex subunit D
ITFG2 integrin alpha FG-GAP repeat containing 2
JMJD4 jumonji domain containing 4
KDM5C lysine (K)-specific demethylase 5C
KLC2 kinesin light chain 2
KLHDC4 kelch domain containing 4
KREMEN2 kringle containing transmembrane protein 2
KRT86 keratin 86, type II
LOC730101 uncharacterized LOC730101
MALL mal, T-cell differentiation protein-like
MCC mutated in colorectal cancers
MGC12488
MPP3 membrane protein, palmitoylated 3 (MAGUK p55 subfamily member 3)
MVD mevalonate (diphospho) decarboxylase
MVP major vault protein
NDE1 nudE neurodevelopment protein 1
NDST2 N-deacetylase/N-sulfotransferase (heparan glucosaminyl) 2
NME5 NME/NM23 family member 5
NPY1R neuropeptide Y receptor Y1
NR1H2 nuclear receptor subfamily 1, group H, member 2
NR1H3 nuclear receptor subfamily 1, group H, member 3
P2RY6 pyrimidinergic receptor P2Y, G-protein coupled, 6
PIK3R2 phosphoinositide-3-kinase, regulatory subunit 2 (beta)
PLA2G10 phospholipase A2, group X
PLD3 phospholipase D family, member 3
PLEKHB1 pleckstrin homology domain containing, family B (evectins) member 1
PLEKHM2 pleckstrin homology domain containing, family M (with RUN domain) member 2
POLR3F polymerase (RNA) III (DNA directed) polypeptide F, 39 kDa
PPP1R3C protein phosphatase 1, regulatory subunit 3C
PRF1 perforin 1 (pore forming protein)
RAB3A RAB3A, member RAS oncogene family
RASSF8 Ras association (RalGDS/AF-6) domain family (N-terminal) member 8
RFTN1 raftlin, lipid raft linker 1
RIBC2 RIB43A domain with coiled-coils 2
RNF122 ring finger protein 122
RPL13P5 ribosomal protein L13 pseudogene 5
RPL23AP32 ribosomal protein L23a pseudogene 32
RPP14 ribonuclease P/MRP 14kDa subunit
SH2D4A SH2 domain containing 4A
SIL1 SIL1 nucleotide exchange factor
SLC25A23 solute carrier family 25 (mitochondrial carrier; phosphate carrier), member 23
SLC35C1 solute carrier family 35 (GDP-fucose transporter), member C1
SLC41A3 solute carrier family 41, member 3
SLC47A1 solute carrier family 47 (multidrug and toxin extrusion), member 1
SPANXC SPANX family, member C
SPINK5 serine peptidase inhibitor, Kazal type 5
SRD5A3 steroid 5 alpha-reductase 3
SRPX sushi-repeat containing protein, X-linked
SUV39H1 suppressor of variegation 3-9 homolog 1 (Drosophila)
TAF15 TAF15 RNA polymerase II, TATA box binding protein (TBP)-associated factor, 68kDa
TGFBRAP1 transforming growth factor, beta receptor associated protein 1
THBS3 thrombospondin 3
TRAF2 TNF receptor-associated factor 2
TRMT2A tRNA methyltransferase 2 homolog A (S. cerevisiae)
TRPS1 trichorhinophalangeal syndrome I
TTC33 tetratricopeptide repeat domain 33
USPL1 ubiquitin specific peptidase like 1
ZC3H3 zinc finger CCCH-type containing 3
ZNF226 zinc finger protein 226
ZNF350 zinc finger protein 350
ZNF862 zinc finger protein 862